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Discovery of highly potent and ALK2/ALK 1 selective kinase inhibitors using DNA- encoded chemistry technology Jimmidi, Ravikumar; Monsivais, Diana; Ta, Hai Minh; Sharma, Kiran L.; Bohren, Kurt M.; Chamakuri, Srinivas; Liao, Zian; Li, Feng; Hakenjos, John M.; Li, Jian - Yuan; Mishina, Yuji; Pan, Haichun; Qin, Xuan; Robers, Matthew B.; Sankaran, Banumathi; Tan, Zhi; Tang, Suni; Vasquez, Yasmin M.; Wilkinson, Jennifer; Young, Damian W.; Palmer, Stephen S.; Mackenzie, Kevin R.; Kim, Choel; Matzuk, Martin M. 分享 收藏
Identification of potent pan- ephrin receptor kinase inhibitors using DNA- encoded chemistry technology Madasu, Chandrashekhar; Liao, Zian; Parks, Sydney E.; Sharma, Kiran L.; Bohren, Kurt M.; Ye, Qiuji; Li, Feng; Palaniappan, Murugesan; Tan, Zhi; Yuan, Fei; Creighton, Chad J.; Tang, Suni; Masand, Ramya P.; Guan, Xiaoming; Young, Damian W.; Monsivais, Diana; Matzuk, Martin M. 分享 收藏
CYP3A Mediates an Unusual C(sp2)-C(sp3) Bond Cleavage via Ipso-Addition of Oxygen in Drug Metabolism Qin, Xuan; Wang, Yong; Ye, Qiuji; Hakenjos, John M.; Wang, Jin; Teng, Mingxing; Guo, Lei; Tan, Zhi; Young, Damian W.; Mackenzie, Kevin R.; Li, Feng 分享 收藏
Expanding Complex Morpholines Using Systematic Chemical Diversity Tang, Sunny Ann; Fults, Afton; Boyd, Shelton R.; Gattu, Nikhil; Tran, Kevin A.; Fan, Jiayi; Mackenzie, Kevin R.; Palzkill, Timothy; Young, Damian W.; Chamakuri, Srinivas 分享 收藏
Chemical Catalysis Guides Structural Identification for the Major In Vivo Metabolite of the BET Inhibitor JQ1 Holmes, Secondra; Jain, Prashi; Rodriguez, Kenneth Guzman; Williams, Jade; Yu, Zhifeng; Cerda-Smith, Christian; Samuel, Errol L. G.; Campbell, James; Hakenjos, John Michael; Monsivais, Diana; Li, Feng; Chamakuri, Srinivas; Matzuk, Martin M.; Santini, Conrad; Mackenzie, Kevin R.; Young, Damian W. 分享 收藏
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DNA-encoded chemical libraries yield non-covalent and non-peptidic SARS-CoV-2 main protease inhibitors Jimmidi, Ravikumar; Chamakuri, Srinivas; Lu, Shuo; Ucisik, Melek Nihan; Chen, Peng-Jen; Bohren, Kurt M.; Moghadasi, Seyed Arad; Versteeg, Leroy; Nnabuife, Christina; Li, Jian-Yuan; Qin, Xuan; Chen, Ying-Chu; Faver, John C.; Nyshadham, Pranavanand; Sharma, Kiran L.; Sankaran, Banumathi; Judge, Allison; Yu, Zhifeng; Li, Feng; Pollet, Jeroen; Harris, Reuben S.; Matzuk, Martin M.; Palzkill, Timothy; Young, Damian W. 分享 收藏
Identifying the Reactive Metabolites of Tyrosine Kinase Inhibitor Pexidartinib In Vitro Using LC-MS-Based Metabolomic Approaches 使用基于lc-ms的代谢组学方法体外鉴定酪氨酸激酶抑制剂Pexidartinib的反应性代谢物 Qin, Xuan; Wang, Yong; MacKenzie, Kevin R.; Hakenjos, John M.; Chen, Si; Khalil, Saleh M.; Jung, Sung Yun; Young, Damian W.; Guo, Lei; Li, Feng 分享 收藏
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Discovery of Highly Potent and BMPR2-Selective Kinase Inhibitors Using DNA-Encoded Chemical Library Screening Modukuri, Ram K.; Monsivais, Diana; Li, Feng; Palaniappan, Murugesan; Bohren, Kurt M.; Tan, Zhi; Ku, Angela F.; Wang, Yong; Madasu, Chandrashekhar; Li, Jian-Yuan; Tang, Suni; Miklossy, Gabriella; Palmer, Stephen S.; Young, Damian W.; Matzuk, Martin M. 分享 收藏
Advancing ASMS with LC-MS/MS for the discovery of novel PDCL2 ligands from DNA-encoded chemical library selections Ye, Qiuji; Belabed, Hassane; Wang, Yong; Yu, Zhifeng; Palaniappan, Murugesan; Li, Jian-Yuan; Kalovidouris, Stacey A.; MacKenzie, Kevin R.; Teng, Mingxing; Young, Damian W.; Fujihara, Yoshitaka; Matzuk, Martin M. 分享 收藏
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