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收藏A structure-based framework for selective inhibitor design and optimization基于结构的框架用于选择性抑制剂的研发与优化
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收藏Design, Synthesis, and Pharmacodynamic Evaluation of Highly Selective PARP1 Inhibitors with Brain Penetrance设计、合成及具有脑渗透性的高选择性PARP1抑制剂的药效学评价
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收藏Discovery of Potent, Specific, and Orally Available NLRP3 Inflammasome Inhibitors Based on Pyridazine Scaffolds for the Treatment of Septic Shock and Peritonitis
Fu, Zhiyuan; Duan, Yangqin; Pei, Heying; Zou, Yurong; Tang, Minghai; Chen, Yong; Yang, Tao; Ma, Ziyan; Yan, Wei; Su, Kaiyue; Cai, Xiaoying; Guo, Tao; Teng, Yaxin; Jia, Tao; Chen, Lijuan
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收藏Design, Synthesis, and Biological Evaluation of 5-Amino-4-fluoro-1H-benzo[d]imidazole-6-carboxamide Derivatives as Novel and Potential MEK/RAF Complex Inhibitors Based on the Clamp Strategy
Wang, Peng; Yuan, Yongting; Yang, Tao; Zou, Yurong; Tang, Minghai; Ma, Ziyan; Bo, Weichen; Qin, Songhui; Chen, Yong; Guo, Tao; Guo, Zhongning; Yang, Jianhong; Xiang, Mingli; Chen, Lijuan
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