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Pharmacologic inhibition of SOX9-CDK4 by CYD-4-61 impairs gastric adenocarcinoma growth and amplifies anti-PD-1 response CYD-4-61通过药理抑制SOX9-CDK4抑制胃腺癌生长并增强抗PD-1反应 Zou, Gengyi; Yoshimura, Katsuhiro; Fan, Yibo; Zeng, Liyong; Bhati, Aryanasingh S.; Vanpariya, Bansi R.; Dai, Enyu; Yamashita, Kohei; Wang, Lingzhi; Wu, Jingjing; Shao, Shan; Scott, Ailing W.; Jin, Jiankang; Pizzi, Melissa Pool; Yao, Xiaodan; Brown, Calena-Abel; Cao, Fang; Wang, Ruiping; Han, Xueshuai; Li, Jun; Chen, Haiying; Wang, Pingyuan; Wang, Linghua; Liu, Bin; Zhou, Jia; Lo, Yuan-Hung; Gan, Qiong; Waters, Rebecca; Yin, Feng; Song, Shumei; Ajani, Jaffer A.; Dhar, Shilpa S. 分享 收藏
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Orally Bioavailable BRD4 BD1 Inhibitor ZL0516 Effectively Suppresses Colonic Inflammation in Animal Models of Inflammatory Bowel Disease 口服生物利用度BRD4 BD1抑制剂ZL0516可有效抑制炎症性肠病动物模型中的结肠炎症 Ma, ZH; McAninch, S; Liu, ZQ; Zhang, C; Chen, HY; He, J; Yang, WJ; Panganiban, RP; Cong, YZ; Yochum, G; Brasier, AR; Pinchuk, IV; Tian, B; Zhou, J 分享 收藏
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Targeting CDK9 with a novel potent and selective inhibitor, YX0798, in CAR-Trelapsed mantle cell lymphoma models Jiang, Vivian; Xue, Yu; Kim, Hong; McIntosh, Joseph; Chen, Haiying; Zhang, Tianci; Liu, Yang; Zhou, Jia; Wang, Michael 分享 收藏
IDR-targeting compounds suppress HPV genome replication via disruption of phospho-BRD4 association with DNA damage response factors Wu, Shwu-Yuan; Lai, Hsien-Tsung; Banerjee, N. Sanjib; Ma, Zonghui; Santana, Juan F.; Wei, Shuguang; Liu, Xisheng; Zhang, Meirong; Zhan, Jian; Chen, Haiying; Posner, Bruce; Chen, Yadong; Price, David H.; Chow, Louise T.; Zhou, Jia; Chiang, Cheng-Ming 分享 收藏
Development and validation of a machine learning model to predict prognosis in HIV-negative cryptococcal meningitis patients: a multicenter study Liu, Junyu; Lu, Yaxin; Liu, Jia; Liang, Jiayin; Zhang, Qilong; Li, Hua; Zhong, Xiufeng; Bu, Hui; Wang, Zhanhang; Fan, Liuxu; Liang, Panpan; Xie, Jia; Wang, Yuan; Gong, Jiayin; Chen, Haiying; Dai, Yangyang; Yang, Lu; Su, Xiaohong; Wang, Anni; Xiong, Lei; Xia, Han; Jiang, Ying; Liu, Zifeng; Peng, Fuhua 分享 收藏
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Discovery of Novel Oleamide Analogues as Brain-Penetrant Positive Allosteric Serotonin 5-HT2C Receptor and Dual 5-HT2C/5-HT2A Receptor Modulators Chen, Jianping; Garcia, Erik J.; Merritt, Christina R.; Zamora, Joshua C.; Bolinger, Andrew A.; Pazdrak, Konrad; Stafford, Susan J.; Mifflin, Randy C.; Wold, Eric A.; Wild, Christopher T.; Chen, Haiying; Anastasio, Noelle C.; Cunningham, Kathryn A.; Zhou, Jia 分享 收藏
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