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Suzanne Skolnik

Novartis

13H指数
32论文数
776被引数
收录论文 10
发表时间
Discovery of EGT710; an Oral Nonpeptidomimetic Reversible Covalent SARS-CoV-2 Main Protease InhibitorEGT710的发现:一种口服非肽类拟似可逆共价SARS-CoV-2主蛋白酶抑制剂
err2026-02-09
err0
PREAI
errJulien P. N. Papillon; Jun Yuan; Matthew J. Hesse; Lei Zhang; Richard I. Robinson; Nathaniel F. Ware; Viktor Hornak; Rajeshri G. Karki; Tom Kirrane; Keira Garland; Sajan Joseph; Stephanie A. Moquin; Suresh B. Lakshminarayana; Laura Tandeske; Dustin Dovala; Mark Knapp; Elizabeth Ornelas; Daniel Fuller; Pei-i Ho; Xuping Xie; Katarina Vulic; Suzanne M. Skolnik; Jinhai Gao; Mark Zambrowski; Meike Spiess; José S. Duca; Scott A. Busby; Markus Schirle; Michael Robinson; Pei-Yong Shi; Heinz E. Moser; Christopher Sarko; James E. Bradner; Thierry T. Diagana; John A. Tallarico
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Paradoxical Increase of Permeability and Lipophilicity with the Increasing Topological Polar Surface Area within a Series of PRMT5 Inhibitors
err2022-09-07
err8
PREAI
errArgikar, Upendra; Blatter, Markus; Bednarczyk, Dallas; Chen, Zhuoliang; Cho, Young Shin; Dore, Michael; Dumouchel, Jennifer L.; Ho, Samuel; Hoegenauer, Klemens; Kawanami, Toshio; Mathieu, Simon; Meredith, Erik; Moebitz, Henrik; Murphy, Stephen K.; Parthasarathy, Saravanan; Soldermann, Carole Pissot; Santos, Jobette; Silver, Serena; Skolnik, Suzanne; Stojanovic, Aleksandar
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Discovery solubility measurement and assessment of small molecules with drug development in mind
err2022-05-01
err40
PREAI
errBarrett, Jaclyn A.; Yang, Wenzhan; Skolnik, Suzanne M.; Belliveau, Lisa M.; Patros, Kellyn M.
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Prediction of pKa Using Machine Learning Methods with Rooted Topological Torsion Fingerprints: Application to Aliphatic Amines
err2019-10-24
err29
PREAI
errLu, Yipin; Anand, Shankara; Shirley, William; Gedeck, Peter; Kelley, Brian P.; Skolnik, Suzanne; Rodde, Stephane; Mai Nguyen; Lindvall, Mika; Jia, Weiping
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Benefit of Retraining pKa Models Studied Using Internally Measured Data
err2015-06-29
err19
PREAI
errGedeck, Peter; Lu, Yipin; Skolnik, Suzanne; Rodde, Stephane; Dollinger, Gavin; Jia, Weiping; Berellin, Giuliano; Vianello, Riccardo; Faller, Bernard; Lombardo, Franco
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Imidazolopiperazines: Lead Optimization of the Second-Generation Antimalarial Agents
err2012-04-23
err90
errOAAI
errNagle, Advait; Wu, Tao; Kuhen, Kelli; Gagaring, Kerstin; Borboa, Rachel; Francek, Caroline; Chen, Zhong; Plouffe, David; Lin, Xuena; Caldwell, Christopher; Ek, Jared; Skolnik, Suzanne; Liu, Fenghua; Wang, Jianling; Chang, Jonathan; Li, Chun; Liu, Bo; Hollenbeck, Thomas; Tuntland, Tove; Isbell, John; Chuan, Tiffany; Alper, Philip B.; Fischli, Christoph; Brun, Reto; Lakshminarayana, Suresh B.; Rottmann, Matthias; Diagana, Thierry T.; Winzeler, Elizabeth A.; Glynne, Richard; Tully, David C.; Chatterjee, Arnab K.
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Optimization of the in Vitro Cardiac Safety of Hydroxamate-Based Histone Deacetylase Inhibitors
err2011-06-17
err66
PREAI
errShultz, Michael D.; Cao, Xueying; Chen, Christine H.; Cho, Young Shin; Davis, Nicole R.; Eckman, Joe; Fan, Jianmei; Fekete, Alex; Firestone, Brant; Flynn, Julie; Green, Jack; Growney, Joseph D.; Holmqvist, Mats; Hsu, Meier; Jansson, Daniel; Jiang, Lei; Kwon, Paul; Liu, Gang; Lombardo, Franco; Lu, Qiang; Majumdar, Dyuti; Meta, Christopher; Perez, Lawrence; Pu, Minying; Ramsey, Tim; Remiszewski, Stacy; Skolnik, Suzanne; Traebert, Martin; Urban, Laszlo; Uttamsingh, Vinita; Wang, Ping; Whitebread, Steven; Whitehead, Lewis; Yan-Neale, Yan; Yao, Yung-Mae; Zhou, Liping; Atadja, Peter
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Imidazolopiperazines: Hit to Lead Optimization of New Antimalarial Agents
err2011-06-06
err99
errOAAI
errWu, Tao; Nagle, Advait; Kuhen, Kelli; Gagaring, Kerstin; Borboa, Rachel; Francek, Caroline; Chen, Zhong; Plouffe, David; Goh, Anne; Lakshminarayana, Suresh B.; Wu, Jeanette; Ang, Hui Qing; Zeng, Peiting; Kang, Min Low; Tan, William; Tan, Maria; Ye, Nicole; Lin, Xuena; Caldwell, Christopher; Ek, Jared; Skolnik, Suzanne; Liu, Fenghua; Wang, Jianling; Chang, Jonathan; Li, Chun; Hollenbeck, Thomas; Tuntland, Tove; Isbell, John; Fischli, Christoph; Brun, Reto; Rottmann, Matthias; Dartois, Veronique; Keller, Thomas; Diagana, Thierry; Winzeler, Elizabeth; Glynne, Richard; Tully, David C.; Chatterjee, Arnab K.
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Towards Prediction of In Vivo Intestinal Absorption Using a 96-Well Caco-2 Assay
err2010-07-01
err123
PREAI
errSkolnik, Suzanne; Lin, Xuena; Wang, Jianling; Chen, Xiao-Hui; He, Timothy; Zhang, Bailin
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