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Damian W. Young

baylor college of medicine

24H指数
96论文数
1.9K被引数
收录论文 48
发表时间
A small molecule inhibits Ebola virus entry through glycoprotein stabilization小分子通过糖蛋白稳定化抑制埃博拉病毒进入
err2026-09-01
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errOAAI
errFan Bu; Gang Ye; Kiran L. Sharma; Bruno La Rosa; Murugesan Palaniappan; Martin M. Matzuk; Damian W. Young; Hailey Turner-Hubbard; Kimberly Morsheimer; Callum Owen; Katalin Toth; Michael Cameron; Robert Davey; Srinivas Chamakuri; Peter Dosa; Fang Li
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Discovery of a novel small molecule degrader of wild type and mutant estrogen receptors using DNA encoded libraries利用DNA编码化合物库发现一种新型小分子降解剂,可靶向野生型和突变型雌激素受体
err2025-11-12
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errOAAI
errAnil Kumar Devakrishnan; Chandrashekhar Madasu; Yong Wang; Ramkumar Modukuri; Kurt M. Bohren; Kevin R. MacKenzie; Damian W. Young; Suzanne A. W. Fuqua; Martin M. Matzuk; Murugesan Palaniappan
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MYC-Targeting PROTACs Lead to Bimodal Degradation and N-Terminal Truncation
err2025-03-01
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PREAI
errBoyd, Shelton R.; Chamakuri, Srinivas; Trostle, Alexander J.; Chen, Hu; Liu, Zhandong; Jian, Antrix; Wang, Jian; Malovannaya, Anna; Young, Damian W.
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Discovery of highly potent and ALK2/ALK 1 selective kinase inhibitors using DNA- encoded chemistry technology
err2024-11-14
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errOAAI
errJimmidi, Ravikumar; Monsivais, Diana; Ta, Hai Minh; Sharma, Kiran L.; Bohren, Kurt M.; Chamakuri, Srinivas; Liao, Zian; Li, Feng; Hakenjos, John M.; Li, Jian - Yuan; Mishina, Yuji; Pan, Haichun; Qin, Xuan; Robers, Matthew B.; Sankaran, Banumathi; Tan, Zhi; Tang, Suni; Vasquez, Yasmin M.; Wilkinson, Jennifer; Young, Damian W.; Palmer, Stephen S.; Mackenzie, Kevin R.; Kim, Choel; Matzuk, Martin M.
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Identification of potent pan- ephrin receptor kinase inhibitors using DNA- encoded chemistry technology
err2024-05-03
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PREAI
errMadasu, Chandrashekhar; Liao, Zian; Parks, Sydney E.; Sharma, Kiran L.; Bohren, Kurt M.; Ye, Qiuji; Li, Feng; Palaniappan, Murugesan; Tan, Zhi; Yuan, Fei; Creighton, Chad J.; Tang, Suni; Masand, Ramya P.; Guan, Xiaoming; Young, Damian W.; Monsivais, Diana; Matzuk, Martin M.
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CYP3A Mediates an Unusual C(sp2)-C(sp3) Bond Cleavage via Ipso-Addition of Oxygen in Drug Metabolism
err2024-04-29
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errOAAI
errQin, Xuan; Wang, Yong; Ye, Qiuji; Hakenjos, John M.; Wang, Jin; Teng, Mingxing; Guo, Lei; Tan, Zhi; Young, Damian W.; Mackenzie, Kevin R.; Li, Feng
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Expanding Complex Morpholines Using Systematic Chemical Diversity
err2024-03-20
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PREAI
errTang, Sunny Ann; Fults, Afton; Boyd, Shelton R.; Gattu, Nikhil; Tran, Kevin A.; Fan, Jiayi; Mackenzie, Kevin R.; Palzkill, Timothy; Young, Damian W.; Chamakuri, Srinivas
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Chemical Catalysis Guides Structural Identification for the Major In Vivo Metabolite of the BET Inhibitor JQ1
err2024-01-02
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errOAAI
errHolmes, Secondra; Jain, Prashi; Rodriguez, Kenneth Guzman; Williams, Jade; Yu, Zhifeng; Cerda-Smith, Christian; Samuel, Errol L. G.; Campbell, James; Hakenjos, John Michael; Monsivais, Diana; Li, Feng; Chamakuri, Srinivas; Matzuk, Martin M.; Santini, Conrad; Mackenzie, Kevin R.; Young, Damian W.
