Jitendar Reddy

AstraZeneca

H指数:17

被引数:1,148

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Evaluating the Impact of CYP1A2 Inhibition on the Pharmacokinetics of Savolitinib: A Phase 1 Open-Label Study

评价CYP1A2抑制对 savolitinib 药代动力学的影响：一项 1 期开放标签研究

Pharmacology Research & Perspectives

IF2.3

2026-09-250

OAAI

Bioequivalence of budesonide/glycopyrrolate/formoterol fumarate with a next-generation propellant versus hydrofluoroalkane-134a in healthy adults: phase I, randomized, double-blind, single-dose, partial-replicate, three-way cross-over lung exposure and total systemic exposure studies

布地奈德/格隆溴铵/富马酸福莫特罗的生物等效性研究：与新一代推进剂相比氢氟烷烃-134a在健康成年人中的相I、随机、双盲、单剂量、部分重复、三向交叉肺暴露和全身总暴露研究

Therapeutic Advances in Respiratory Disease

IF3

2026-02-120

PRE

Discovery of Imidazo[1,2-a]pyridine Ethers and Squaramides as Selective and Potent Inhibitors of Mycobacterial Adenosine Triphosphate (ATP) Synthesis

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2017-02-0395

PREAI

Tantry, Subramanyam J.; Markad, Shankar D.; Shinde, Vikas; Bhat, Jyothi; Balakrishnan, Gayathri; Gupta, Amit K.; Ambady, Anisha; Raichurkar, Anandkumar; Kedari, Chaitanyakumar; Sharma, Sreevalli; Mudugal, Naina V.; Narayan, Ashwini; Kumar, C. N. Naveen; Nanduri, Robert; Bharath, Sowmya; Reddy, Jitendar; Panduga, Vijender; Prabhakar, K. R.; Kandaswamy, Karthikeyan; Saralaya, Ramanatha; Kaur, Parvinder; Dinesh, Neela; Guptha, Supreeth; Rich, Kirsty; Murray, David; Plant, Helen; Preston, Marian; Ashton, Helen; Plant, Darren; Walsh, Jarrod; Alcock, Peter; Naylor, Kathryn; Collier, Matthew; Whiteaker, James; McLaughlin, Robert E.; Mallya, Meenakshi; Panda, Manoranjan; Rudrapatna, Suresh; Ramachandran, Vasanthi; Shandil, Radha; Sambandamurthy, Vasan K.; Mdluli, Khisi; Cooper, Christopher B.; Rubin, Harvey; Yano, Takahiro; Iyer, Pravin; Narayanan, Shridhar; Kavanagh, Stefan; Mukherjee, Kakoli; Balasubramanian, V.; Hosagrahara, Vinayak P.; Solapure, Suresh; Ravishankar, Sudha; Hameed, Shahul P.

In Silico-Based High-Throughput Screen for Discovery of Novel Combinations for Tuberculosis Treatment

ANTIMICROBIAL AGENTS AND CHEMOTHERAPY

IF4.5

2015-09-019

OAAI

Triaminopyrimidine is a fast-killing and long-acting antimalarial clinical candidate

NATURE COMMUNICATIONS

IF15.7

2015-03-3161

OAAI

Hameed, Shahul P.; Solapure, Suresh; Patil, Vikas; Henrich, Philipp P.; Magistrado, Pamela A.; Bharath, Sowmya; Murugan, Kannan; Viswanath, Pavithra; Puttur, Jayashree; Srivastava, Abhishek; Bellale, Eknath; Panduga, Vijender; Shanbag, Gajanan; Awasthy, Disha; Landge, Sudhir; Morayya, Sapna; Koushik, Krishna; Saralaya, Ramanatha; Raichurkar, Anandkumar; Rautela, Nikhil; Choudhury, Nilanjana Roy; Ambady, Anisha; Nandishaiah, Radha; Reddy, Jitendar; Prabhakar, K. R.; Menasinakai, Sreenivasaiah; Rudrapatna, Suresh; Chatterji, Monalisa; Belen Jimenez-Diaz, Maria; Santos Martinez, Maria; Maria Sanz, Laura; Coburn-Flynn, Olivia; Fidock, David A.; Lukens, Amanda K.; Wirth, Dyann F.; Bandodkar, Balachandra; Mukherjee, Kakoli; McLaughlin, Robert E.; Waterson, David; Rosenbrier-Ribeiro, Lyn; Hickling, Kevin; Balasubramanian, V.; Warner, Peter; Hosagrahara, Vinayak; Dudley, Adam; Iyer, Pravin S.; Narayanan, Shridhar; Kavanagh, Stefan; Sambandamurthy, Vasan K.

