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Clinical and veterinary trypanocidal benzoxaboroles target CPSF3 Wall, Richard J.; Rico, Eva; Lukac, Iva; Zuccotto, Fabio; Elg, Sara; Gilbert, Ian H.; Freund, Yvonne; Alley, M. R. K.; Field, Mark C.; Wyllie, Susan; Horn, David 分享 收藏
Discovery of a Potent and Specific M-tuberculosis Leucyl-tRNA Synthetase Inhibitor: (S)-3-(Aminomethyl)-4-chloro-7-(2hydroxyethoxy)benzo[c][1,2]oxaborol-1(3H)-ol (GSK656) Li, Xianfeng; Hernandez, Vincent; Rock, Fernando L.; Choi, Wai; Mak, Yvonne S. L.; Mohan, Manisha; Mao, Weimin; Zhou, Yasheen; Easom, Eric E.; Plattner, Jacob J.; Zou, Wuxin; Perez-Herran, Esther; Giordano, Ilaria; Mendoza-Losana, Alfonso; Alemparte, Carlos; Rullas, Joaquin; Angulo-Barturen, Inigo; Crouch, Sabrinia; Ortega, Fatima; Barros, David; Alley, M. R. K. 分享 收藏
A Novel 6-Benzyl Ether Benzoxaborole Is Active against Mycobacterium tuberculosis In Vitro Patel, Nipul; O'Malley, Theresa; Zhang, Yong-Kang; Xia, Yi; Sunde, Bjorn; Flint, Lindsay; Korkegian, Aaron; Ioerger, Thomas R.; Sacchettini, Jim; Alley, M. R. K.; Parish, Tanya 分享 收藏
A potent antimalarial benzoxaborole targets a Plasmodium falciparum cleavage and polyadenylation specificity factor homologue Sonoiki, Ebere; Ng, Caroline L.; Lee, Marcus C. S.; Guo, Denghui; Zhang, Yong-Kang; Zhou, Yasheen; Alley, M. R. K.; Ahyong, Vida; Sanz, Laura M.; Jose Lafuente-Monasterio, Maria; Dong, Chen; Schupp, Patrick G.; Gut, Jiri; Legac, Jenny; Cooper, Roland A.; Gamo, Francisco-Javier; DeRisi, Joseph; Freund, Yvonne R.; Fidock, David A.; Rosenthal, Philip J. 分享 收藏
Discovery of Novel Oral Protein Synthesis Inhibitors of Mycobacterium tuberculosis That Target Leucyl-tRNA Synthetase Palencia, Andres; Li, Xianfeng; Bu, Wei; Choi, Wai; Ding, Charles Z.; Easom, Eric E.; Feng, Lisa; Hernandez, Vincent; Houston, Paul; Liu, Liang; Meewan, Maliwan; Mohan, Manisha; Rock, Fernando L.; Sexton, Holly; Zhang, Suoming; Zhou, Yasheen; Wan, Baojie; Wang, Yuehong; Franzblau, Scott G.; Woolhiser, Lisa; Gruppo, Veronica; Lenaerts, Anne J.; O'Malley, Theresa; Parish, Tanya; Cooper, Christopher B.; Waters, M. Gerard; Ma, Zhenkun; Ioerger, Thomas R.; Sacchettini, James C.; Rullas, Joaquin; Angulo-Barturen, Inigo; Perez-Herran, Esther; Mendoza, Alfonso; Barros, David; Cusack, Stephen; Plattner, Jacob J.; Alley, M. R. K. 分享 收藏
Cryptosporidium and Toxoplasma Parasites Are Inhibited by a Benzoxaborole Targeting Leucyl-tRNA Synthetase Palencia, Andres; Liu, Ru-Juan; Lukarska, Maria; Gut, Jiri; Bougdour, Alexandre; Touquet, Bastien; Wang, En-Duo; Li, Xianfeng; Alley, M. R. K.; Freund, Yvonne R.; Rosenthal, Philip J.; Hakimi, Mohamed-Ali; Cusack, Stephen 分享 收藏
Antimalarial Benzoxaboroles Target Plasmodium falciparum Leucyl-tRNA Synthetase Sonoiki, Ebere; Palencia, Andres; Guo, Denghui; Ahyong, Vida; Dong, Chen; Li, Xianfeng; Hernandez, Vincent S.; Zhang, Yong-Kang; Choi, Wai; Gut, Jiri; Legac, Jennifer; Cooper, Roland; Alley, M. R. K.; Freund, Yvonne R.; DeRisi, Joseph; Cusack, Stephen; Rosenthal, Philip J. 分享 收藏
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Discovery of a Novel Class of Boron-Based Antibacterials with Activity against Gram-Negative Bacteria Hernandez, Vincent; Crepin, Thibaut; Palencia, Andres; Cusack, Stephen; Akama, Tsutomu; Baker, Stephen J.; Bu, Wei; Feng, Lisa; Freund, Yvonne R.; Liu, Liang; Meewan, Maliwan; Mohan, Manisha; Mao, Weimin; Rock, Fernando L.; Sexton, Holly; Sheoran, Anita; Zhang, Yanchen; Zhang, Yong-Kang; Zhou, Yasheen; Nieman, James A.; Anugula, Mahipal Reddy; Keramane, El Mehdi; Savariraj, Kingsley; Reddy, D. Shekhar; Sharma, Rashmi; Subedi, Rajendra; Singh, Rajeshwar; O'Leary, Ann; Simon, Nerissa L.; De Marsh, Peter L.; Mushtaq, Shazad; Warner, Marina; Livermore, David M.; Alley, M. R. K.; Plattner, Jacob J. 分享 收藏
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Discovery of a new boron-containing antifungal agent, 5-fluoro-1,3-dihydro-1-hydroxy-2,1-benzoxaborole (AN2690), for the potential treatment of onychomycosis Baker, Stephen J.; Zhang, Yong-Kang; Akama, Tsutomu; Lau, Agnes; Zhou, Huchen; Hernandez, Vincent; Mao, Weimin; Alley, M. R. K.; Sanders, Virginia; Plattner, Jacob J. 分享 收藏
Identification of borinic esters as inhibitors of bacterial cell growth and bacterial methyltransferases, CcrM and MenH Benkovic, SJ; Baker, SJ; Alley, MRK; Woo, YH; Zhang, YK; Akama, T; Mao, WM; Baboval, J; Rajagopalan, PTR; Wall, M; Kahng, LS; Tavassoli, A; Shapiro, L 分享 收藏
Complete genome sequence of Caulobacter crescentus Nierman, WC; Feldblyum, TV; Laub, MT; Paulsen, IT; Nelson, KE; Eisen, J; Heidelberg, JF; Alley, MRK; Ohta, N; Maddock, JR; Potocka, I; Nelson, WC; Newton, A; Stephens, C; Phadke, ND; Ely, B; DeBoy, RT; Dodson, RJ; Durkin, AS; Gwinn, ML; Haft, DH; Kolonay, JF; Smit, J; Craven, MB; Khouri, H; Shetty, J; Berry, K; Utterback, T; Tran, K; Wolf, A; Vamathevan, J; Ermolaeva, M; White, O; Salzberg, SL; Venter, JC; Shapiro, L; Fraser, CM 分享 收藏