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Paul R. Lockman

west virginia university school of pharmacy

48H-index
197Paper Count
9.1KCitation Count
Published Papers 79
Publication Date
PACM-13 ENDOTHELIN RECEPTOR ANTAGONISTS ENHANCE NERATINIB EFFICACY IN PRECLINICAL MODELS OF BREAST CANCER BRAIN METASTASIS THROUGH DEPRESSION OF BLOOD-BRAIN BARRIER EFFLUX TRANSPORT
err2026-08-07
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errGeoffrey Pecar; Cullen Wolford; Olivia Carpenter Milam; Austin Nestor; Dominic Gabriele; Joshua Applegate; Maxine Casto; Paul Lockman
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Correction: Characterization of blood-brain barrier L-arginine uptake using in situ brain perfusions in a female mouse model
err2026-07-19
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errOlivia C. Milam; Cullen P. Wolford; Geoffrey L. Pecar; Joshua J. Applegate; Maxine E. Casto; Dominic J. Gabriele; Austin S. Nestor; Paul R. Lockman
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Single Exposure to Low-Intensity Focused Ultrasound Causes Biphasic Opening of the Blood-Brain Barrier Through Secondary Mechanisms
err2025-01-08
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errArsiwala, Tasneem A.; Blethen, Kathryn E.; Wolford, Cullen P.; Pecar, Geoffrey L.; Panchal, Dhruvi M.; Kielkowski, Brooke N.; Wang, Peng; Ranjan, Manish; Carpenter, Jeffrey S.; Finomore, Victor; Rezai, Ali; Lockman, Paul R.
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Stromal PDGFRβ hyperactivation modulates the myeloid lineage in the brain metastatic microenvironment
err2024-02-01
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PREAI
errMossing, Alexis A.; Schiebel, Johnathon G.; Packard, Rebecca L.; Kumar, Amrendra; Steck, Sarah A.; Grabinski, Nathaniel S.; Thies, Katie A.; Wasik, Bri; Ariswala, Tasneem; Tozbikian, Gary; Godbout, Johnathan; Sizemore, Steven T.; Lockman, Paul R.; Vilgelm, Anna E.; Sizemore, Gina M.
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Study the efficacy of hypomethylating agent in treating regular and brain metastasized HER2-positive breast cancer
err2023-04-04
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PREAI
errLiu, Tuoen; Butler, Christopher; Donoughe, Kelsey; Forchette, Lauren; Sebastian, William; Szalai, Gabor; Lockman, Paul
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Vascular effects of Platelet-derived growth factor-B (PDGFB) in breast cancer metastasis to the brain
err2023-03-01
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PREAI
errShah, Sajita; Packard, Rebecca; Steck, Sarah; Mossing, Alexis; Ramamoorthy, Yalini; Thies, Katie; Didier, Alexander; Spehar, Jonathan; Richardson, Dillon; Arsiwala, Tasneem; Godbout, Jonathan; Sizemore, Steven; Lockman, Paul; Sizemore, Gina
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Blood-tumor barrier opening by MRI-guided transcranial focused ultrasound in a preclinical breast cancer brain metastasis model improves efficacy of combinatorial chemotherapy
err2023-02-10
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errArsiwala, Tasneem A.; Blethen, Kathryn E.; Wolford, Cullen P.; Panchal, Dhruvi M.; Sprowls, Samuel A.; Fladeland, Ross A.; Kielkowski, Brooke N.; Pritt, Trenton A.; Wang, Peng; Wilson, Olivia; Carpenter, Jeffrey S.; Finomore, Victor; Rezai, Ali; Lockman, Paul R.
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Effects of whole-brain radiation therapy on the blood-brain barrier in immunocompetent and immunocompromised mouse models
err2023-02-03
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errBlethen, K. E.; Sprowls, S. A.; Arsiwala, T. A.; Wolford, C. P.; Panchal, D. M.; Fladeland, R. A.; Glass, M. J.; Dykstra, L. P.; Kielkowski, B. N.; Blackburn, J. R.; Andrick, C. J.; Lockman, P. R.
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Characterization of passive permeability after low intensity focused ultrasound mediated blood-brain barrier disruption in a preclinical model
err2022-09-08
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errArsiwala, Tasneem A.; Sprowls, Samuel A.; Blethen, Kathryn E.; Fladeland, Ross A.; Wolford, Cullen P.; Kielkowski, Brooke N.; Glass, Morgan J.; Wang, Peng; Wilson, Olivia; Carpenter, Jeffrey S.; Ranjan, Manish; Finomore, Victor; Rezai, Ali; Lockman, Paul R.