1,4-Azaindole, a Potential Drug Candidate for Treatment of Tuberculosis

ANTIMICROBIAL AGENTS AND CHEMOTHERAPY

IF4.5

2014-09-0197

OAAI

Optimization of Pyrrolamides as Mycobacterial GyrB ATPase Inhibitors: Structure-Activity Relationship and In Vivo Efficacy in a Mouse Model of Tuberculosis (vol 58, pg 61, 2014)

ANTIMICROBIAL AGENTS AND CHEMOTHERAPY

IF4.5

2014-08-013

OAAI

Hameed, Shahul P.; Solapure, Suresh; Mukherjee, Kakoli; Nandi, Vrinda; Waterson, David; Shandil, Radha; Balganesh, Meenakshi; Sambandamurthy, Vasan K.; Raichurkar, Anand Kumar; Deshpande, Abhijeet; Ghosh, Anirban; Awasthy, Disha; Shanbhag, Gajanan; Sheikh, Gulebahar; McMiken, Helen; Puttur, Jayashree; Reddy, Jitendar; Werngren, Jim; Read, Jon; Kumar, Mahesh; Manjunatha, R.; Chinnapattu, Murugan; Madhavapeddi, Prashanti; Manjrekar, Praveena; Basu, Reetobrata; Gaonkar, Sheshagiri; Sharma, Sreevalli; Hoffner, Sven; Humnabadkar, Vaishali; Subbulakshmi, Venkita; Panduga, Vijender

N-Aryl-2-aminobenzimidazoles: Novel, Efficacious, Antimalarial Lead Compounds

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2014-07-2138

PREAI

Ramachandran, Sreekanth; Hameed, Shahul P.; Srivastava, Abhishek; Shanbhag, Gajanan; Morayya, Sapna; Rautela, Nikhil; Awasthy, Disha; Kavanagh, Stefan; Bharath, Sowmya; Reddy, Jitendar; Panduga, Vijender; Prabhakar, K. R.; Saralaya, Ramanatha; Nanduri, Robert; Raichurkar, Anandkumar; Menasinakai, Sreenivasaiah; Achar, Vijayashree; Belen Jimenez-Diaz, Maria; Santos Martinez, Maria; Angulo-Barturen, Inigo; Ferrer, Santiago; Maria Sanz, Laura; Javier Gamo, Francisco; Duffy, Sandra; Avery, Vicky M.; Waterson, David; Lee, Marcus C. S.; Coburn-Flynn, Olivia; Fidock, David A.; Iyer, Pravin S.; Narayanan, Shridhar; Hosagrahara, Vinayak; Sambandamurthy, Vasan K.

Lead Optimization of 1,4-Azaindoles as Antimycobacterial Agents

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2014-06-2077

PREAI

Shirude, Pravin S.; Shandil, Radha K.; Manjunatha, M. R.; Sadler, Claire; Panda, Manoranjan; Panduga, Vijender; Reddy, Jitendar; Saralaya, Ramanatha; Nanduri, Robert; Ambady, Anisha; Ravishankar, Sudha; Sambandamurthy, Vasan K.; Humnabadkar, Vaishali; Jena, Lalit K.; Suresh, Rudrapatna S.; Srivastava, Abhishek; Prabhakar, K. R.; Whiteaker, James; McLaughlin, Robert E.; Sharma, Sreevalli; Cooper, Christopher B.; Mdluli, Khisi; Butler, Scott; Iyer, Pravin S.; Narayanan, Shridhar; Chatterji, Monalisa

4-Aminoquinolone Piperidine Amides: Noncovalent Inhibitors of DprE1 with Long Residence Time and Potent Antimycobacterial Activity

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2014-06-1186

PREAI

Naik, Maruti; Humnabadkar, Vaishali; Tantry, Subramanyam J.; Panda, Manoranjan; Narayan, Ashwini; Guptha, Supreeth; Panduga, Vijender; Manjrekar, Praveena; Jena, Lalit Kumar; Koushik, Krishna; Shanbhag, Gajanan; Jatheendranath, Sandesh; Manjunatha, M. R.; Gorai, Gopinath; Bathula, Chandramohan; Rudrapatna, Suresh; Achar, Vijayashree; Sharma, Sreevalli; Ambady, Anisha; Hegde, Naina; Mahadevaswamy, Jyothi; Kaur, Parvinder; Sambandamurthy, Vasan K.; Awasthy, Disha; Narayan, Chandan; Ravishankar, Sudha; Madhavapeddi, Prashanti; Reddy, Jitendar; Prabhakar, K. R.; Saralaya, Ramanatha; Chatterji, Monalisa; Whiteaker, James; McLaughlin, Bob; Chiarelli, Laurent R.; Riccardi, Giovanna; Pasca, Maria Rosalia; Binda, Claudia; Neres, Joao; Dhar, Neeraj; Signorino-Gelo, Francois; McKinney, John D.; Ramachandran, Vasanthi; Shandil, Radha; Tommasi, Ruben; Iyer, Pravin S.; Narayanan, Shridhar; Hosagrahara, Vinayak; Kavanagh, Stefan; Dinesh, Neela; Ghorpade, Sandeep R.

