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Lee E. Schechter

Pfizer

46H指数
153论文数
6.6K被引数
收录论文 36
发表时间
Negative allosteric modulation of metabotropic glutamate receptor 5 results in broad spectrum activity relevant to treatment resistant depression
err2013-03-01
err72
PREAI
errHughes, Z. A.; Neal, S. J.; Smith, D. L.; Rizzo, S. J. Sukoff; Pulicicchio, C. M.; Lotarski, S.; Lu, S.; Dwyer, J. M.; Brennan, J.; Olsen, M.; Bender, C. N.; Kouranova, E.; Andree, T. H.; Harrison, J. E.; Whiteside, G. T.; Springer, D.; O'Neil, S. V.; Leonard, S. K.; Schechter, L. E.; Dunlop, J.; Rosenzweig-Lipson, S.; Ring, R. H.
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Characterization of Vabicaserin (SCA-136), a Selective 5-Hydroxytryptamine 2C Receptor Agonist
err2011-06-01
err49
PREAI
errDunlop, John; Watts, Stephanie W.; Barrett, James E.; Coupet, Joseph; Harrison, Boyd; Mazandarani, Hossein; Nawoschik, Stanley; Pangalos, Menelas N.; Ramamoorthy, Siva; Schechter, Lee; Smith, Deborah; Stack, Gary; Zhang, Jean; Zhang, Guoming; Rosenzweig-Lipson, Sharon
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Identification of 3-sulfonylindazole derivatives as potent and selective 5-HT6 antagonists
err2011-01-01
err19
PREAI
errLiu, Kevin G.; Robichaud, Albert J.; Greenfield, Alexander A.; Lo, Jennifer R.; Grosanu, Cristina; Mattes, James F.; Cai, Yanxuan; Zhang, Guo Ming; Zhang, Jean Y.; Kowal, Dianne M.; Smith, Deborah L.; Di, Li; Kerns, Edward H.; Schechter, Lee E.; Comery, Thomas A.
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5-Piperazinyl-3-sulfonylindazoles as Potent and Selective 5-Hydroxytryptamine-6 Antagonists
err2010-10-08
err62
PREAI
errLiu, Kevin G.; Robichaud, Albert J.; Bernotas, Ronald C.; Yan, Yinfa; Lo, Jennifer R.; Zhang, Mei-Yi; Hughes, Zoe A.; Huselton, Christine; Zhang, Guo Ming; Zhang, Jean Y.; Kowal, Dianne M.; Smith, Deborah L.; Schechter, Lee E.; Comery, Thomas A.
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Angiotensin IV elevates oxytocin levels in the rat amygdala and produces anxiolytic-like activity through subsequent oxytocin receptor activation
err2010-03-12
err31
PREAI
errBeyer, Chad E.; Dwyer, Jason M.; Platt, Brian J.; Neal, Sarah; Luo, Bin; Ling, Huai-Ping; Lin, Qian; Mark, Robert J.; Rosenzweig-Lipson, Sharon; Schechter, Lee E.
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Antidepressant and anxiolytic effects of selective 5-HT6 receptor agonists in rats
err2010-03-09
err77
errOAAI
errCarr, Gregory V.; Schechter, Lee E.; Lucki, Irwin
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5-Cyclic Amine-3-arylsulfonylindazoles as Novel 5-HT6 Receptor Antagonists
err2010-02-19
err24
PREAI
errHaydar, Simon N.; Yun, Heedong; Andrae, Patrick M.; Mattes, James; Zhang, Jean; Kramer, Angela; Smith, Deborah L.; Huselton, Christine; Graf, Radka; Aschmies, Suzan; Schechter, Lee E.; Comery, Thomas A.; Robichaud, Albert J.
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Synthesis, Potency, and in Vivo Evaluation of 2-Piperazin-1-ylquinoline Analogues as Dual Serotonin Reuptake Inhibitors and Serotonin 5-HT1A Receptor Antagonists
err2009-07-21
err17
PREAI
errZhou, Dahui; Stack, Gary P.; Lo, Jennifer; Failli, Amedeo A.; Evrard, Deborah A.; Harrison, Boyd L.; Hatzenbuhler, Nicole T.; Tran, Megan; Croce, Susan; Yi, Soo; Golembieski, Jeannette; Hornby, Geoffrey A.; Lai, Margaret; Lin, Qian; Schechter, Lee E.; Smith, Deborah L.; Shilling, Adam D.; Huselton, Christine; Mitchell, Paul; Beyer, Chad E.; Andree, Terrance H.
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Novel 1-aminoethyl-3-arylsulfonyl-1H-pyrrolo[2,3-b]pyridines are potent 5-HT6 agonists
err2009-07-01
err20
PREAI
errBernotas, Ronald C.; Lenicek, Steven; Antane, Schuyler; Cole, Derek C.; Harrison, Boyd L.; Robichaud, Albert J.; Zhang, Guo Ming; Smith, Deborah; Platt, Brian; Lin, Qian; Li, Ping; Coupet, Joseph; Rosenzweig-Lipson, Sharon; Beyer, Chad E.; Schechter, Lee E.
