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J

Joseph B. Bolen

Takeda Pharmaceutical Company Ltd

75H指数
245论文数
2.1W被引数
收录论文 35
发表时间
PHASE1/2 STUDY OF AN ANTI-GALECTIN-9 ANTIBODY, LYT-200, IN PATIENTS WITH METASTATIC SOLID TUMORS
err2021-11-10
err4
errOAAI
errFilipovic, Aleksandra; Wainber, Zev; Wang, Judy; Bendell, Johanna; Janku, Filip; Sharma, Manish; Mahipal, Amit; Bolen, Joseph; Elenko, Eric; Korth, Christopher; Dranitsaris, George
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MLN8054 and Alisertib (MLN8237): Discovery of Selective Oral Aurora A Inhibitors
err2015-05-05
err81
errOAAI
errSells, Todd B.; Chau, Ryan; Ecsedy, Jeffrey A.; Gershman, Rachel E.; Hoar, Kara; Huck, Jessica; Janowick, David A.; Kadambi, Vivek J.; LeRoy, Patrick J.; Stirling, Matthew; Stroud, Stephen G.; Vos, Tricia J.; Weatherhead, Gabriel S.; Wysong, Deborah R.; Zhang, Mengkun; Balani, Suresh K.; Bolen, Joseph B.; Manfredi, Mark G.; Claiborne, Christopher F.
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Choosing the right schedule for progression free survival: A systems pharmacology approach
err2014-10-01
err0
PREAI
errPatel, Mayankbhai; Mettetal, Jerome; Cohen, Matthew; Palani, Santhosh; Kuida, Keisuke; Hixon, Mark; Bolen, Joseph; Shyu, Wen Chyi; Noe, Dennis; Chakravarty, Arijit
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Combinatorial therapy design in cancer as a directed attack on the hubs of a scale-free network.
err2013-11-01
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PREAI
errChen, Andrew; Chakravarty, Arijit; Mettetal, Jerome; Shyu, Wen Chyi; Bolen, Joseph; Palani, Santhosh
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Evaluation of Predictive Biomarkers for the Antineoplastic Effect of TAK-733, a Novel Investigational Allosteric Inhibitor of MEK1/2
err2012-11-01
err0
PREAI
errGangolli, E.; Blair, D.; Schu, M.; Szynal, C.; Ecsedy, J.; Hori, A.; Dorner, A.; Bolen, J.; Vincent, P.; Chakravarty, A.
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Characterization of Alisertib (MLN8237), an Investigational Small-Molecule Inhibitor of Aurora A Kinase Using Novel In Vivo Pharmacodynamic Assays
err2011-12-18
err274
errOAAI
errManfredi, Mark G.; Ecsedy, Jeffrey A.; Chakravarty, Arijit; Silverman, Lee; Zhang, Mengkun; Hoar, Kara M.; Stroud, Stephen G.; Chen, Wei; Shinde, Vaishali; Huck, Jessica J.; Wysong, Deborah R.; Janowick, David A.; Hyer, Marc L.; Leroy, Patrick J.; Gershman, Rachel E.; Silva, Matthew D.; Germanos, Melissa S.; Bolen, Joseph B.; Claiborne, Christopher F.; Sells, Todd B.
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Antitumor Activity of the Investigational Proteasome Inhibitor MLN9708 in Mouse Models of B-cell and Plasma Cell Malignancies
err2011-11-30
err101
errOAAI
errLee, Edmund C.; Fitzgerald, Michael; Bannerman, Bret; Donelan, Jill; Bano, Kristen; Terkelsen, Jennifer; Bradley, Daniel P.; Subakan, Ozlem; Silva, Matthew D.; Liu, Ray; Pickard, Michael; Li, Zhi; Tayber, Olga; Li, Ping; Hales, Paul; Carsillo, Mary; Neppalli, Vishala T.; Berger, Allison J.; Kupperman, Erik; Manfredi, Mark; Bolen, Joseph B.; Van Ness, Brian; Janz, Siegfried
