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Nanomolar inhibitor of the galectin-8 N-terminal domain binds via a non-canonical cation-π interaction (vol 8, 59, 2025) Galectin-8 N末端域的纳摩尔级抑制剂的结合是通过非经典阳离子-π相互作用实现的(卷8,59,2025) Puric, Edvin; Hassan, Mujtaba; Sjovall, Fredrik; Tomasic, Tihomir; Pevec, Mojca; Lah, Jurij; Forteza, Jaume Adrover; Sundin, Anders; Leffler, Hakon; Nilsson, Ulf J.; Logan, Derek T.; Anderluh, Marko 分享 收藏
Nanomolar inhibitor of the galectin-8 N-terminal domain binds via a non-canonical cation-π interaction Puric, Edvin; Hassan, Mujtaba; Sjovall, Fredrik; Tomasic, Tihomir; Pevec, Mojca; Lah, Jurij; Forteza, Jaume Adrover; Sundin, Anders; Leffler, Hakon; Nilsson, Ulf J.; Logan, Derek T.; Anderluh, Marko 分享 收藏
Elevated Galectin-3 levels in the tumor microenvironment of ovarian cancer - implication of ROS mediated suppression of NK cell antitumor response via tumor-associated neutrophils Karlsson, Veronika; Stal, Ebba; Stoopendahl, Emma; Ivarsson, Anton; Leffler, Hakon; Lycke, Maria; Sundqvist, Martina; Sundfeldt, Karin; Christenson, Karin; Bernson, Elin 分享 收藏
Development and Characterization of a High-Affinity Selective Galectin-3 Mouse Tool Compound in Mouse Models of Cancer Peterson, Kristoffer; Nilsson, Ulf J.; Gravelle, Lise; Holyer, Ian; Jansson, Karl; Kahl-Knutson, Barbro; Leffler, Hakon; Mackinnon, Alison C.; Roper, James A.; Slack, Robert J.; von Wachenfeldt, Henrik; Pedersen, Anders; Zetterberg, Fredrik R. 分享 收藏
Effect of GB1107, a novel galectin-3 inhibitor on pro-fibrotic signalling in the liver Mackinnon, Alison C.; Humphries, Duncan C.; Herman, Kimberley; Roper, James A.; Holyer, Ian; Mabbitt, Joseph; Mills, Ross; Nilsson, Ulf J.; Leffler, Hakon; Pedersen, Anders; Schambye, Hans; Zetterberg, Fredrik; Slack, Robert J. 分享 收藏
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Galectin-8N-Selective 4-Halophenylphthalazinone-Galactals Double π-Stack in a Unique Pocket van Klaveren, Sjors; Hassan, Mujtaba; Hakansson, Maria; Johnsson, Richard E.; Larsson, Jessica; Jakopin, Ziga; Anderluh, Marko; Leffler, Hakon; Tomasic, Tihomir; Nilsson, Ulf J. 分享 收藏
Discovery of the Selective and Orally Available Galectin-1 Inhibitor GB1908 as a Potential Treatment for Lung Cancer 发现选择性和口服Galectin-1抑制剂GB1908作为肺癌的潜在治疗方法 Zetterberg, Fredrik R.; Peterson, Kristoffer; Nilsson, Ulf J.; Dahlgren, Kajsa Andreasson; Diehl, Carl; Holyer, Ian; Hakansson, Maria; Khabut, Areej; Kahl-Knutson, Barbro; Leffler, Hakon; MacKinnon, Alison C.; Roper, James A.; Slack, Robert J.; Zarrizi, Reihaneh; Pedersen, Anders 分享 收藏
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Novel inhibitory effect of galectin-3 on the respiratory burst induced by Staphylococcus aureus in human neutrophils Venkatakrishnan, Vignesh; Elmwall, Jonas; Lahiri, Trisha; Sundqvist, Martina; Bergqvist, Linda; Leffler, Hakon; Nilsson, Ulf J.; Welin, Amanda; Bylund, Johan; Karlsson-Bengtsson, Anna 分享 收藏
Correction to: Galectin-3, a novel endogenous TREM2 ligand, detrimentally regulates inflammatory response in Alzheimer's disease (vol 138, pg 251, 2019) 修正为: Galectin-3,一种新型的内源性TREM2配体,对阿尔茨海默氏病的炎症反应产生不利的调节作用 (138卷,251页,2019页) Boza-Serrano, Antonio; Ruiz, Rocio; Sanchez-Varo, Raquel; Garcia-Revilla, Juan; Yang, Yiyi; Jimenez-Ferrer, Itzia; Paulus, Agnes; Wennstroem, Malin; Vilalta, Anna; Allendorf, David; Davila, Jose Carlos; Stegmayr, John; Jimenez, Sebastian; Roca-Ceballos, Maria A.; Navarro-Garrido, Victoria; Swanberg, Maria; Hsieh, Christine L.; Real, Luis M.; Englund, Elisabet; Linse, Sara; Leffler, Hakon; Nilsson, Ulf J.; Brown, Guy C.; Gutierrez, Antonia; Vitorica, Javier; Venero, Jose Luis; Deierborg, Tomas 分享 收藏
Increased Galectin-9 Levels Correlate with Disease Activity in Patients with DMARD-Naive Rheumatoid Arthritis and Modulate the Secretion of MCP-1 and IL-6 from Synovial Fibroblasts Galectin-9水平升高与DMARD初治类风湿性关节炎患者的疾病活动相关,并调节滑膜成纤维细胞MCP-1和IL-6的分泌 Nielsen, Morten A. A.; Koster, Ditte; Mehta, Akul Y. Y.; Stengaard-Pedersen, Kristian; Busson, Pierre; Junker, Peter; Horslev-Petersen, Kim; Hetland, Merete Lund; ostergaard, Mikkel; Hvid, Malene; Leffler, Hakon; Kragstrup, Tue W. W.; Cummings, Richard D. D.; Deleuran, Bent 分享 收藏
Discovery and Optimization of the First Highly Effective and Orally Available Galectin-3 Inhibitors for Treatment of Fibrotic Disease 用于治疗纤维化疾病的首个高效且可口服的Galectin-3抑制剂的发现和优化 Zetterberg, Fredrik R.; MacKinnon, Alison; Brimert, Thomas; Gravelle, Lise; Johnsson, Richard E.; Kahl-Knutson, Barbro; Leffler, Hakon; Nilsson, Ulf J.; Pedersen, Anders; Peterson, Kristoffer; Roper, James A.; Schambye, Hans; Slack, Robert J.; Tantawi, Susan 分享 收藏
Galectin-9 Signaling Drives Breast Cancer Invasion through Extracellular Matrix Galectin-9信号通过细胞外基质驱动乳腺癌侵袭 Pally, Dharma; Banerjee, Mallar; Hussain, Shahid; Kumar, Rekha, V; Petersson, Alexandra; Rosendal, Ebba; Gunnarsson, Ludvig; Peterson, Kristoffer; Leffler, Hakon; Nilsson, Ulf J.; Bhat, Ramray 分享 收藏
Novel Selective Galectin-3 Antagonists Are Cytotoxic to Acute Lymphoblastic Leukemia 新型选择性Galectin-3拮抗剂对急性淋巴细胞白血病具有细胞毒性 Bum-Erdene, Khuchtumur; Collins, Patrick M.; Hugo, Matthew W.; Tarighat, Somayeh S.; Fei, Fei; Kishor, Chandan; Leffler, Hakon; Nilsson, Ulf J.; Groffen, John; Grice, I. Darren; Heisterkamp, Nora; Blanchard, Helen 分享 收藏