未登录Discovery of a Novel Potent and Selective HSD17B13 Inhibitor, BI-3231, a Well-Characterized Chemical Probe Available for Open Science
Thamm, Sven; Willwacher, Marina K.; Aspnes, Gary E.; Bretschneider, Tom; Brown, Nicholas F.; Buschbom-Helmke, Silke; Veser, Thomas; Gargano, Emanuele M.; Grabowski, Daniel; Hoenke, Christoph; Matera, Damian; Mueck, Katja; Peters, Stefan; Reindl, Sophia; Riether, Doris; Schmid, Matthias; Tautermann, Christofer S.; Teitelbaum, Aaron M.; Truenkle, Cornelius; Winter, Martin; Fox, Thomas; Wortmann, Lars
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收藏Allosteric Activation of Striatal-Enriched Protein Tyrosine Phosphatase (STEP, PTPN5) by a Fragment-like Molecule
Tautermann, Christofer S.; Binder, Florian; Buettner, Frank H.; Eickmeier, Christian; Fiegen, Dennis; Gross, Ulrike; Grundl, Marc A.; Heilker, Ralf; Hobson, Scott; Hoerer, Stefan; Luippold, Andreas; Mack, Volker; Montel, Florian; Peters, Stefan; Bhattacharya, Supriyo; Vaidehi, Nagarajan; Schnapp, Gisela; Thamm, Sven; Zeeb, Markus
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收藏Sequential C-H Arylation and Enantioselective Hydrogenation Enables Ideal Asymmetric Entry to the Indenopiperidine Core of an 11β-HSD-1 Inhibitor
Wei, Xudong; Qu, Bo; Zeng, Xingzhong; Savoie, Jolaine; Fandrick, Keith R.; Desrosiers, Jean -Nicolas; Tcyrulnikov, Sergei; Marsini, Maurice A.; Buono, Frederic G.; Li, Zhibin; Yang, Bing-Shiou; Tang, Wenjun; Haddad, Nizar; Gutierrez, Osvaldo; Wang, Jun; Lee, Heewon; Ma, Shengli; Campbell, Scot; Lorenz, Jon C.; Eckhardt, Matthias; Himmelsbach, Frank; Peters, Stefan; Patel, Nitinchandra D.; Tan, Zhulin; Yee, Nathan K.; Song, Jinhua J.; Roschangar, Frank; Kozlowski, Marisa C.; Senanayake, Chris H.
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收藏Lymphohematopoietic stem cell engraftment
Quesenberry, PJ; Stewart, FM; Zhong, SJ; Habibiani, H; McAuliffe, C; Reilly, J; Carlson, J; Dooner, M; Nilsson, S; Peters, S; Stein, G; Stein, J; Emmons, R; Benoit, B; Bertoncello, I; Becker, P
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