Benzimidazoles: Novel Mycobacterial Gyrase Inhibitors from Scaffold Morphing

苯并咪唑: 来自支架变形的新型分枝杆菌促旋酶抑制剂

ACS MEDICINAL CHEMISTRY LETTERS

IF4

2014-06-0552

OAAI

Novel N-Linked Aminopiperidine-Based Gyrase Inhibitors with Improved hERG and in Vivo Efficacy against Mycobacterium tuberculosis

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2014-05-2349

PREAI

Hameed, Shahul P.; Patil, Vikas; Solapure, Suresh; Sharma, Umender; Madhavapeddi, Prashanti; Raichurkar, Anandkumar; Chinnapattu, Murugan; Manjrekar, Praveena; Shanbhag, Gajanan; Puttur, Jayashree; Shinde, Vikas; Menasinakai, Sreenivasaiah; Rudrapatana, Suresh; Achar, Vijayashree; Awasthy, Disha; Nandishaiah, Radha; Humnabadkar, Vaishali; Ghosh, Anirban; Narayan, Chandan; Ramya, V. K.; Kaur, Parvinder; Sharma, Sreevalli; Werngren, Jim; Hoffner, Sven; Panduga, Vijender; Kumar, C. N. Naveen; Reddy, Jitendar; Kumar, Mahesh K. N.; Ganguly, Samit; Bharath, Sowmya; Bheemarao, Ugarkar; Mukherjee, Kakoli; Arora, Uma; Gaonkar, Sheshagiri; Coulson, Michelle; Waterson, David; Sambandamurthy, Vasan K.; de Sousa, Sunita M.

Optimization of Pyrrolamides as Mycobacterial GyrB ATPase Inhibitors: Structure-Activity Relationship and In Vivo Efficacy in a Mouse Model of Tuberculosis

ANTIMICROBIAL AGENTS AND CHEMOTHERAPY

IF4.5

2014-01-0140

OAAI

Azaindoles: Noncovalent DprE1 Inhibitors from Scaffold Morphing Efforts, Kill Mycobacterium tuberculosis and Are Efficacious in Vivo

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2013-11-21139

PREAI

Shirude, Pravin S.; Shandil, Radha; Sadler, Claire; Naik, Maruti; Hosagrahara, Vinayak; Hameed, Shahul; Shinde, Vikas; Bathula, Chandramohan; Humnabadkar, Vaishali; Kumar, Naveen; Reddy, Jitendar; Panduga, Vijender; Sharma, Sreevalli; Ambady, Anisha; Hegde, Naina; Whiteaker, James; McLaughlin, Robert E.; Gardner, Humphrey; Madhavapeddi, Prashanti; Ramachandran, Vasanthi; Kaur, Parvinder; Narayan, Ashwini; Guptha, Supreeth; Awasthy, Disha; Narayan, Chandan; Mahadevaswamy, Jyothi; Vishwas, K. G.; Ahuja, Vijaykamal; Srivastava, Abhishek; Prabhakar, K. R.; Bharath, Sowmya; Kale, Ramesh; Ramaiah, Manjunatha; Choudhury, Nilanjana Roy; Sambandamurthy, Vasan K.; Solapure, Suresh; Iyer, Pravin S.; Narayanan, Shridhar; Chatterji, Monalisa

Thiazolopyridine Ureas as Novel Antitubercular Agents Acting through Inhibition of DNA Gyrase B

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2013-10-1861

PREAI

Kale, Manoj G.; Raichurkar, Anandkumar; Hameed, Shahul P.; Waterson, David; McKinney, David; Manjunatha, M. R.; Kranthi, Usha; Koushik, Krishna; Jena, Lalit Kumar; Shinde, Vikas; Rudrapatna, Suresh; Barde, Shubhada; Humnabadkar, Vaishali; Madhavapeddi, Prashanti; Basavarajappa, Halesha; Ghosh, Anirban; Ramya, V. K.; Guptha, Supreeth; Sharma, Sreevalli; Vachaspati, Prakash; Kumar, K. N. Mahesh; Giridhar, Jayashree; Reddy, Jitendar; Panduga, Vijender; Ganguly, Samit; Ahuja, Vijaykamal; Gaonkar, Sheshagiri; Kumar, C. N. Naveen; Ogg, Derek; Tucker, Julie A.; Boriack-Sjodin, P. Ann; de Sousa, Sunita M.; Sambandamurthy, Vasan K.; Ghorpade, Sandeep R.

In Vitro and In Vivo Efficacy of β-Lactams against Replicating and Slowly Growing/Nonreplicating Mycobacterium tuberculosis

ANTIMICROBIAL AGENTS AND CHEMOTHERAPY

IF4.5

2013-06-0170

OAAI

Effect of repeated dosing on rifampin exposure in BALB/c mice

EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES

IF4.7

2013-04-0116

PREAI

Fast mouse PK (Fast PK): A rapid screening method to increase pharmacokinetic throughput in pre-clinical drug discovery

EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES