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SaveDiscovery of a potent and orally bioavailable reversible TEAD inhibitor (R)-3-(5-(1-methyl-3-((4-(trifluoromethyl)phenyl) amino)-1H-pyrazol-4-yl)-1,3,4-oxadiazol-2-yl)-3-vinylpyrrolidin-2-one
Cao, Jianguo; Han, Xiaojun; Fischer, Kimberlee; Villanueva, Nicolas; Lee, Christian C.; Do, Quyen-Quyen; Li, Jiali; Pan, Wen-An; Sund, Summer; Pronk, Gijsbertus J.; Mochalkin, Igor; Huang, Peter; Bunker, Kevin; Orr, Suvi T. M.
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