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Affibody-Derived Drug Conjugates Targeting The Epidermal Growth Factor Receptor Are Potent And Specific Cytotoxic Agents Rinne, Sara S.; Yin, Wen; Li, Ruonan; Ding, Haozhong; Mestre Borras, Anna; Mahmod, Chenar; Stahl, Stefan; Orlova, Anna; Lofblom, John; Vorobyeva, Anzhelika; Graslund, Torbjorn 分享 收藏
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Single-Photon Emission Computer Tomography Imaging of Prostate-Specific Membrane Antigen (PSMA) Expression in Prostate Cancer Patients Using a Novel Peptide-Based Probe [99mTc]Tc-BQ0413 with Picomolar Affinity to PSMA: A Phase I/II Clinical Study 使用具有皮摩尔亲和力的新型肽基探针[⁹⁹mTc]Tc-BQ0413对前列腺癌患者中前列腺特异性膜抗原(PSMA)表达的单光子发射计算机断层成像研究:一项Ⅰ/Ⅱ期临床试验 Medvedeva, A; Chernov, V; Larkina, M; Rybina, A; Zelchan, R; Bragina, O; Varvashenya, R; Zebzeeva, O; Bezverkhniaia, E; Tolmachev, V; Orlova, A 分享 收藏
First-in-human experience with GRPR antagonist [68Ga]Ga-NOTA-PEG2-RM26 in prostate and breast cancer patients using PET/CT Bjareback, Annie; Jonmarker, Olof; Tzortzakakis, Antonios; Jussing, Emma; Li, Chunde; Altena, Renske; Hindorf, Cecilia; Orlova, Anna; Axelsson, Rimma; Tran, Thuy A. 分享 收藏
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Gastrin-releasing peptide receptor as theranostic target in estrogen-receptor positive breast cancer: A preclinical study of the theranostic pair [55Co]Co- and [177Lu]Lu-DOTA-RM26 Baun, Christina; Olsen, Birgitte Brinkmann; Alves, Carla Maria Lourenco; Ditzel, Henrik Jorn; Terp, Mikkel; Hildebrandt, Malene Grubbe; Poulsen, Charlotte Aaberg; Ge, Lorraine Gaenaelle; Gammelsrod, Vigga Sand; Orlova, Anna; Dam, Johan Hygum; Thisgaard, Helge 分享 收藏
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Evaluation of a novel 177Lu-labelled therapeutic Affibody molecule with a deimmunized ABD domain and improved biodistribution profile 评估具有脱敏ABD结构域和改善的生物分布特征的新型177lu-标记的治疗性亲和体分子 Liu, Yongsheng; Oroujeni, Maryam; Liao, Yunqi; Vorobyeva, Anzhelika; Bodenko, Vitalina; Orlova, Anna; Konijnenberg, Mark; Carlqvist, Matilda; Wahlberg, Elisabet; Loftenius, Annika; Frejd, Fredrik Y.; Tolmachev, Vladimir 分享 收藏
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Evaluation of affinity matured Affibody molecules for imaging of the immune checkpoint protein B7-H3 Oroujeni, Maryam; Bezverkhniaia, Ekaterina A.; Xu, Tianqi; Liu, Yongsheng; V. Plotnikov, Evgenii; Klint, Susanne; Ryer, Eva; Karlberg, Ida; Orlova, Anna; Frejd, Fredrik Y.; Tolmachev, Vladimir 分享 收藏
The GRPR Antagonist [99mTc]Tc-maSSS-PEG2-RM26 towards Phase I Clinical Trial: Kit Preparation, Characterization and Toxicity Abouzayed, Ayman; Borin, Jesper; Lundmark, Fanny; Rybina, Anastasiya; Hober, Sophia; Zelchan, Roman; Tolmachev, Vladimir; Chernov, Vladimir; Orlova, Anna 分享 收藏
Phase I clinical evaluation of 99mTc-labeled Affibody molecule for imaging HER2 expression in breast cancer Bragina, Olga; Chernov, Vladimir; Larkina, Mariia; Rybina, Anstasiya; Zelchan, Roman; Garbukov, Eugeniy; Oroujeni, Maryam; Loftenius, Annika; Orlova, Anna; Soerensen, Jens; Frejd, Fredrik Y.; Tolmachev, Vladimir 分享 收藏