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Luciano De Petrocellis

consiglio nazionale delle ricerche

82H指数
279论文数
2.6W被引数
收录论文 114
发表时间
Targeting TRPA1 with Novel Synthetic Compounds Based on Different Scaffolds to Reduce Acute and Chronic Pain基于不同骨架的新型合成化合物靶向TRPA1以减轻急性和慢性疼痛
err2026-02-11
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errAlessia Agata Corallo; Samuele Maramai; Carlotta Noli; Marco Paolino; Antonella Brizzi; Alessia Ligresti; Marco Allarà; Luciano De Petrocellis; Rosa Maria Vitale; Aniello Schiano Moriello; Carmela Belardo; Rosmara Infantino; Sabatino Maione; Claudia Mugnaini; Federico Corelli
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The Impact of a Quinone Scaffold on Thermo-TRPs Modulation by Dimethylheptyl Phytocannabinoids基于二甲基庚基类大麻酚对热敏TRP通道调节的醌骨架影响
err2025-03-17
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errSchiano Moriello, Aniello; Bossoni, Aurora; Mattoteia, Daiana; Caprioglio, Diego; Minassi, Alberto; Appendino, Giovanni; De Petrocellis, Luciano; Amodeo, Pietro; Vitale, Rosa Maria
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Indole-2-Carboxamide as an Effective Scaffold for the Design of New TRPV1 Agonists
err2025-02-05
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errMaramai, Samuele; Mugnaini, Claudia; Paolino, Marco; Moriello, Aniello Schiano; De Petrocellis, Luciano; Corelli, Federico; Aiello, Francesca; Brizzi, Antonella
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An updated patent review of TRPA1 antagonists (2020-present)
err2024-06-17
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PREAI
errVitale, Rosa Maria; de Petrocellis, Luciano; Amodeo, Pietro
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Phytochemical Characterization and TRPA1/TRPM8 Modulation Profile of the Cannabigerol-Rich Cannabis sativa L. Chemotype IV
err2024-02-26
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PREAI
errGargiulo, Ernesto; Moriello, Aniello Schiano; Benetti, Emanuele; Pagni, Luca; Arnoldi, Lolita; De Petrocellis, Luciano; Chianese, Giuseppina; Vitale, Rosa Maria; Taglialatela-Scafati, Orazio
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In Silico-Guided Rational Drug Design and Synthesis of Novel 4-(Thiophen-2-yl)butanamides as Potent and Selective TRPV1 Agonists
err2023-05-16
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PREAI
errRomeo, Isabella; Brizzi, Antonella; Pessina, Federica; Ambrosio, Francesca Alessandra; Aiello, Francesca; Belardo, Carmela; Carullo, Gabriele; Costa, Giosue; De Petrocellis, Luciano; Frosini, Maria; Luongo, Livio; Maramai, Samuele; Paolino, Marco; Moriello, Aniello Schiano; Mugnaini, Claudia; Scorzelli, Francesco; Maione, Sabatino; Corelli, Federico; Di Marzo, Vincenzo; Alcaro, Stefano; Artese, Anna
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The Combined Effect of Branching and Elongation on the Bioactivity Profile of Phytocannabinoids. Part I: Thermo-TRPs
err2021-08-23
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errMattoteia, Daiana; Moriello, Aniello Schiano; Taglialatela-Scafati, Orazio; Amodeo, Pietro; De Petrocellis, Luciano; Appendino, Giovanni; Vitale, Rosa Maria; Caprioglio, Diego
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Synthesis and molecular targets of N-13-hydroxy-octadienoyl-ethanolamine, a novel endogenous bioactive 15-lipoxygenase-derived metabolite of N-linoleoyl-ethanolamine found in the skin and saliva
err2021-08-01
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PREAI
errTinto, Francesco; Archambault, Anne-Sophie; Dumais, Elizabeth; Rakotoarivelo, Volatiana; Kostrzewa, Magdalena; Martin, Cyril; Plante, Pier-Luc; Desjardins, Yves; Simard, Melissa; Pouliot, Roxane; De Petrocellis, Luciano; Ligresti, Alessia; Di Marzo, Vincenzo; Flamand, Nicolas
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A Glucuronic Acid-Palmitoylethanolamide Conjugate (GLUPEA) Is an Innovative Drug Delivery System and a Potential Bioregulator
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IF5.2
err2021-02-20
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errManzo, Emiliano; Schiano Moriello, Aniello; Tinto, Francesco; Verde, Roberta; Allara, Marco; De Petrocellis, Luciano; Pagano, Ester; Izzo, Angelo A.; Di Marzo, Vincenzo; Petrosino, Stefania
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Discovery of a Remarkable Methyl Shift Effect in the Vanilloid Activity of Triterpene Amides
err2020-11-02
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errVitale, Rosa Maria; Avonto, Cristina; Del Prete, Danilo; Moriello, Aniello Schiano; Amodeo, Pietro; Appendino, Giovanni; De Petrocellis, Luciano
