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Xavier Lucas

monte rosa therapeutics inc, boston, ma, usa.

25H指数
89论文数
3.3K被引数
收录论文 26
发表时间
Mining the CRBN target space redefines rules for molecular glue–induced neosubstrate recognition挖掘CRBN靶点空间重新定义了分子胶诱导的新型底物识别规则
errScience
IF45.8
err2025-07-03
err0
errOAAI
errGeorg Petzold; Pablo Gainza; Stefano Annunziato; Ilaria Lamberto; Peter Trenh; Laura A. McAllister; Bradley DeMarco; Laura Schwander; Richard D. Bunker; Mary Zlotosch; Rohitha SriRamaratnam; Samuel Gilberto; Gerasimos Langousis; Etienne J. Donckele; Chao Quan; Vaik Strande; Gian Marco De Donatis; Shanique B. Alabi; Jessica Alers; Michelle Matysik; Camille Staehly; Aurélie Dubois; Arnaud Osmont; Mackenzie Garskovas; David Lyon; Lars Wiedmer; Vladimiras Oleinikovas; Raphael Lieberherr; Nooreen T. Rubin; Daniel T. Lam; Xavier Lucas; Elisa Liardo; Nina Ilic Widlund; Andreas Ritzén; Ramon Miguel Caceres; Dominico Vigil; Jennifer Tsai; Owen Wallace; Marisa Peluso; Amine Sadok; Ralph Tiedt; Alison M. Paterson; Vladislav Zarayskiy; Bernhard Fasching; Debora Bonenfant; Markus Warmuth; John C. Castle; Sharon A. Townson
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The molecular basis of drug selectivity for α5 subunit-containing GABAA receptors
err2023-10-30
err6
errOAAI
errKasaragod, Vikram Babu; Malinauskas, Tomas; Wahid, Ayla A.; Lengyel, Judith; Knoflach, Frederic; Hardwick, Steven W.; Jones, Charlotte F.; Chen, Wan-Na; Lucas, Xavier; El Omari, Kamel; Chirgadze, Dimitri Y.; Aricescu, A. Radu; Cecere, Giuseppe; Hernandez, Maria-Clemencia; Miller, Paul S.
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Peptide conformational sampling using the Quantum Approximate Optimization Algorithm
err2023-07-17
err8
errOAAI
errBoulebnane, Sami; Lucas, Xavier; Meyder, Agnes; Adaszewski, Stanislaw; Montanaro, Ashley
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Collaborative Assessment of Molecular Geometries and Energies from the Open Force Field
err2022-11-26
err13
errOAAI
errD'Amore, Lorenzo; Hahn, David F.; Dotson, David L.; Horton, Joshua T.; Anwar, Jamshed; Craig, Ian; Fox, Thomas; Gobbi, Alberto; Lakkaraju, Sirish Kaushik; Lucas, Xavier; Meier, Katharina; Mobley, David L.; Narayanan, Arjun; Schindler, Christina E. M.; Swope, William C.; in't Veld, Pieter J.; Wagner, Jeffrey; Xue, Bai; Tresadern, Gary
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Development and Benchmarking of Open Force Field v1.0.0-the Parsley Small-Molecule Force Field
err2021-09-22
err93
errOAAI
errQiu, Yudong; Smith, Daniel G. A.; Boothroyd, Simon; Jang, Hyesu; Hahn, David F.; Wagner, Jeffrey; Bannan, Caitlin C.; Gokey, Trevor; Lim, Victoria T.; Stern, Chaya D.; Rizzi, Andrea; Tjanaka, Bryon; Tresadern, Gary; Lucas, Xavier; Shirts, Michael R.; Gilson, Michael K.; Chodera, John D.; Bayly, Christopher, I; Mobley, David L.; Wang, Lee-Ping
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4-Acyl Pyrroles as Dual BET-BRD7/9 Bromodomain Inhibitors Address BETi Insensitive Human Cancer Cell Lines
err2020-12-04
err16
PREAI
errHuegle, Martin; Regenass, Pierre; Warstat, Robin; Hau, Mirjam; Schmidtkunz, Karin; Lucas, Xavier; Wohlwend, Daniel; Einsle, Oliver; Jung, Manfred; Breit, Bernhard; Guenther, Stefan
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The ChemicalToolbox: reproducible, user-friendly cheminformatics analysis on the Galaxy platform
err2020-06-01
err28
errOAAI
errBray, Simon A.; Lucas, Xavier; Kumar, Anup; Gruening, Bjoern A.