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Substrate-Assisted Inhibition of Ubiquitin-like Protein-Activating Enzymes: The NEDD8 E1 Inhibitor MLN4924 Forms a NEDD8-AMP Mimetic In Situ
err2010-01-01
err449
errOAAI
errBrownell, James E.; Sintchak, Michael D.; Gavin, James M.; Liao, Hua; Bruzzese, Frank J.; Bump, Nancy J.; Soucy, Teresa A.; Milhollen, Michael A.; Yang, Xiaofeng; Burkhardt, Anne L.; Ma, Jingya; Loke, Huay-Keng; Lingaraj, Trupti; Wu, Dongyun; Hamman, Kristin B.; Spelman, James J.; Cullis, Courtney A.; Langston, Steven P.; Vyskocil, Stepan; Sells, Todd B.; Mallender, William D.; Visiers, Irache; Li, Ping; Claiborne, Christopher F.; Rolfe, Mark; Bolen, Joseph B.; Dick, Lawrence R.
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Antitumor activity of MLN8054, an orally active small-molecule inhibitor of Aurora A kinase
err2007-03-06
err421
errOAAI
errManfredi, Mark G.; Ecsedy, Jeffrey A.; Meetze, Kristan A.; Balani, Suresh K.; Burenkova, Olga; Chen, Wei; Galvin, Katherine M.; Hoar, Kara M.; Huck, Jessica J.; LeRoy, Patrick J.; Ray, Emily T.; Sells, Todd B.; Stringer, Bradley; Stroud, Stephen G.; Vos, Tricia J.; Weatherhead, Gabriel S.; Wysong, Deborah R.; Zhang, Mengkun; Bolen, Joseph B.; Claiborne, Christopher F.
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Longitudinally quantitative 2-deoxy-2-[18F] fluoro-D-glucose micro positron emission tomography imaging for efficacy of new anticancer drugs:: A case study with bortezomib in prostate cancer murine model
err2006-08-04
err18
PREAI
errZhang, Yumin; Saylor, Melissa; Wen, Shenhua; Silva, Matthew D.; Rolfe, Mark; Bolen, Joseph; Muir, Craig; Reimer, Corinne; Chandra, Sudeep
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BICYCLIC COMPOUNDS AS RING-CONSTRAINED INHIBITORS OF PROTEIN-TYROSINE KINASE-P56LCK
err2002-05-01
err111
PREAI
errBURKE, TR; LIM, B; MARQUEZ, VE; LI, ZH; BOLEN, JB; STEFANOVA, I; HORAK, ID
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The MMAC1 tumor suppressor phosphatase inhibits phospholipase C and integrin-linked kinase-activity
err2000-01-20
err45
PREAI
errMorimoto, AM; Tomlinson, MG; Nakatani, K; Bolen, JB; Roth, RA; Herbst, R
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Reconstitution of Btk signaling by the atypical Tec family tyrosine kinases Bmx and Txk
err1999-05-01
err58
errOAAI
errTomlinson, MG; Kurosaki, T; Berson, AE; Fujii, GH; Johnston, JK; Bolen, JB
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Paired immunoglobulin-like receptor B (PIR-B) inhibits BCR-induced activation of Syk and Btk by SHP-1
err1999-04-08
err142
errOAAI
errMaeda, A; Scharenberg, AM; Tsukada, S; Bolen, JB; Kinet, JP; Kurosaki, T
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Phenotypic analysis of human glioma cells expressing the MMAC1 tumor suppressor phosphatase表达MMAC1肿瘤抑制磷酸酶的人神经胶质瘤细胞的表型分析
err1999-02-16
err34
PREAI
errMorimoto, AM; Berson, AE; Fujii, GH; Teng, DHF; Tavtigian, SV; Bookstein, R; Steck, PA; Bolen, JB
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Signaling pathways controlling trophoblast cell differentiation: Src family protein tyrosine kinases in the rat
err1997-12-01
err23
errOAAI
errKamei, T; Hamlin, GP; Chapman, BM; Burkhardt, AL; Bolen, JB; Soares, MJ
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