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Design, Synthesis and In Vitro Experimental Validation of Novel TRPV4 Antagonists Inspired by Labdane Diterpenes
err2020-10-18
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errMazzotta, Sarah; Carullo, Gabriele; Schiano Moriello, Aniello; Amodeo, Pietro; Di Marzo, Vincenzo; Vega-Holm, Margarita; Vitale, Rosa Maria; Aiello, Francesca; Brizzi, Antonella; De Petrocellis, Luciano
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Cannabitwinol, a Dimeric Phytocannabinoid from Hemp, Cannabis sativa L., Is a Selective Thermo-TRP Modulator
err2020-09-03
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PREAI
errChianese, Giuseppina; Lopatriello, Annalisa; Schiano-Moriello, Aniello; Caprioglio, Diego; Mattoteia, Daiana; Benetti, Emanuele; Ciceri, Daniele; Arnoldi, Lolita; De Combarieu, Eric; Vitale, Rosa M.; Amodeo, Pietro; Appendino, Giovanni; De Petrocellis, Luciano; Taglialatela-Scafati, Orazio
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Synthetic bioactive olivetol-related amides: The influence of the phenolic group in cannabinoid receptor activity
err2020-06-01
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PREAI
errBrizzi, Antonella; Aiello, Francesca; Boccella, Serena; Cascio, Maria Grazia; De Petrocellis, Luciano; Frosini, Maria; Gado, Francesca; Ligresti, Alessia; Luongo, Livio; Marini, Pietro; Mugnaini, Claudia; Pessina, Federica; Corelli, Federico; Maione, Sabatino; Manera, Clementina; Pertwee, Roger G.; Di Marzo, Vincenzo
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Identification and Characterization of Cannabimovone, a Cannabinoid from Cannabis sativa, as a Novel PPARγ Agonist via a Combined Computational and Functional Study
err2020-03-03
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errIannotti, Fabio Arturo; De Maio, Fabrizia; Panza, Elisabetta; Appendino, Giovanni; Taglialatela-Scafati, Orazio; De Petrocellis, Luciano; Amodeo, Pietro; Vitale, Rosa Maria
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Moringin, A Stable Isothiocyanate from Moringa oleifera, Activates the Somatosensory and Pain Receptor TRPA1 Channel In Vitro
err2020-02-22
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errBorgonovo, Gigliola; De Petrocellis, Luciano; Moriello, Aniello Schiano; Bertoli, Simona; Leone, Alessandro; Battezzati, Alberto; Mazzini, Stefania; Bassoli, Angela
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Life cycle of scientific publications in the field of high social impact
err2019-10-18
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PREAI
errRuggiero, B.; Amato, U.; Franco, B.; De Petrocellis, L.; Vettoliere, A.; Granata, C.; Silvestrini, S.; Bonavolonta, C.; Valentino, M.; Brocchieri, J.; Silvestrini, P.
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Isothiocyanates and Glucosinolates from Sisymbrium officinale (L.) Scop. (the Singers' Plant): Isolation and in Vitro Assays on the Somatosensory and Pain Receptor TRPA1 Channel
err2019-03-08
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errBorgonovo, Gigliola; Zimbaldi, Nathan; Guarise, Marta; De Nisi, Patrizia; De Petrocellis, Luciano; Moriello, Aniello Schiano; Bassoli, Angela
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Effects of non-euphoric plant cannabinoids on muscle quality and performance of dystrophic mdx mice
err2018-09-09
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errIannotti, Fabio Arturo; Pagano, Ester; Moriello, Aniello Schiano; Alvino, Filomena Grazia; Sorrentino, Nicolina Cristina; D'Orsi, Luca; Gazzerro, Elisabetta; Capasso, Raffaele; De Leonibus, Elvira; De Petrocellis, Luciano; Di Marzo, Vincenzo
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Elongation of the Hydrophobic Chain as a Molecular Switch: Discovery of Capsaicin Derivatives and Endogenous Lipids as Potent Transient Receptor Potential Vanilloid Channel 2 Antagonists
err2018-09-03
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PREAI
errMoriello, Aniello Schiano; Lopez Chinarro, Silvia; Novo Fernandez, Olalla; Eras, Jordi; Amodeo, Pietro; Canela-Garayoa, Ramon; Vitale, Rosa Maria; Di Marzo, Vincenzo; De Petrocellis, Luciano
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TRPA1 Modulating C14 Polyacetylenes from the Iranian Endemic Plant Echinophora platyloba
err2018-07-17
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errChianese, Giuseppina; Sirignano, Carmina; Shokoohinia, Yalda; Mohammadi, Zeynab; Bazvandi, Leili; Jafari, Fataneh; Jalilian, Fereshteh; Moriello, Aniello Schiano; De Petrocellis, Luciano; Taglialatela-Scafati, Orazio; Rigano, Daniela
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