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Advances toward New Antidepressants with Dual Serotonin Transporter and 5-HT1A Receptor Affinity within a Class of 3-Aminochroman Derivatives. Part 2
err2008-10-04
err31
PREAI
errHatzenbuhler, Nicole T.; Baudy, Reinhardt; Evrard, Deborah A.; Failli, Amedeo; Harrison, Boyd L.; Lenicek, Steven; Mewshaw, Richard E.; Saab, Annmarie; Shao, Uresh; Sze, Jean; Zhang, Minsheng; Zhou, Dahui; Chlenov, Michael; Kagan, Michael; Golembieski, Jeannette; Hornby, Geoffrey; Lai, Margaret; Smith, Deborah L.; Sullivan, Kelly M.; Schechter, Lee E.; Andree, Terrance H.
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Antidepressant-like behavioral effects of IGF-I produced by enhanced serotonin transmission
err2008-10-01
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errOAAI
errHoshaw, Brian A.; Hill, Tiffany I.; Crowley, James J.; Malberg, Jessica E.; Khawaja, Xavier; Rosenzweig-Lipson, Sharon; Schechter, Lee E.; Lucki, Irwin
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Studies toward the discovery of the next generation of antidepressants.: Part 6:: Dual 5-HT1A receptor and serotonin transporter affinity within a class of arylpiperazinyl-cyclohexyl indole derivatives
err2008-07-01
err32
PREAI
errZhou, Dahui; Zhou, Ping; Evrard, Deborah A.; Meagher, Kristin; Webb, Michael; Harrison, Boyd L.; Huryn, Donna M.; Golembieski, Jeannette; Hornby, Geoffrey A.; Schechter, Lee E.; Smith, Deborah L.; Andree, Terrance H.; Mewshaw, Richard E.
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Correlating efficacy in rodent cognition models with in vivo 5-hydroxytryptamine1A receptor occupancy by a novel antagonist, (R)-N-(2-methyl-(4-indolyl-1-piperazinyl)ethyl)-N-(2-pyridinyl)-cyclohexane carboxamide (WAY-101405)
err2008-04-01
err39
PREAI
errHirst, Warren D.; Andree, Terrance H.; Aschmies, Suzan; Childers, Wayne E.; Comery, Thomas A.; Dawson, Lee A.; Day, Mark; Feingold, Irene B.; Grauer, Steven M.; Harrison, Boyd L.; Hughes, Zoe A.; Kao, John; Kelly, Michael G.; van der Lee, Heidi; Rosenzweig-Lipson, Sharon; Saab, Annmarie L.; Smith, Deborah L.; Sullivan, Kelly; Rizzo, Stacey J. Sukoff; Tio, Cesario; Zhang, Mei-Yi; Schechter, Lee E.
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Pharmacology of neuropeptide S in mice: therapeutic relevance to anxiety disorders
err2008-03-03
err132
PREAI
errLeonard, Sarah K.; Dwyer, Jason M.; Rizzo, Stacey J. Sukoff; Platt, Brian; Logue, Sheree F.; Neal, Sarah J.; Malberg, Jessica E.; Beyer, Chad E.; Schechter, Lee E.; Rosenzweig-Lipson, Sharon; Ring, Robert H.
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Discovery of N1-(6-chloroimidazo[2,1-b][1,3]-thiazole-5-sulfonyl)tryptamine as a potent, selective, and orally active 5-HT6 receptor agonist
err2007-10-19
err53
PREAI
errCole, Derek C.; Stock, Joseph R.; Lennox, William J.; Bernotas, Ronald C.; Ellingboe, John W.; Boikess, Steve; Coupet, Joseph; Smith, Deborah L.; Leung, Louis; Zhang, Guo-Ming; Feng, Xidong; Kelly, Michael F.; Galante, Rocco; Huang, Pingzhong; Dawson, Lee A.; Marquis, Karen; Rosenzweig-Lipson, Sharon; Beyer, Chad E.; Schechter, Lee E.
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A novel approach for predicting antidepressant-induced sexual dysfunction in rats
err2007-09-16
err22
PREAI
errRizzo, Stacey J. Sukoff; Schechter, Lee E.; Rosenzweig-Lipson, Sharon
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Novel 1-(azacyclyl)-3-aryisulfonyl-1H-pyrrolo[2,3-b]pyridines as 5-HT6 agonists and antagonists
err2007-09-01
err15
PREAI
errElokdah, Hassan; Li, David; McFarlane, Geraldine; Bernotas, Ronald C.; Robichaud, Albert J.; Magolda, Ronald L.; Zhang, Guo Ming; Smith, Deborah; Schechter, Lee E.
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