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Heterocyclic Merging of Stereochemically Diverse Chiral Piperazines and Morpholines with Indazoles
err2023-08-29
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errOAAI
errViveki, Amol B.; Mansfield, Timothy M.; Tran, Kevin A.; Lenkeit, Evan; Mackenzie, Kevin R.; Young, Damian W.; Chamakuri, Srinivas
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DNA-encoded chemical libraries yield non-covalent and non-peptidic SARS-CoV-2 main protease inhibitors
err2023-08-04
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errOAAI
errJimmidi, Ravikumar; Chamakuri, Srinivas; Lu, Shuo; Ucisik, Melek Nihan; Chen, Peng-Jen; Bohren, Kurt M.; Moghadasi, Seyed Arad; Versteeg, Leroy; Nnabuife, Christina; Li, Jian-Yuan; Qin, Xuan; Chen, Ying-Chu; Faver, John C.; Nyshadham, Pranavanand; Sharma, Kiran L.; Sankaran, Banumathi; Judge, Allison; Yu, Zhifeng; Li, Feng; Pollet, Jeroen; Harris, Reuben S.; Matzuk, Martin M.; Palzkill, Timothy; Young, Damian W.
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SPOP loss places the prostate luminal epithelial cells at a selective disadvantage
err2023-06-02
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PREAI
errRizwan, Kinza; Skapura, Darlene; Mason, Cammy; Coarfa, Cristian; Mitsiades, Nicholas; Young, Damian; Kaochar, Salma
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SPOP: An essential gene for normal and prostate tumor cells
err2023-04-04
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PREAI
errRizwan, Kinza; Skapura, Darlene; Mason, Cammy; Coarfa, Cristian; Mitsiades, Nicholas; Young, Damian; Kaochar, Salma
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Discovery and Development of Next-Generation Estrogen Receptor Mutant Inhibitors using DNA-Encoded Chemical Library Screening
err2023-03-01
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PREAI
errPalaniappan, Murugesan; Bohren, Kurt M.; Wang, Yong; Young, Damian W.; Fuqua, Suzanne A.; Matzuk, Martin M.
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The roles of Cyp1a2 and Cyp2d in pharmacokinetic profiles of serotonin and norepinephrine reuptake inhibitor duloxetine and its metabolites in mice
err2023-02-01
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errOAAI
errQin, Xuan; Xie, Cen; Hakenjos, John M.; MacKenzie, Kevin R.; Boyd, Shelton R.; Barzi, Mercedes; Bissig, Karl-Dimiter; Young, Damian W.; Li, Feng
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Discovery of Highly Potent and BMPR2-Selective Kinase Inhibitors Using DNA-Encoded Chemical Library Screening
err2023-01-31
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errOAAI
errModukuri, Ram K.; Monsivais, Diana; Li, Feng; Palaniappan, Murugesan; Bohren, Kurt M.; Tan, Zhi; Ku, Angela F.; Wang, Yong; Madasu, Chandrashekhar; Li, Jian-Yuan; Tang, Suni; Miklossy, Gabriella; Palmer, Stephen S.; Young, Damian W.; Matzuk, Martin M.
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Advancing ASMS with LC-MS/MS for the discovery of novel PDCL2 ligands from DNA-encoded chemical library selections
err2022-11-02
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errYe, Qiuji; Belabed, Hassane; Wang, Yong; Yu, Zhifeng; Palaniappan, Murugesan; Li, Jian-Yuan; Kalovidouris, Stacey A.; MacKenzie, Kevin R.; Teng, Mingxing; Young, Damian W.; Fujihara, Yoshitaka; Matzuk, Martin M.
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The Pursuit of Enzyme Activation: A Snapshot of the Gold Rush
err2022-10-20
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PREAI
errTeng, Mingxing; Young, Damian W.; Tan, Zhi
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