arrow
Back
C

Christoph Klenk

university of zurich

18H-index
44Paper Count
1.3KCitation Count
Published Papers 24
Publication Date
Docking of virtual libraries identifies small-molecule agonists of neurotensin receptors with analgesic activity
err2026-07-22
err0
errOAAI
errNicolas Panel; Duy Duc Vo; Harald Hübner; Mattia Deluigi; Szymon Pach; Félix Bélair; Dorothee Weikert; Christoph Klenk; Mark Hilge; Niharika Shiva; Isabelle Brochu; Jean-Michel Longpré; Frida Bällgren; Aljona Saleh; Huabin Hu; Jon Kapla; Stefanie Kampen; Israel Cabeza de Vaca; Jan Kihlberg; Nina Wettschureck; Philippe Sarret; Andreas Plückthun; Peter Gmeiner; Jens Carlsson
errShare
errSave
ADAM19 cleaves the PTH receptor and associates with brachydactyly type E
err2024-02-08
err1
errOAAI
errAydin, Atakan; Klenk, Christoph; Nemec, Katarina; Isbilir, Ali; Martin, Lisa M.; Zauber, Henrik; Rrustemi, Trendelina; Toka, Hakan R.; Schuster, Herbert; Gong, Maolian; Stricker, Sigmar; Bock, Andreas; Baehring, Sylvia; Selbach, Matthias; Lohse, Martin J.; Luft, Friedrich C.
errShare
errSave
A Vaccinia-based system for directed evolution of GPCRs in mammalian cells
err2023-03-30
err3
errOAAI
errKlenk, Christoph; Scrivens, Maria; Niederer, Anina; Shi, Shuying; Mueller, Loretta; Gersz, Elaine; Zauderer, Maurice; Smith, Ernest S.; Strohner, Ralf; Pluckthun, Andreas
errShare
errSave
Crystal structure of the α1B-adrenergic receptor reveals molecular determinants of selective ligand recognition
err2022-01-19
err19
errOAAI
errDeluigi, Mattia; Morstein, Lena; Schuster, Matthias; Klenk, Christoph; Merklinger, Lisa; Cridge, Riley R.; de Zhang, Lazarus A.; Klipp, Alexander; Vacca, Santiago; Vaid, Tasneem M.; Mittl, Peer R. E.; Egloff, Pascal; Eberle, Stefanie A.; Zerbe, Oliver; Chalmers, David K.; Scott, Daniel J.; Pluckthun, Andreas
errShare
errSave
Engineering of Challenging G Protein-Coupled Receptors for Structure Determination and Biophysical Studies
err2021-03-08
err5
errOAAI
errWaltenspuhl, Yann; Ehrenmann, Janosch; Klenk, Christoph; Pluckthun, Andreas
errShare
errSave
Cryo-EM structure of an activated GPCR-G protein complex in lipid nanodiscs
err2021-02-25
err73
errOAAI
errZhang, Meng; Gui, Miao; Wang, Zi-Fu; Gorgulla, Christoph; Yu, James J.; Wu, Hao; Sun, Zhen-yu J.; Klenk, Christoph; Merklinger, Lisa; Morstein, Lena; Hagn, Franz; Pluckthun, Andreas; Brown, Alan; Nasr, Mahmoud L.; Wagner, Gerhard
errShare
errSave
Complexes of the neurotensin receptor 1 with small-molecule ligands reveal structural determinants of full, partial, and inverse agonism
err2021-01-29
err33
errOAAI
errDeluigi, Mattia; Klipp, Alexander; Klenk, Christoph; Merklinger, Lisa; Eberle, Stefanie A.; Morstein, Lena; Heine, Philipp; Mittl, Peer R. E.; Ernst, Patrick; Kamenecka, Theodore M.; He, Yuanjun; Vacca, Santiago; Egloff, Pascal; Honegger, Annemarie; Pluckthun, Andreas
errShare
errSave
New views into class B GPCRs from the crystal structure of PTH1R
err2019-11-18
err5
errOAAI
errEhrenmann, Janosch; Schoeppe, Jendrik; Klenk, Christoph; Plueckthun, Andreas
errShare
errSave