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Circadian Influences on Chemotherapy Efficacy in a Mouse Model of Brain Metastases of Breast Cancer
err2021-12-09
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errWalker, William H.; Sprowls, Samuel A.; Bumgarner, Jacob R.; Liu, Jennifer A.; Melendez-Fernandez, O. Hecmarie; Walton, James C.; Lockman, Paul R.; DeVries, A. Courtney; Nelson, Randy J.
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Modulation of the blood-tumor barrier to enhance drug delivery and efficacy for brain metastases
err2021-11-27
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errBlethen, Kathryn E.; Arsiwala, Tasneem A.; Fladeland, Ross A.; Sprowls, Samuel A.; Panchal, Dhruvi M.; Adkins, Chris E.; Kielkowski, Brooke N.; Earp, Leland E.; Glass, Morgan J.; Pritt, Trenton A.; Cabuyao, Yssabela M.; Aulakh, Sonikpreet; Lockman, Paul R.
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Overcoming the acquired resistance to gefitinib in lung cancer brain metastasis in vitro and in vivo
err2021-08-28
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errLiu, Zhongwei; Shah, Neal; Marshall, Kent L.; Sprowls, Samuel A.; Saralkar, Pushkar; Mohammad, Afroz; Blethen, Kathryn E.; Arsiwala, Tasneem A.; Fladeland, Ross; Lockman, Paul R.; Gao, Weimin
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Ultrasound-mediated disruption of the blood tumor barrier for improved therapeutic delivery
err2021-07-01
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errArsiwala, T. A.; Sprowls, S. A.; Blethen, K. E.; Adkins, C. E.; Saralkar, P. A.; Fladeland, R. A.; Pentz, W.; Gabriele, A.; Kielkowski, B.; Mehta, R. I.; Wang, P.; Carpenter, J. S.; Ranjan, M.; Najib, U.; Rezai, A. R.; Lockman, P. R.
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Nanoparticles as a Tool in Neuro-Oncology Theranostics
err2021-06-24
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errKlein, Andrea L.; Nugent, Grant; Cavendish, John; Geldenhuys, Werner J.; Sriram, Krishnan; Porter, Dale; Fladeland, Ross; Lockman, Paul R.; Sherman, Jonathan H.
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A Review of Mathematics Determining Solute Uptake at the Blood-Brain Barrier in Normal and Pathological Conditions
err2021-05-19
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errSprowls, Samuel A.; Saralkar, Pushkar; Arsiwala, Tasneem; Adkins, Christopher E.; Blethen, Kathryn E.; Pizzuti, Vincenzo J.; Shah, Neal; Fladeland, Ross; Lockman, Paul R.
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Blood-Brain Barrier Opening with MRI-guided Focused Ultrasound Elicits Meningeal Venous Permeability in Humans with Early Alzheimer Disease
errRADIOLOGY
IF15.2
err2021-03-01
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errMehta, Rashi, I; Carpenter, Jeffrey S.; Mehta, Rupal, I; Haut, Marc W.; Ranjan, Manish; Najib, Umer; Lockman, Paul; Wang, Peng; D'haese, Pierre-Francois; Rezai, Ali R.
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DNA Methylation of the Keratin 18 Gene Regulates Brain Metastasis of Triple Negative Breast Cancer
err2020-04-15
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errLiu, Tuoen; Kohler, William; Wolff, Benjamin; Butler, Christopher; Szalai, Gabor; Straight, Benjamin; Lockman, Paul
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Drug resistance occurred in a newly characterized preclinical model of lung cancer brain metastasis
err2020-04-07
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errShah, Neal; Liu, Zhongwei; Tallman, Rachel M.; Mohammad, Afroz; Sprowls, Samuel A.; Saralkar, Pushkar A.; Vickers, Schuyler D.; Pinti, Mark V.; Gao, Weimin; Lockman, Paul R.
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MiR-34a Interacts with Cytochrome c and Shapes Stroke Outcomes
err2020-02-24
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errHu, Heng; Hone, Emily A.; Provencher, Edward A. P.; Sprowls, Samuel A.; Farooqi, Imran; Corbin, Deborah R.; Sarkar, Saumyendra N.; Hollander, John M.; Lockman, Paul R.; Simpkins, James W.; Ren, Xuefang
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