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Macrofilaricidal Benzimidazole-Benzoxaborole Hybrids as an Approach to the Treatment of River Blindness: Part 1. Amide Linked Analogs Akama, Tsutomu; Freund, Yvonne R.; Berry, Pamela W.; Carter, David S.; Easom, Eric E.; Jarnagin, Kurt; Lunde, Christopher S.; Plattner, Jacob J.; Rock, Fernando; Stefanakis, Rianna; Fischer, Chelsea; Bulman, Christina A.; Lim, Kee Chong; Suzuki, Brian M.; Tricoche, Nancy; Mansour, Abdelmoneim; DiCosty, Utami; McCall, Scott; Carson, Ben; McCall, John W.; McKerrow, James; Huebner, Marc P.; Specht, Sabine; Hoerauf, Achim; Lustigman, Sara; Sakanari, Judy A.; Jacobs, Robert T. 分享 收藏
Macrofilaricidal Benzimidazole-Benzoxaborole Hybrids as an Approach to the Treatment of River Blindness: Part 2. Ketone Linked Analogs Carter, David S.; Jacobs, Robert T.; Freund, Yvonne R.; Berry, Pamela W.; Akama, Tsutomu; Easom, Eric E.; Lunde, Christopher S.; Rock, Fernando; Stefanakis, Rianna; McKerrow, James; Fischer, Chelsea; Bulman, Christina A.; Lim, Kee Chong; Suzuki, Brian M.; Tricoche, Nancy; Sakanari, Judy A.; Lustigman, Sara; Plattner, Jacob J. 分享 收藏
Efficacy and Improved Resistance Potential of a Cofactor-Independent InhA Inhibitor of Mycobacterium tuberculosis in the C3HeB/FeJ Mouse Model Robertson, Gregory T.; Ektnitphong, Victoria A.; Scherman, Michael S.; McNeil, Matthew B.; Dennison, Devon; Korkegian, Aaron; Smith, Anthony J.; Halladay, Jason; Carter, David S.; Xia, Yi; Zhou, Yasheen; Choi, Wai; Berry, Pamela W.; Mao, Weimin; Hernandez, Vincent; Alley, R. K.; Parish, Tanya; Lenaerts, Anne J. 分享 收藏
Boron-Pleuromutilins as Anti-Wolbachia Agents with Potential for Treatment of Onchocerciasis and Lymphatic Filariasis Jacobs, Robert T.; Lunde, Christopher S.; Freund, Yvonne R.; Hernandez, Vincent; Li, Xianfeng; Xia, Yi; Carter, David S.; Berry, Pamela W.; Halladay, Jason; Rock, Fernando; Stefanakis, Rianna; Easom, Eric; Plattner, Jacob J.; Ford, Louise; Johnston, Kelly L.; Cook, Darren A. N.; Clare, Rachel; Cassidy, Andrew; Myhill, Laura; Tyrer, Hayley; Gamble, Joanne; Guimaraes, Ana F.; Steven, Andrew; Lenz, Franziska; Ehrens, Alexandra; Frohberger, Stefan J.; Koschel, Marianne; Hoerauf, Achim; Huebner, Marc P.; McNamara, Case W.; Bakowski, Malina A.; Turner, Joseph D.; Taylor, Mark J.; Ward, Stephen A. 分享 收藏
Discovery of a cofactor-independent inhibitor of Mycobacterium tuberculosis InhA Xia, Yi; Zhou, Yasheen; Carter, David S.; McNeil, Matthew B.; Choi, Wai; Halladay, Jason; Berry, Pamela W.; Mao, Weimin; Hernandez, Vincent; O'Malley, Theresa; Korkegian, Aaron; Sunde, Bjorn; Flint, Lindsay; Woolhiser, Lisa K.; Scherman, Michael S.; Gruppo, Veronica; Hastings, Courtney; Robertson, Gregory T.; Ioerger, Thomas R.; Sacchettini, Jim; Tonge, Peter J.; Lenaerts, Anne J.; Parish, Tanya; Alley, M. R. K. 分享 收藏
Discovery of N-[4-[6-tert-Butyl-5-methoxy-8-(6-methoxy-2-oxo-1H-pyridin-3-yl)-3-quinolyl]phenyl]methanesulfonamide (RG7109), a Potent Inhibitor of the Hepatitis C Virus NS5B Polymerase Talamas, Francisco X.; Abbot, Sarah C.; Anand, Shalini; Brameld, Ken A.; Carter, David S.; Chen, Jun; Davis, Dana; de Vicente, Javier; Fung, Amy D.; Gong, Leyi; Harris, Seth F.; Inbar, Petra; Labadie, Sharada S.; Lee, Eun K.; Lemoine, Remy; Le Pogam, Sophie; Leveque, Vincent; Li, Jim; McIntosh, Joel; Najera, Isabel; Park, Jaehyeon; Railkar, Aruna; Rajyaguru, Sonal; Sangi, Michael; Schoenfeld, Ryan C.; Staben, Leanna R.; Tan, Yunchou; Taygerly, Joshua P.; Villasenor, Armando G.; Weller, Paul E. 分享 收藏
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