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Modulating multi-functional ERK complexes by covalent targeting of a recruitment site in vivo Kaoud, Tamer S.; Johnson, William H.; Ebelt, Nancy D.; Piserchio, Andrea; Zamora-Olivares, Diana; Van Ravenstein, Sabrina X.; Pridgen, Jacey R.; Edupuganti, Ramakrishna; Sammons, Rachel; Cano, Micael; Warthaka, Mangalika; Harger, Matthew; Tavares, Clint D. J.; Park, Jihyun; Radwan, Mohamed F.; Ren, Pengyu; Anslyn, Eric V.; Tsai, Kenneth Y.; Ghose, Ranajeet; Dalby, Kevin N. 分享 收藏
Targeting multi-functional ERK-protein complexes in vivo Kaoud, Tamer S.; Johnson, William H.; Ebelt, Nancy D.; Piserchio, Andrea; Zamora-Olivares, Diana; Ravenstein, Sabrina V.; Pridgen, Jacey R.; Edupuganti, Ramakrishna; Sammons, Rachel; Cano, Micael; Warthaka, Mangalika; Ren, Pengyu; Anslyn, Eric V.; Tsai, Kenneth Y.; Ghose, Ranajeet; Dalby, Kevin N. 分享 收藏
A Novel Class of Common Docking Domain Inhibitors That Prevent ERK2 Activation and Substrate Phosphorylation Sammons, Rachel M.; Perry, Nicole A.; Li, Yangmei; Cho, Eun Jeong; Piserchio, Andrea; Zamora-Olivares, Diana P.; Ghose, Ranajeet; Kaoud, Tamer S.; Debevec, Ginamarie; Bartholomeusz, Chandra; Gurevich, Vsevolod V.; Iverson, Tina M.; Giulianotti, Marc; Houghten, Richard A.; Dalby, Kevin N. 分享 收藏
Protein Unfolded States are Characterized by the Duality of Sequence-Specific Conformational Preferences and Ensemble-Averaged Features of Canonical Random Coils Holehouse, Alex S.; Peran, Ivan; Stenzoski, Natalie E.; Zou, Junjie; Piserchio, Andrea; Ghose, Ranajeet; Carrico, Isaac S.; Bilsel, Osman; Raleigh, Daniel P.; Pappu, Rohit V. 分享 收藏
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Discovery of a covalent inhibitor of ERK docking-interactions that inhibits A375 melanoma cells proliferation Kaoud, Tamer S.; Johnson, William H.; Ebelt, Nancy D.; Piserchio, Andrea; Warthaka, Mangalika; Cano, Micael; Sammons, Rachel; Wang, Qiantao; Ren, Pengyu; Ghose, Ranajeet; Dalby, Kevin N. 分享 收藏
Structural and Dynamic Features of F-recruitment Site Driven Substrate Phosphorylation by ERK2 (vol 5, 11127, 2015) Piserchio, Andrea; Ramakrishan, Venkatesh; Wang, Hsin; Kaoud, Tamer S.; Arshava, Boris; Dutta, Kaushik; Dalby, Kevin N.; Ghose, Ranajeet 分享 收藏