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Florian Lesage

universite cote d'azur and inserm and cnrs

63H指数
168论文数
1.6W被引数
收录论文 77
发表时间
SPARC: a Structural Pathogenicity Algorithm for Risk Classification of hERG Variants
err2025-12-25
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errFrank C Chatelain; Barbara Ribeiro de Oliveira; Guillaume Grataloup; Noé Robert; Malak Alameh; Aurélie Thollet; Jérôme Montnach; Sylvain Feliciangeli; Aline Rio; Floriane Bibault; Delphine Bichet; Olivier Bignucolo; Fabrice Extramiana; Rupamanjari Majumder; Jean-Jacques Schott; Vincent Probst; Isabelle Denjoy; Florian Lesage; Gildas Loussouarn; Michel De Waard
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Mechanistic basis of the dynamic response of TWIK1 ionic selectivity to pH
err2024-05-08
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errChatelain, Franck C.; Gilbert, Nicolas; Bichet, Delphine; Jauch, Annaise; Feliciangeli, Sylvain; Lesage, Florian; Bignucolo, Olivier
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Predicting hERG repolarization power at 37°C from recordings at room temperature
err2023-05-18
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errOliveira-Mendes, Barbara B. R.; Alameh, Malak; Montnach, Jerome; Ollivier, Beatrice; Gibaud, Solene; Feliciangeli, Sylvain; Lesage, Florian; Charpentier, Flavien; Loussouarn, Gildas; De Waard, Michel; Baro, Isabelle
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A photoswitchable inhibitor of TREK channels controls pain in wild-type intact freely moving animals
err2023-03-01
err6
errOAAI
errLandra-Willm, Arnaud; Karapurkar, Ameya; Duveau, Alexia; Chassot, Anne Amandine; Esnault, Lucille; Callejo, Gerard; Bied, Marion; Hafner, Stephanie; Lesage, Florian; Wdziekonski, Brigitte; Baron, Anne; Fossat, Pascal; Marsollier, Laurent; Gasull, Xavier; Boue-Grabot, Eric; Kienzler, Michael A.; Sandoz, Guillaume
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A need for exhaustive and standardized characterization of ion channels activity. The case of KV11.1
err2023-02-13
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errAlameh, Malak; Oliveira-Mendes, Barbara Ribeiro; Kyndt, Florence; Rivron, Jordan; Denjoy, Isabelle; Lesage, Florian; Schott, Jean-Jacques; De Waard, Michel; Loussouarn, Gildas
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Alkaline-sensitive two-pore domain potassium channels form functional heteromers in pancreatic β-cells
err2022-10-01
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errKhoubza, Lamyaa; Gilbert, Nicolas; Kim, Eun-Jin; Chatelain, Franck C.; Feliciangeli, Sylvain; Abelanet, Sophie; Kang, Dawon; Lesage, Florian; Bichet, Delphine
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A standardised hERG phenotyping pipeline to evaluate KCNH2 genetic variant pathogenicity
err2021-11-23
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errOliveira-Mendes, Barbara; Feliciangeli, Sylvain; Menard, Melissa; Chatelain, Frank; Alameh, Malak; Montnach, Jerome; Nicolas, Sebastien; Ollivier, Beatrice; Barc, Julien; Baro, Isabelle; Schott, Jean-Jacques; Probst, Vincent; Kyndt, Florence; Denjoy, Isabelle; Lesage, Florian; Loussouarn, Gildas; De Waard, Michel
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Piezo1 and Piezo2 foster mechanical gating of K2P channelsPiezo1和Piezo2促进了K2P通道的机械门控
err2021-11-01
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errGlogowska, Edyta; Arhatte, Malika; Chatelain, Franck C.; Lesage, Florian; Xu, Aimin; Grashoff, Carsten; Discher, Dennis E.; Patel, Amanda; Honore, Eric
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TREK1 channel activation as a new analgesic strategy devoid of opioid adverse effects (vol 177, pg 4782, 2020)
err2020-10-27
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errBusserolles, Jerome; Ben Soussia, Ismail; Poucho, Laetitia; Marie, Nicolas; Melein, Mathieu; Devilliers, Maily; Judon, Celine; Schopp, Julien; Clemenceau, Loic; Poupon, Laura; Chapuy, Eric; Richard, Serge; Noble, Florence; Lesage, Florian; Sylvie, Ducki; Eschalier, Alain; Lolignier, Stephane
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TREK1 channel activation as a new analgesic strategy devoid of opioid adverse effects
err2020-09-21
