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Charles Sawyers

Memorial Sloan Kettering Cancer Center

8H-index
30Paper Count
4.3KCitation Count
Published Papers 189
Publication Date
NSD2 targeting reverses plasticity and drug resistance in prostate cancer
errNature
IF48.5
err2025-11-26
err0
errOAAI
errJia J. Li; Alessandro Vasciaveo; Dimitris Karagiannis; Zhen Sun; Kristjan H. Gretarsson; Xiao Chen; Ouathek Ouerfelli; Fabio Socciarelli; Ziv Frankenstein; Hanyang Dong; Min Zou; Wei Yuan; Guangli Yang; Gabriel M. Aizenman; Tania Pannellini; Xinjing Xu; Himisha Beltran; Yu Chen; Kevin Gardner; Brian D. Robinson; Johann de Bono; Or Gozani; Cory Abate-Shen; Mark A. Rubin; Massimo Loda; Charles L. Sawyers; Andrea Califano; Chao Lu; Michael M. Shen
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ERG-driven prostate cancer initiation is cell-context dependent and requires KMT2A and DOT1L
err2025-08-26
err0
errOAAI
errWeiran Feng; Erik Ladewig; Matthew Lange; Nazifa Salsabeel; Huiyong Zhao; Young Sun Lee; Anuradha Gopalan; Hanzhi Luo; Wenfei Kang; Ning Fan; Eric Rosiek; Elisa de Stanchina; Yu Chen; Brett S. Carver; Christina S. Leslie; Charles L. Sawyers
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The neuroendocrine transition in prostate cancer is dynamic and dependent on ASCL1
err2024-10-11
err1
errOAAI
errRomero, Rodrigo; Chu, Tinyi; Robles, Tania J. Gonzalez; Smith, Perianne; Xie, Yubin; Kaur, Harmanpreet; Yoder, Sara; Zhao, Huiyong; Mao, Chenyi; Kang, Wenfei; Pulina, Maria V.; Lawrence, Kayla E.; Gopalan, Anuradha; Zaidi, Samir; Yoo, Kwangmin; Choi, Jungmin; Fan, Ning; Gerstner, Olivia; Karthaus, Wouter R.; Destanchina, Elisa; Ruggles, Kelly V.; Westcott, Peter M. K.; Chaligne, Ronan; Pe'er, Dana; Sawyers, Charles L.
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Single- cell analysis of treatment- resistant prostate cancer: Implications of cell state changes for cell surface antigen- targeted therapies
err2024-07-05
err4
errOAAI
errZaidi, Samir; Park, Jooyoung; Chan, Joseph M.; Roudier, Martine P.; Zhao, Jimmy L.; Gopalan, Anuradha; Wadosky, Kristine M.; Patel, Radhika A.; Sayar, Erolcan; Karthaus, Wouter R.; Kates, D. Henry; Chaudhary, Ojasvi; Xu, Tianhao; Masilionis, Ignas; Mazutis, Linas; Chaligne, Ronan; Obradovic, Aleksandar; Linkov, Irina; Barlas, Afsar; Jungbluth, Achim A.; Rekhtman, Natasha; Silber, Joachim; Manova-Todorova, Katia; Watson, Philip A.; True, Lawrence D.; Morrissey, Colm; Scher, Howard I.; Rathkopf, Dana E.; Morris, Michael J.; Goodrich, David W.; Choi, Jungmin; Nelson, Peter S.; Haffner, Michael C.; Sawyers, Charles L.
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Assessment of TROP2, CEACAM5 and DLL3 in metastatic prostate cancer: Expression landscape and molecular correlates
err2024-05-17
err3
errOAAI
errAjkunic, Azra; Sayar, Erolcan; Roudier, Martine P.; Patel, Radhika A.; Coleman, Ilsa M.; De Sarkar, Navonil; Hanratty, Brian; Adil, Mohamed; Zhao, Jimmy; Zaidi, Samir; True, Lawrence D.; Sperger, Jamie M.; Cheng, Heather H.; Yu, Evan Y.; Montgomery, Robert B.; Hawley, Jessica E.; Ha, Gavin; Persse, Thomas; Galipeau, Patricia; Lee, John K.; Harmon, Stephanie A.; Corey, Eva; Lang, Joshua M.; Sawyers, Charles L.; Morrissey, Colm; Schweizer, Michael T.; Gulati, Roman; Nelson, Peter S.; Haffner, Michael C.
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ROLE OF TUMOR MICROENVIRONMENT DERIVED NRG1 IN ANDROGEN RESISTANCE: IMPLICATIONS FOR A NOVEL PROSTATE CANCER TREATMENT STRATEGY
err2024-05-01
err0
PREAI
errShinder, Brian; Mao, Ninghui; Zhang, Zeda; Sawyers, Charles L.; Carver, Brett S.
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The histone methyltransferase KMT2D mediates subtype-specific transcriptional regulation and therapeutic response in prostate cancer
err2024-03-22
err0
PREAI
errKittane, Srushti; Ladewig, Erik; Li, Taibo; Love, Jillian; Arruabarrena-Aristorena, Amaia; Guo, Xinyu; Sallaku, Mirna; Garcia-Martinez, Liliana; Blawski, Ryan; Sanz, Javier Carmona; Simpkins, Christopher; Chen, Wanlu; Vokshi, Bujamin; Zhao, Peihua; Kelkar, Nachiket; Baldino, Laura; Kalemi, Ingrid; Castel, Pau; Cocco, Emiliano; Morey, Lluis; Sawyers, Charles; Ji, Hongkai; Scaltriti, Maurizio; Battle, Alexis; Leslie, Christina; Eneda, Wouter Karthaus
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CDC7 inhibition prevents neuroendocrine transformation in the lung and prostate through MYC degradation
err2024-03-22
err0
PREAI
errQuintanal-Villalonga, Alvaro; Uddin, Fathema; Kawasaki, Kenta; Redin, Esther; Durani, Vidushi; Sabet, Amin; Karthaus, Wouter; Zhan, Yingqian A.; Zaidi, Samir; Shaffer, Moniquetta; Sridhar, Harsha; Qiu, Juan; Manoj, Parvathy; De Stanchina, Elisa; Haffner, Michael C.; Sawyers, Charles L.; Rudin, Charles M.
