Relating Conformational Equilibria to Conformer-Specific Lipophilicities: New Opportunities in Drug DiscoveryANGEWANDTE CHEMIE-INTERNATIONAL EDITIONIF16.92021-12-2920OA
Skipped Fluorination Motifs: Synthesis of Building Blocks and Comparison of Lipophilicity Trends with Vicinal and Isolated Fluorination MotifsJOURNAL OF ORGANIC CHEMISTRYIF3.62021-01-0515OA
Systematic Investigation of Lipophilicity Modulation by Aliphatic Fluorination MotifsJOURNAL OF MEDICINAL CHEMISTRYIF6.82020-01-02100OAAI
Reducing the Lipophilicity of Perfluoroalkyl Groups by CF2-F/CF2-Me or CF3/CH3 ExchangeJOURNAL OF MEDICINAL CHEMISTRYIF6.82018-11-0980OAAI