Crystal structures of the human neurokinin 1 receptor in complex with clinically used antagonists
err2019-01-03
err60
errOAAI
errSchoeppe, Jendrik; Ehrenmann, Janosch; Klenk, Christoph; Rucktooa, Prakash; Schuetz, Marco; Dore, Andrew S.; Plueckthun, Andreas
errShare
errSave
High-resolution crystal structure of parathyroid hormone 1 receptor in complex with a peptide agonist
err2018-11-19
err91
PREAI
errEhrenmann, Janosch; Schoeppe, Jendrik; Klenk, Christoph; Rappas, Mathieu; Kummer, Lutz; Dore, Andrew S.; Plueckthun, Andreas
errShare
errSave
Directed evolution of G protein-coupled receptors in yeast for higher functional production in eukaryotic expression hosts
err2016-02-25
err62
errOAAI
errSchuetz, Marco; Schoeppe, Jendrik; Sedlak, Erik; Hillenbrand, Matthias; Nagy-Davidescu, Gabriela; Ehrenmann, Janosch; Klenk, Christoph; Egloff, Pascal; Kummer, Lutz; Plueckthun, Andreas
errShare
errSave
A generic selection system for improved expression and thermostability of G protein-coupled receptors by directed evolution
err2016-02-18
err29
errOAAI
errKlenk, Christoph; Ehrenmann, Janosch; Schuetz, Marco; Plueckthun, Andreas
errShare
errSave
Sumoylation of Influenza A Virus Nucleoprotein Is Essential for Intracellular Trafficking and Virus Growth
err2014-08-15
err63
errOAAI
errHan, Qinglin; Chang, Chong; Li, Li; Klenk, Christoph; Cheng, Jinke; Chen, Yixin; Xia, Ningshao; Shu, Yuelong; Chen, Ze; Gabriel, Guelsah; Sun, Bing; Xu, Ke
errShare
errSave
Structure of signaling-competent neurotensin receptor 1 obtained by directed evolution in Escherichia coli
err2014-01-22
err199
errOAAI
errEgloff, Pascal; Hillenbrand, Matthias; Klenk, Christoph; Batyuk, Alexander; Heine, Philipp; Balada, Stefanie; Schlinkmann, Karola M.; Scott, Daniel J.; Schuetz, Marco; Plueckthun, Andreas
errShare
errSave
The Guanine Nucleotide Exchange Factor Vav2 Is a Negative Regulator of Parathyroid Hormone Receptor/Gq Signaling
err2012-08-01
err1
errOAAI
errEmami-Nemini, Alexander; Gohla, Antje; Urlaub, Henning; Lohse, Martin J.; Klenk, Christoph
errShare
errSave
Modification of Nonstructural Protein 1 of Influenza A Virus by SUMO1
err2011-01-15
err92
errOAAI
errXu, Ke; Klenk, Christoph; Liu, Bin; Keiner, Bjoern; Cheng, Jinke; Zheng, Bo-Jian; Li, Li; Han, Qinglin; Wang, Chen; Li, Tianxian; Chen, Ze; Shu, Yuelong; Liu, Jinhua; Klenk, Hans-Dieter; Sun, Bing
errShare
errSave
Formation of a Ternary Complex among NHERF1, β-Arrestin, and Parathyroid Hormone Receptor
err2010-09-01
err33
errOAAI
errKlenk, Christoph; Vetter, Thorsten; Zuern, Alexander; Vilardaga, Jean-Pierre; Friedman, Peter A.; Wang, Bin; Lohse, Martin J.
errShare
errSave
Immunohistochemical identification of the PTHR1 parathyroid hormone receptor in normal and neoplastic human tissues
err2010-05-01
err61
PREAI
errLupp, Amelie; Klenk, Christoph; Roecken, Christoph; Evert, Matthias; Mawrin, Christian; Schulz, Stefan
errShare
errSave
Site-Specific, Orthogonal Labeling of Proteins in Intact Cells with Two Small Biarsenical Fluorophores
err2010-04-29
err46
PREAI
errZuern, Alexander; Klenk, Christoph; Zabel, Ulrike; Reiner, Susanne; Lohse, Martin J.; Hoffmann, Carsten
errShare
errSave