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Structure-Based Design of a Macrocyclic PROTAC基于结构的大环PROTAC设计
err2019-12-12
err156
errOAAI
errTesta, Andrea; Hughes, Scott J.; Lucas, Xavier; Wright, Jane E.; Ciulli, Alessio
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3-Fluoro-4-hydroxyprolines: Synthesis, Conformational Analysis, and Stereoselective Recognition by the VHL E3 Ubiquitin Ligase for Targeted Protein Degradation (vol 140, pg 9299, 2018)
err2019-04-24
err1
errOAAI
errTesta, Andrea; Lucas, Xavier; Castro, Guilherme V.; Chan, Kwok-Ho; Wright, Jane E.; Runcie, Andrew C.; Gadd, Morgan S.; Harrison, William T. A.; Ko, Eun-Jung; Fletcher, Daniel; Ciulli, Alessio
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3-Fluoro-4-hydroxyprolines: Synthesis, Conformational Analysis, and Stereoselective Recognition by the VHL E3 Ubiquitin Ligase for Targeted Protein Degradation
err2018-06-27
err106
errOAAI
errTesta, Andrea; Lucas, Xavier; Castro, Guilherme, V; Chan, Kwok-Ho; Wright, Jane E.; Runcie, Andrew C.; Gadd, Morgan S.; Harrison, William T. A.; Ko, Eun-Jung; Fletcher, Daniel; Ciulli, Alessio
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Targeting Ligandable Pockets on Plant Homeodomain (PHD) Zinc Finger Domains by a Fragment-Based Approach
err2018-03-12
err29
errOAAI
errAmato, Anastasia; Lucas, Xavier; Bortoluzzi, Alessio; Wright, David; Ciulli, Alessio
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Beyond the BET Family: Targeting CBP/p300 with 4-Acyl Pyrroles
err2017-09-07
err29
errOAAI
errHuegle, Martin; Lucas, Xavier; Ostrovskyi, Dmytro; Regenass, Pierre; Gerhardt, Stefan; Einsle, Oliver; Hau, Mirjam; Jung, Manfred; Breit, Bernhard; Guenther, Stefan; Wohlwend, Daniel
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Structural basis of molecular recognition of helical histone H3 tail by PHD finger domains
err2017-05-04
err25
errOAAI
errBortoluzzi, Alessio; Amato, Anastasia; Lucas, Xavier; Blank, Manuel; Ciulli, Alessio
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Structural basis of PROTAC cooperative recognition for selective protein degradation选择性蛋白质降解的PROTAC协同识别的结构基础
err2017-03-13
err857
errOAAI
errGadd, Morgan S.; Testa, Andrea; Lucas, Xavier; Chan, Kwok-Ho; Chen, Wenzhang; Lamont, Douglas J.; Zengerle, Michael; Ciulli, Alessio
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4-Acyl Pyrrole Derivatives Yield Novel Vectors for Designing Inhibitors of the Acetyl-Lysine Recognition Site of BRD4(1)
err2016-01-14
err52
PREAI
errHuegle, Martin; Lucas, Xavier; Weitzel, Gerhard; Ostrovskyi, Dmytro; Breit, Bernhard; Gerhardt, Stefan; Einsle, Oliver; Guenther, Stefan; Wohlwend, Daniel
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A thorough anion-π interaction study in biomolecules: on the importance of cooperativity effects
err2016-01-01
err189
errOAAI
errLucas, Xavier; Bauza, Antonio; Frontera, Antonio; Quinonero, David
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StreptomeDB 2.0-an extended resource of natural products produced by streptomycetes
err2015-11-28
err77
errOAAI
errKlementz, Dennis; Doering, Kersten; Lucas, Xavier; Telukunta, Kiran K.; Erxleben, Anika; Deubel, Denise; Erber, Astrid; Santillana, Irene; Thomas, Oliver S.; Bechthold, Andreas; Guenther, Stefan
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