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High-Throughput Screen for Inhibitors of Klebsiella pneumoniae Virulence Using a Tetrahymena pyriformis Co-Culture Surrogate Host Model Woods, Angela L.; Parker, David; Glick, Meir M.; Peng, Yunshan; Lenoir, Francois; Mulligan, Evan; Yu, Vincent; Piizzi, Grazia; Lister, Troy; Lilly, Maria-Dawn; Dzink-Fox, Joann; Jansen, Johanna M.; Ryder, Neil S.; Dean, Charles R.; Smith, Thomas M. 分享 收藏
Development of a cyclosporin A derivative with excellent anti-hepatitis C virus potency Fu, Jiping; Becker, Christopher; Cao, Li; Capparelli, Michael; Denay, Regis; Fujimoto, Roger; Gai, Yu; Gao, Zhaobo; Guenat, Christian; Karur, Subramanian; Kim, Hongyong; Li, Weikuan; Li, Xiaolin; Li, Wei; Lochmann, Thomas; Lu, Amy; Lu, Peichao; Luneau, Alexandre; Meier, Nicole; Mergo, Wosenu; Ng, Simon; Parker, David; Peng, Yunshan; Riss, Bernard; Rivkin, Alexey; Roggo, Silvio; Schroeder, Harald; Schuerch, Friedrich; Simmons, Robert L.; Sun, Feng; Sweeney, Zachary K.; Tjandra, Meiliana; Wang, Michael; Wang, Ruidong; Weiss, Andrew H.; Wenger, Nicolas; Wu, Quanbing; Xiong, Xin; Xu, Su; Xu, Wenjian; Yifru, Aregahegn; Zhao, Jibin; Zhou, Jianguang; Zurcher, Christian; Gallou, Fabrice 分享 收藏
Design, Synthesis, and Properties of a Potent Inhibitor of Pseudomonas aeruginosa Deacetylase LpxC Piizzi, Grazia; Parker, David T.; Peng, Yunshan; Dobler, Markus; Patnaik, Anup; Wattanasin, Som; Liu, Eugene; Lenoir, Francois; Nunez, Jill; Kerrigan, John; McKenney, David; Osborne, Colin; Yu, Donghui; Lanieri, Leanne; Bojkovic, Jade; Dzink-Fox, Joann; Lilly, Maria-Dawn; Sprague, Elizabeth R.; Lu, Yipin; Wang, Hongming; Ranjitkar, Srijan; Xie, Lili; Wang, Bing; Glick, Meir; Hamann, Lawrence G.; Tommasi, Ruben; Yang, Xia; Dean, Charles R. 分享 收藏
Potent Nonimmunosuppressive Cyclophilin Inhibitors With Improved Pharmaceutical Properties and Decreased Transporter Inhibition Fu, Jiping; Tjandra, Meiliana; Becker, Christopher; Bednarczyk, Dallas; Capparelli, Michael; Elling, Robert; Hanna, Imad; Fujimoto, Roger; Furegati, Markus; Karur, Subramanian; Kasprzyk, Theresa; Knapp, Mark; Leung, Kwan; Li, Xiaolin; Lu, Peichao; Mergo, Wosenu; Miault, Charlotte; Ng, Simon; Parker, David; Peng, Yunshan; Roggo, Silvio; Rivkin, Alexey; Simmons, Robert L.; Wang, Michael; Wiedmann, Brigitte; Weiss, Andrew H.; Xiao, Linda; Xie, Lili; Xu, Wenjian; Yifru, Aregahegn; Yang, Shengtian; Zhou, Bo; Sweeney, Zachary K. 分享 收藏
Improved Syntheses of 5′-S-(2-Aminoethyl)-6-N-(4-nitrobenzyl)-5′-thioadenosine (SAENTA), Analogues, and Fluorescent Probe Conjugates: Analysis of Cell-Surface Human Equilibrative Nucleoside Transporter 1 (hENT1) Levels for Prediction of the Antitumor Efficacy of Gemcitabine Robins, Morris J.; Peng, Yunshan; Damaraju, Vijaya L.; Mowles, Delores; Barron, Geraldine; Tackaberry, Tracey; Young, James D.; Cass, Carol E. 分享 收藏
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Residues 334 and 338 in transmembrane segment 8 of human equilibrative nucleoside transporter 1 are important determinants of inhibitor sensitivity, protein folding, and catalytic turnover Visser, Frank; Sun, Lijie; Damaraju, Vijaya; Tackaberry, Tracey; Peng, Yunshan; Robins, Morris J.; Baldwin, Stephen A.; Young, James D.; Cass, Carol E. 分享 收藏