未登录 Design, Synthesis, and Biological Evaluation of the Novel Neutrophil Elastase Inhibitor CHF-6333 for the Inhaled Treatment of Bronchiectasis 新型中性粒细胞弹性蛋白酶抑制剂CHF-6333的设计、合成及生物活性评价:用于支气管扩张的吸入治疗 Armani, Elisabetta; Rizzi, Andrea; Miglietta, Daniela; Bassanetti, Irene; Amadei, Francesco; Brogin, Giandomenico; Capaldi, Carmelida; Rancati, Fabio; Carnini, Chiara; Fernandez, Sergio Xanxo; Civelli, Maurizio; Puccini, Paola; Bellini, Marta; Jennings, Andrew; Heald, Robert A.; Alcaraz, Lilian; Sutton, Jonathan M.; Finch, Harry; Fitzgerald, Mary; Fox, Craig; Villetti, Gino 分享 收藏
Design, Synthesis, and Biological Characterization of Inhaled p38?/? MAPK Inhibitors for the Treatment of Lung Inflammatory Diseases Armani, Elisabetta; Capaldi, Carmelida; Bagnacani, Valentina; Saccani, Francesca; Aquino, Giancarlo; Puccini, Paola; Facchinetti, Fabrizio; Martucci, Cataldo; Moretto, Nadia; Villetti, Gino; Patacchini, Riccardo; Civelli, Maurizio; Hurley, Chris; Jennings, Andrew; Alcaraz, Lilian; Bloomfield, Dawn; Briggs, Michael; Daly, Stephen; Panchal, Terry; Russell, Vince; Wicks, Sharon; Finch, Harry; Fitzgerald, Mary; Fox, Craig; Delcanale, Maurizio 分享 收藏
Conformational Sampling of Macrocyclic Drugs in Different Environments: Can We Find the Relevant Conformations? 大环药物在不同环境中的构象取样: 我们能找到相关的构象吗? Poongavanam, Vasanthanathan; Danelius, Emma; Peintner, Stefan; Alcaraz, Lilian; Caron, Giulia; Cummings, Maxwell D.; Wlodek, Stanislaw; Erdelyi, Mate; Hawkins, Paul C. D.; Ermondi, Giuseppe; Kihlberg, Jan 分享 收藏
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Discovery of AZD3199, An Inhaled Ultra long Acting β2 Receptor Agonist with Rapid Onset of Action Stocks, Michael J.; Alcaraz, Lilian; Bailey, Andrew; Bonnert, Roger; Cadogan, Elaine; Christie, Jadeen; Dixon, John; Connolly, Stephen; Cook, Anthony; Fisher, Adrian; Flaherty, Alice; Humphries, Alexander; Ingall, Anthony; Jordan, Stephen; Lawson, Mandy; Mullen, Alex; Nicholls, David; Paine, Stuart; Pairaudeau, Garry; Young, Alan 分享 收藏
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Discovery of potent and selective adamantane-based small-molecule P2X7 receptor antagonists/interleukin-1β,6 inhibitors Furber, Mark; Alcaraz, Lilian; Bent, Janice E.; Beyerbach, Armin; Bowers, Keith; Braddock, Martin; Caffrey, Moya V.; Cladingboel, David; Collington, John; Donald, David K.; Fagura, Malbinder; Ince, Frank; Kinchin, Elizabeth C.; Laurent, Celine; Lawson, Mandy; Luker, Timothy J.; Mortimore, Michael M. P.; Pimm, Austen D.; Riley, Robert J.; Roberts, Nicola; Robertson, Mark; Theaker, Jill; Thorne, Philip V.; Weaver, Richard; Webborn, Peter; Willis, Paul 分享 收藏
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