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Discovery of A-910, a Highly Potent and Orally Bioavailable Dual MerTK/Axl-Selective Tyrosine Kinase Inhibitor Yu, Yiyun; Jang, Miyeon; Miyashiro, Julie; Clark, Richard F.; Zhu, Gui-Dong; Gong, Jane; Dai, Yujia; Frey, Robin R.; Penning, Thomas D.; Kim, Hadong; Lee, Hyung Ki; Kim, Jin Kwan; Ryu, Ki Moon; Park, Seong Jin; Yoon, Taeyoung; Li, Tao; Kurnick, Matthew D.; Kapecki, Nicolas J.; Li, Leiming; Gorman, Jacob V.; Montgomery, Debra A.; Manaves, Vlasios; Bromberg, Kenneth D.; Doktor, Stella Z.; Thakur, Ashish; Wang, Jin; Smith, Heath A.; Buchanan, Fritz G.; Ferguson, Debra C.; Torrent, Maricel; Jakob, Clarissa G.; Qiu, Wei; Upadhyay, Anup K.; Martin, Ruth L.; Lai, Albert; Michaelides, Michael R. 分享 收藏
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Multiple evaluations, risk assessment, and source identification of heavy metals in surface water and sediment of the Golmud River, northeastern Qinghai-Tibet Plateau, China Cai, Na; Li, Leiming; Zhu, Haixia; Chen, Liang; Li, Shanping; Meng, Fanwei; Zhang, Xiying 分享 收藏
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Essential role of the Crk family-dosage in DiGeorge-like anomaly and metabolic homeostasis Imamoto, Akira; Ki, Sewon; Li, Leiming; Iwamoto, Kazunari; Maruthamuthu, Venkat; Devany, John; Lu, Ocean; Kanazawa, Tomomi; Zhang, Suxiang; Yamada, Takuji; Hirayama, Akiyoshi; Fukuda, Shinji; Suzuki, Yutaka; Okada, Mariko 分享 收藏
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Discovery of N-(4-(2,4-Difluorophenoxy)-3-(6-methyl-7-oxo-6,7-dihydro-1H-pyrrolo[2,3-c]pyridin-4-yl)phenyl)ethanesulfonamide (ABBV-075/Mivebresib), a Potent and Orally Available Bromodomain and Extraterminal Domain (BET) Family Bromodomain Inhibitor McDaniel, Keith F.; Wang, Le; Soltwedel, Todd; Fidanze, Steven D.; Hasvold, Lisa A.; Liu, Dachun; Mantei, Robert A.; Pratt, John K.; Sheppard, George S.; Bui, Mai H.; Faivre, Emily J.; Huang, Xiaoli; Li, Leiming; Lin, Xiaoyu; Wang, Rongqi; Warder, Scott E.; Wilcox, Denise; Albert, Daniel H.; Magoc, Terrance J.; Rajaraman, Ganesh; Park, Chang H.; Hutchins, Charles W.; Shen, Jianwei J.; Edalji, Rohinton P.; Sun, Chaohong C.; Martin, Ruth; Gao, Wenqing; Wong, Shekman; Fang, Guowei; Elmore, Steven W.; Shen, Yu; Kati, Warren M. 分享 收藏
Preclinical Characterization of BET Family Bromodomain Inhibitor ABBV-075 Suggests Combination Therapeutic Strategies Bui, Mai H.; Lin, Xiaoyu; Albert, Daniel H.; Li, Leiming; Lam, Lloyd T.; Faivre, Emily J.; Warder, Scott E.; Huang, Xiaoli; Wilcox, Denise; Donawho, Cherrie K.; Sheppard, George S.; Wang, Le; Fidanze, Steve; Pratt, John K.; Liu, Dachun; Hasvold, Lisa; Uziel, Tamar; Lu, Xin; Kohlhapp, Fred; Fang, Guowei; Elmore, Steven W.; Rosenberg, Saul H.; McDaniel, Keith F.; Kati, Warren M.; Shen, Yu 分享 收藏
Fragment-Based, Structure-Enabled Discovery of Novel Pyridones and Pyridone Macrocycles as Potent Bromodomain and Extra-Terminal Domain (BET) Family Bromodomain Inhibitors Wang, Le; Pratt, John K.; Soltwedel, Todd; Sheppard, George S.; Fidanze, Steven D.; Liu, Dachun; Hasvold, Lisa A.; Mantei, Robert A.; Holms, James H.; McClellan, William J.; Wendt, Michael D.; Wada, Carol; Frey, Robin; Hansen, T. Matthew; Hubbard, Robert; Park, Chang H.; Li, Leiming; Magoc, Terrance J.; Albert, Daniel H.; Lin, Xiaoyu; Warder, Scott E.; Kovar, Peter; Huang, Xiaoli; Wilcox, Denise; Wang, Rongqi; Rajaraman, Ganesh; Petros, Andrew M.; Hutchins, Charles W.; Panchal, Sanjay C.; Sun, Chaohong; Elmore, Steven W.; Shen, Yu; Kati, Warren M.; McDaniel, Keith F. 分享 收藏