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收藏Sulfonamide-Bearing Pyrazolone Derivatives as Multitarget Therapeutic Agents: Design, Synthesis, Characterization, Biological Evaluation, In Silico ADME/T Profiling and Molecular Docking Study含磺胺基的吡唑酮衍生物作为多靶点治疗剂:设计、合成、表征、生物评价、计算机ADME/T分析及分子对接研究
Lolak, Nebih; Akocak, Suleyman; Topal, Meryem; Kocyigit, Umit Muhammet; Isik, Mesut; Turkes, Cuneyt; Topal, Fevzi; Durgun, Mustafa; Beydemir, Sukru
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收藏Synthesis of Thiazole-methylsulfonyl Derivatives, X-ray Study, and Investigation of Their Carbonic Anhydrase Activities: In Vitro and In Silico Potentials
Maryam, Zahra; Isik, Aysen; Bagci, Emine Rana; Yildiz, Maksut; Unver, Hakan; Kocyigit, U''mit M.; Kirilmaz, Burak; Celik, Ismail; Cevik, Ulviye Acar; Ozkay, Yusuf; Kaplancikli, Zafer Asim
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收藏Novel diarylated tacrine derivatives: Synthesis, characterization, anticancer, antiepileptic, antibacterial, and antifungal activities
Misir, Busra A.; Derin, Yavuz; Okten, Salih; Aydin, Ali; Kocyigit, Umit M.; Sahin, Hatice; Tutar, Ahmet
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收藏Molecular hybrids integrated with imidazole and hydrazone structural motifs: Design, synthesis, biological evaluation, and molecular docking studies与咪唑和腙结构基序整合的分子杂种: 设计,合成,生物学评估和分子对接研究
Tapera, Michael; Saripinar, Emin; Kekecmuhammed, Hueseyin; Dogan, Murat; Tuzun, Burak; Kocyigit, Uemit M.; Cetin, Feyza Nur
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收藏Synthesis, carbonic anhydrase inhibitory activity, anticancer activity and molecular docking studies of new imidazolyl hydrazone derivatives
Tapera, Michael; Kekecmuhammed, Huseyin; Tuzun, Burak; Saripinar, Emin; Kocyigit, Umit M.; Yildirim, Ebrar; Dogan, Murat; Zorlu, Yunus
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收藏Potential thiosemicarbazone-based enzyme inhibitors: Assessment of antiproliferative activity, metabolic enzyme inhibition properties, and molecular docking calculations潜在的基于缩氨基硫脲的酶抑制剂: 抗增殖活性,代谢酶抑制特性和分子对接计算的评估
Yakan, Hasan; Kocyigit, Umit M.; Muglu, Halit; Ergul, Mustafa; Erkan, Sultan; Guzel, Emre; Taslimi, Parham; Gulcin, Ilhami
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收藏Synthesis, characterization, crystal structures, theoretical calculations and biological evaluations of novel substituted tacrine derivatives as cholinesterase and carbonic anhydrase enzymes inhibitors
Okten, Salih; Ekiz, Makbule; Kocyigit, Umit Muhammet; Tutar, Ahmet; Celik, Ismail; Akkurt, Mehmet; Gokalp, Faik; Taslimi, Parham; Gulcin, Ilhami
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收藏In vitro cytotoxic and in vivo antitumoral activities of some aminomethyl derivatives of 2,4-dihydro-3H-1,2,4-triazole-3-thiones-Evaluation of their acetylcholinesterase and carbonic anhydrase enzymes inhibition profiles
Timur, Irfan; Kocyigit, Umit M.; Dastan, Taner; Sandal, Suleyman; Ceribasi, Ali Osman; Taslimi, Parham; Gulcin, Ilhami; Koparir, Metin; Karatepe, Mustafa; Ciftci, Mehmet
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收藏Synthesis of some novel pyridine compounds containing bis-1,2,4-triazole/thiosemicarbazide moiety and investigation of their antioxidant properties, carbonic anhydrase, and acetylcholinesterase enzymes inhibition profiles含有bis-1,2,4-三唑/氨基硫脲部分的一些新型吡啶化合物的合成及其抗氧化性能,碳酸酐酶和乙酰胆碱酯酶抑制特性的研究
Bulut, Nilufer; Kocyigit, Umit M.; Gecibesler, Ibrahim H.; Dastan, Taner; Karci, Huseyin; Taslimi, Parham; Dastan, Sevgi Durna; Gulcin, Ilhami; Cetin, Ahmet
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