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Development of Potent Mcl-1 Inhibitors: Structural Investigations on Macrocycles Originating from a DNA-Encoded Chemical Library Screen 开发有效的Mcl-1抑制剂: 源自DNA编码的化学文库筛选的大环的结构研究 Hekking, Koen F. W.; Maroto, Sergio; van Kekem, Kees; Haasjes, Frank S.; Slootweg, Jack C.; Oude Alink, Patrick G. B.; Dirks, Ron; Sardana, Malvika; Bolster, Marjon G.; Kuijpers, Brian; Smith, Dennis; Doodeman, Robin; Scheepstra, Marcel; Zech, Birgit; Mulvihill, Mark; Renzetti, Louis M.; Babiss, Lee; Centrella, Paolo A.; Clark, Matthew A.; Cuozzo, John W.; Guie, Marie-Aude; Sigel, Eric; Habeshian, Sevan; Hupp, Christopher D.; Liu, Julie; Thomson, Heather A.; Zhang, Ying; Keefe, Anthony D.; Muller, Gerhard; Gremmen, Stijn 分享 收藏
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Discovery of 2,4-1H-Imidazole Carboxamides as Potent and Selective TAK1 Inhibitors Veerman, Johan J. N.; Bruseker, Yorik B.; Damen, Eddy; Heijne, Erik H.; van Bruggen, Wendy; Hekking, Koen F. W.; Winkel, Rob; Hupp, Christopher D.; Keefe, Anthony D.; Liu, Julie; Thomson, Heather A.; Zhang, Ying; Cuozzo, John W.; McRiner, Andrew J.; Mulvihill, Mark J.; van Rijnsbergen, Peter; Zech, Birgit; Renzetti, Louis M.; Babiss, Lee; Muller, Gerhard 分享 收藏
Fast Iterative Synthetic Approach toward Identification of Novel Highly Selective p38 MAP Kinase Inhibitors Roehm, Sandra; Berger, Benedict-Tilman; Schroeder, Martin; Chaikuad, Apirat; Winkel, Rob; Hekking, Koen F. W.; Benningshof, Jorg J. C.; Mueller, Gerhard; Tesch, Roberta; Kudolo, Mark; Forster, Michael; Laufer, Stefan; Knapp, Stefan 分享 收藏
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Expansion of chemical space for collaborative lead generation and drug discovery: the European Lead Factory Perspective Karawajczyk, Anna; Giordanetto, Fabrizio; Benningshof, Jorg; Hamza, Daniel; Kalliokoski, Tuomo; Pouwer, Kees; Morgentin, Remy; Nelson, Adam; Muller, Gerhard; Piechot, Alexander; Tzalis, Dimitrios 分享 收藏