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Modifying a Hydroxyl Patch in Glucagon-like Peptide 1 Produces Biased Agonists with Unique Signaling Profiles Wang, Peiqi; Hill, Timothy A.; Mitchell, Justin; Fitzsimmons, Rebecca L.; Xu, Weijun; Loh, Zhixuan; Suen, Jacky Y.; Lim, Junxian; Iyer, Abishek; Fairlie, David P. 分享 收藏
Temporal perturbation of histone deacetylase activity reveals a requirement for HDAC1-3 in mesendoderm cell differentiation Sinniah, Enakshi; Wu, Zhixuan; Shen, Sophie; Naval-Sanchez, Marina; Chen, Xiaoli; Lim, Junxian; Helfer, Abbigail; Iyer, Abishek; Tng, Jiahui; Lucke, Andrew J.; Reid, Robert C.; Redd, Meredith A.; Nefzger, Christian M.; Fairlie, David P.; Palpant, Nathan J. 分享 收藏
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The histone deacetylase Hdac7 supports LPS-inducible glycolysis and Il-1β production in murine macrophages via distinct mechanisms Ramnath, Divya; Das Gupta, Kaustav; Wang, Yizhuo; Abrol, Rishika; Curson, James E. B.; Lim, Junxian; Reid, Robert C.; Mansell, Ashley; Blumenthal, Antje; Karunakaran, Denuja; Fairlie, David P.; Sweet, Matthew J. 分享 收藏
HDAC7 Inhibition by Phenacetyl and Phenylbenzoyl Hydroxamates Mak, Jeffrey Y. W.; Wu, Kai-Chen; Gupta, Praveer K.; Barbero, Sheila; McLaughlin, Maddison G.; Lucke, Andrew J.; Tng, Jiahui; Lim, Junxian; Loh, Zhixuan; Sweet, Matthew J.; Reid, Robert C.; Liu, Ligong; Fairlie, David P. 分享 收藏
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Protease-activated receptor-2 ligands reveal orthosteric and allosteric mechanisms of receptor inhibition Kennedy, Amanda J.; Sundstrom, Linda; Geschwindner, Stefan; Poon, Eunice K. Y.; Jiang, Yuhong; Chen, Rongfeng; Cooke, Rob; Johnstone, Shawn; Madin, Andrew; Lim, Junxian; Liu, Qingqi; Lohman, Rink-Jan; Nordqvist, Anneli; Friden-Saxin, Maria; Yang, Wenzhen; Brown, Dean G.; Fairlie, David P.; Dekker, Niek 分享 收藏
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Potent Thiophene Antagonists of Human Complement C3a Receptor with Anti-Inflammatory Activity 具有抗炎活性的人补体C3a受体的有效噻吩拮抗剂 Rowley, Jessica A.; Reid, Robert C.; Poon, Eunice K. Y.; Wu, Kai-Chen; Lim, Junxian; Lohman, Rink-Jan; Hamidon, Johan K.; Yau, Mei-Kwan; Halili, Maria A.; Durek, Thomas; Iyer, Abishek; Fairlie, David P. 分享 收藏
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Exploiting a novel conformational switch to control innate immunity mediated by complement protein C3a Lohman, Rink-Jan; Hamidon, Johan K.; Reid, Robert C.; Rowley, Jessica A.; Yau, Mei-Kwan; Halili, Maria A.; Nielsen, Daniel S.; Lim, Junxian; Wu, Kai-Chen; Loh, Zhixuan; Anh Do; Suen, Jacky Y.; Iyer, Abishek; Fairlie, David P. 分享 收藏
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