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errBusserolles, Jerome; Ben Soussia, Ismail; Pouchol, Laetitia; Marie, Nicolas; Meleine, Mathieu; Devilliers, Maily; Judon, Celine; Schopp, Julien; Clemenceau, Loic; Poupon, Laura; Chapuy, Eric; Richard, Serge; Noble, Florence; Lesage, Florian; Ducki, Sylvie; Eschalier, Alain; Lolignier, Stephane
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Inhibition of histone deacetylation rescues phenotype in a mouse model of Birk-Barel intellectual disability syndrome抑制组蛋白去乙酰化可挽救birk-barel智力障碍综合征小鼠模型的表型
err2020-01-24
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errCooper, Alexis; Butto, Tamer; Hammer, Niklas; Jagannath, Somanath; Fend-Guella, Desiree Lucia; Akhtar, Junaid; Radyushkin, Konstantin; Lesage, Florian; Winter, Jennifer; Strand, Susanne; Roeper, Jochen; Zechner, Ulrich; Schweiger, Susann
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Mutation of a single residue promotes gating of vertebrate and invertebrate two-pore domain potassium channels
err2019-02-15
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errBen Soussia, Ismail; El Mouridi, Sonia; Kang, Dawon; Leclercq-Blondel, Alice; Khoubza, Lamyaa; Tardy, Philippe; Zariohi, Nora; Gendrel, Marie; Lesage, Florian; Kim, Eun-Jin; Bichet, Delphine; Andrini, Olga; Boulin, Thomas
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Migraine-Associated TRESK Mutations Increase Neuronal Excitability through Alternative Translation Initiation and Inhibition of TREK
errNEURON
IF15
err2019-01-01
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errRoyal, Perrine; Andres-Bilbe, Alba; Prado, Pablo Avalos; Verkest, Clement; Wdziekonski, Brigitte; Schaub, Sebastien; Baron, Anne; Lesage, Florian; Gasull, Xavier; Levitz, Joshua; Sandoz, Guillaume
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Antagonistic Effect of a Cytoplasmic Domain on the Basal Activity of Polymodal Potassium Channels
err2018-09-04
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errBen Soussia, Ismail; Choveau, Frank S.; Blin, Sandy; Kim, Eun-Jin; Feliciangeli, Sylvain; Chatelain, Franck C.; Kang, Dawon; Bichet, Delphine; Lesage, Florian
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Lack of p11 expression facilitates acidity-sensing function of TASK1 channels in mouse adrenal medullary cells
err2018-07-12
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errInoue, Masumi; Matsuoka, Hidetada; Lesage, Florian; Harada, Keita
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Recombinant tandem of pore-domains in a Weakly Inward rectifying K+ channel 2 (TWIK2) forms active lysosomal channels
err2017-04-05
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errBobak, Nicole; Feliciangeli, Sylvain; Chen, Cheng-Chang; Ben Soussia, Ismail; Bittner, Stefan; Pagnotta, Sophie; Ruck, Tobias; Biel, Martin; Wahl-Schott, Christian; Grimm, Christian; Meuth, Sven G.; Lesage, Florian
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Development of the First Two-Pore Domain Potassium Channel TWIK-Related K+ Channel 1-Selective Agonist Possessing in Vivo Antinociceptive Activity
err2017-01-20
err52
PREAI
errVivier, Delphine; Ben Soussia, Ismail; Rodrigues, Nuno; Lolignier, Stephane; Devilliers, Maily; Chatelain, Franck C.; Prival, Laetitia; Chapuy, Eric; Bourdier, Geoffrey; Bennis, Khalil; Lesage, Florian; Eschalier, Alain; Busserolles, Jerome; Ducki, Sylvie
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The two-pore domain potassium channel, TWIK-1, has a role in the regulation of heart rate and atrial size
err2016-08-01
err31
PREAI
errChristensen, Alex Horby; Chatelain, Franck C.; Huttner, Inken G.; Olesen, Morten Sailing; Soka, Magdalena; Feliciangeli, Sylvain; Horvat, Claire; Santiago, Celine F.; Vandenberg, Jamie I.; Schmitt, Nicole; Olesen, Soren-Peter; Lesage, Florian; Fatkin, Diane
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In cellulo phosphorylation induces pharmacological reprogramming of maurocalcin, a cell-penetrating venom peptide
err2016-04-11
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errRonjat, Michel; Feng, Wei; Dardevet, Lucie; Dong, Yao; Al Khoury, Sawsan; Chatelain, Franck C.; Vialla, Virginie; Chahboun, Samir; Lesage, Florian; Darbon, Herve; Pessah, Isaac N.; De Waard, Michel
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