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Erg-driven prostate cancer emerges from a basal subset of cells with luminal transcriptomic features
err2024-03-22
err0
PREAI
errLadewig, Erik; Feng, Weiran; Leslie, Christina; Sawyers, Charles
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Strategies to decrease inequalities in cancer therapeutics, care and preventionProceedings on a conference organized by the Pontifical Academy of Sciences and the European Academy of Cancer Sciences, Vatican City, February 23-24, 2023
err2024-01-22
err11
errOAAI
errRingborg, Ulrik; von Braun, Joachim; Celis, Julio; Baumann, Michael; Berns, Anton; Eggermont, Alexander; Heard, Edith; Heitor, Manuel; Chandy, Mammen; Chen, Chien-Jen; Costa, Alberto; De Lorenzo, Francesco; De Robertis, Edward M.; Dubee, Frederick Charles; Ernberg, Ingemar; Gabriel, Mariya; Helland, Aslaug; Henrique, Rui; Joensson, Bengt; Kallioniemi, Olli; Korbel, Jan; Krause, Mechthild; Lowy, Douglas R.; Michielin, Olivier; Nagy, Peter; Oberst, Simon; Paglia, Vincenzo; Parker, M. Iqbal; Ryan, Kevin; Sawyers, Charles L.; Schuz, Joachim; Silkaitis, Katherine; Solary, Eric; Thomas, David; Turkson, Peter; Weiderpass, Elisabete; Yang, Huanming
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CDC7 inhibition constrains lineage plasticity and prevents resistance and neuroendocrine transformation in the lung and prostate
err2023-10-01
err0
errOAAI
errQuintanal-Villalonga, A.; Zaidi, S.; Karthaus, W. R.; Zhan, Y. A.; Shafer, M.; Qiu, J.; de Stanchina, E.; Haffner, M. C.; Sawyers, C. L.; Rudin, C. M.
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Addressing racial and ethnic disparities in AACR project GENIE
err2023-08-31
err2
errOAAI
errSweeney, Shawn M.; Lavery, Jessica A.; Fuchs, Hannah E.; Lee, Jocelyn A.; Brown, Samantha; Panageas, Katherine S.; Sawyers, Charles L.; Bedard, Philippe L.
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Exportin 1 inhibition prevents neuroendocrine transformation through SOX2 down-regulation in lung and prostate cancers
err2023-08-02
err17
PREAI
errQuintanal-Villalonga, Alvaro; Durani, Vidushi; Sabet, Amin; Redin, Esther; Kawasaki, Kenta; Shafer, Moniquetta; Karthaus, Wouter R.; Zaidi, Samir; Zhan, Yingqian A.; Manoj, Parvathy; Sridhar, Harsha; Shah, Nisargbhai S.; Chow, Andrew; Bhanot, Umesh K.; Linkov, Irina; Asher, Marina; Yu, Helena A.; Qiu, Juan; de Stanchina, Elisa; Patel, Radhika A.; Morrissey, Colm; Haffner, Michael C.; Koche, Richard P.; Sawyers, Charles L.; Rudin, Charles M.
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Chromatin regulation of transcriptional enhancers and cell fate by the Sotos syndrome gene NSD1
err2023-07-01
err9
errOAAI
errSun, Zhen; Lin, Yuan; Islam, Mohammed T.; Koche, Richard; Hedehus, Lin; Liu, Dingyu; Huang, Chang; Vierbuchen, Thomas; Sawyers, Charles L.; Helin, Kristian
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ERG-driven luminal prostate cancers emerge from Ck5+/Nkx3.1+basal cells
err2023-06-02
err0
PREAI
errFeng, Weiran; Ladewig, Erik; Salsabeel, Nazifa; Zhao, Huiyong; Lee, Young Sun; Gopalan, Anuradha; Luo, Hanzhi; Kang, Wenfei; Fan, Ning; Rosiek, Eric; Masilionis, Ignas; Manova-Todorova, Katia; Chaligne, Ronan; de Stanchina, Elisa; Carver, Brett S.; Chen, Yu; Gao, Dong; Leslie, Christina S.; Sawyers, Charles L.
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Mutations in FOXA1 alter chromatin remodeling and cell fate in prostate organoids
err2023-04-04
err0
PREAI
errLadewig, Erik; Nazir, Abbas; Leslie, Christina; Sawyers, Charles
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Macrophages promote anti-androgen resistance in prostate cancer bone disease
err2023-02-07
err33
errOAAI
errLi, Xue-Feng; Selli, Cigdem; Zhou, Han-Lin; Cao, Jian; Wu, Shuiqing; Ma, Ruo-Yu; Lu, Ye; Zhang, Cheng-Bin; Xun, Bijie; Lam, Alyson D.; Pang, Xiao-Cong; Fernando, Anu; Zhang, Zeda; Unciti-Broceta, Asier; Carragher, Neil O.; Ramachandran, Prakash; Henderson, Neil C.; Sun, Ling-Ling; Hu, Hai-Yan; Li, Gui-Bo; Sawyers, Charles; Qian, Bin-Zhi
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