Not logged inSelective blockade of Cav1.2 (α1C) versus Cav1.3 (α1D) L-type calcium channels by the black mamba toxin calciseptine
Mesirca, Pietro; Chemin, Jean; Barrere, Christian; Torre, Eleonora; Gallot, Laura; Monteil, Arnaud; Bidaud, Isabelle; Diochot, Sylvie; Lazdunski, Michel; Soong, Tuck Wah; Barrere-Lemaire, Stephanie; Mangoni, Matteo E.; Nargeot, Joel
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SaveChemical Synthesis, Proper Folding, Nav Channel Selectivity Profile and Analgesic Properties of the Spider Peptide Phlotoxin 1
Nicolas, Sebastien; Zoukimian, Claude; Bosmans, Frank; Montnach, Jerome; Diochot, Sylvie; Cuypers, Eva; De Waard, Stephan; Beroud, Remy; Mebs, Dietrich; Craik, David; Boturyn, Didier; Lazdunski, Michel; Tytgat, Jan; De Waard, Michel
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SaveAcute and long-term cardioprotective effects of the Traditional Chinese Medicine MLC901 against myocardial ischemia-reperfusion injury in mice
Vincent, Anne; Covinhes, Aurelie; Barrere, Christian; Gallot, Laura; Thoumala, Soulit; Piot, Christophe; Heurteaux, Catherine; Lazdunski, Michel; Nargeot, Joel; Barrere-Lemaire, Stephanie
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SaveRole of the TREK2 potassium channel in cold and warm thermosensation and in pain perception
Pereira, Vanessa; Busserolles, Jerome; Christin, Marine; Devilliers, Maily; Poupon, Laura; Legha, Wassim; Alloui, Abdelkrim; Aissouni, Youssef; Bourinet, Emmanuel; Lesage, Florian; Eschalier, Alain; Lazdunski, Michel; Noel, Jacques
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SaveActivation of TREK-1 by morphine results in analgesia without adverse side effects
Devilliers, Maily; Busserolles, Jerome; Lolignier, Stephane; Deval, Emmanuel; Pereira, Vanessa; Alloui, Abdelkrim; Christin, Marine; Mazet, Bruno; Delmas, Patrick; Noel, Jacques; Lazdunski, Michel; Eschalier, Alain
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SavePeripheral contribution of NGF and ASIC1a to colonic hypersensitivity in a rat model of irritable bowel syndrome
Matricon, J.; Muller, E.; Accarie, A.; Meleine, M.; Etienne, M.; Voilley, N.; Busserolles, J.; Eschalier, A.; Lazdunski, M.; Bourdu, S.; Gelot, A.; Ardid, D.
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SaveOxaliplatin-induced cold hypersensitivity is due to remodelling of ion channel expression in nociceptors
Descoeur, Juliette; Pereira, Vanessa; Pizzoccaro, Anne; Francois, Amaury; Ling, Bing; Maffre, Violette; Couette, Brigitte; Busserolles, Jerome; Courteix, Christine; Noel, Jacques; Lazdunski, Michel; Eschalier, Alain; Authier, Nicolas; Bourinet, Emmanuel
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SaveThe mechano-activated K+ channels TRAAK and TREK-1 control both warm and cold perception
Noel, Jacques; Zimmermann, Katharina; Busserolles, Jerome; Deval, Emanuel; Alloui, Abdelkrim; Diochot, Sylvie; Guy, Nicolas; Borsotto, Marc; Reeh, Peter; Eschalier, Alain; Lazdunski, Michel
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SaveASIC3, a sensor of acidic and primary inflammatory pain
Deval, Emmanuel; Noel, Jacques; Lay, Nadege; Alloui, Abdelkrim; Diochot, Sylvie; Friend, Valerie; Jodar, Martine; Lazdunski, Michel; Lingueglia, Eric
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SaveAltered acetylcholine, bradykinin and cutaneous pressure-induced vasodilation in mice lacking the TREK1 potassium channel: the endothelial link
Garry, Ambroise; Fromy, Berengere; Blondeau, Nicolas; Henrion, Daniel; Brau, Frederic; Gounon, Pierre; Guy, Nicolas; Heurteaux, Catherine; Lazdunski, Michel; Saumet, Jean Louis
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SaveAKAP150, a switch to convert mechano-, pH- and arachidonic acid- sensitive TREK K+ channels into open leak channels
Sandoz, Guillaume; Thummler, Susanne; Duprat, Fabrice; Feliciangeli, Sylvain; Vinh, Joelle; Escoubas, Pierre; Guy, Nicolas; Lazdunski, Michel; Lesage, Florian
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