未登录 The Concise Guide to PHARMACOLOGY 2025/26: Catalytic receptors 《药物学简明指南2025/26:催化性受体》 Alexander, Stephen P. H.; Fabbro, Doriano; Peach, Chloe J.; Gibb, Alasdair J.; Kelly, Eamonn; Mathie, Alistair A.; Veale, Emma L.; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Southan, Christopher; Davies, Jamie A.; Beuve, Annie; Brouckaert, Peter; Bryant, Clare; Burnett, John C.; Farndale, Richard W.; Friebe, Andreas; Garthwaite, John; Hobbs, Adrian J.; Jarvis, Gavin E.; Kilpatrick, Laura; Koesling, Doris; Kuhn, Michaela; Leitinger, Birgit; Macewan, David; Monie, Tom P.; Potter, Lincoln R.; Russwurm, Michael; Schmidt, Harald H. H. W.; Stasch, Johannes-peter; Waldman, Scott A. 分享 收藏
The Concise Guide to PHARMACOLOGY 2025/26: Enzymes 《药理学简明指南》2025/26:酶 Alexander, Stephen P. H.; Fabbro, Doriano; Gibb, Alasdair J.; Kelly, Eamonn; Mathie, Alistair A.; Peach, Chloe J.; Veale, Emma L.; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Southan, Christopher; Davies, Jamie A.; Annett, Stephanie; Boison, Detlev; Burns, Kathryn Elisa; Dessauer, Carmen; Gertsch, Jurg; Helsby, Nuala Ann; Izzo, Angelo A.; Ostrom, Rennolds; Pagano, Ester; Papapetropoulos, Andreas; Pyne, Nigel J.; Pyne, Susan; Robson, Tracy; Seifert, Roland; Stasch, Johannes-peter; Szabo, Csaba; van der Stelt, Mario; Van Der Vliet, Albert; Watts, Val; Wong, Szu Shen 分享 收藏
The Concise Guide to PHARMACOLOGY 2025/26: Introduction and Other Protein Targets 《简明药理学指南2025/26:引言与其他蛋白质靶点》 Alexander, Stephen P. H.; Gibb, Alasdair J.; Kelly, Eamonn; Mathie, Alistair A.; Peach, Chloe J.; Veale, Emma L.; Cidlowski, John A.; Davenport, Anthony P.; Fabbro, Doriano; Spedding, Michael; Striessnig, Jorg; Armstrong, Jane F.; Buneman, O. Peter; Faccenda, Elena; Harding, Simon D.; Southan, Christopher; Davies, Jamie A.; Ahlers-dannen, Katelin E.; Alqinyah, Mohammed; Arumugam, Thiruma V.; Bodle, Christopher; Dagner, Josephine Buo; Chakravarti, Bandana; Choudhuri, Shreoshi P.; Druey, Kirk M.; Fisher, Rory A.; Gerber, Kyle J.; Hepler, John R.; Hooks, Shelley B.; Kantheti, Havish S.; Karaj, Behirda; Layeghi-ghalehsoukhteh, Somayeh; Lee, Jae-kyung; Luo, Zili; Martemyanov, Kirill; Mascarenhas, Luke D.; McNabb, Harrison; Montanez-Miranda, Carolina; Ogujiofor, Osita; Phan, Hoa; Roman, David L.; Shaw, Vincent; Sjogren, Benita; Sobey, Christopher; Spicer, Mackenzie M.; Squires, Katherine E.; Sutton, Laurie; Wendimu, Menbere; Wilkie, Thomas; Xie, Keqiang; Zhang, Qian; Zolghadri, Yalda 分享 收藏
The Concise Guide to PHARMACOLOGY 2023/24: Enzymes Alexander, Stephen P. H.; Fabbro, Doriano; Kelly, Eamonn; Mathie, Alistair A.; Peters, John A.; Veale, Emma L.; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Davies, Jamie A.; Annett, Stephanie; Boison, Detlev; Burns, Kathryn Elisa; Dessauer, Carmen; Gertsch, Jurg; Helsby, Nuala Ann; Izzo, Angelo A.; Ostrom, Rennolds; Papapetropoulos, Andreas; Pyne, Nigel J.; Pyne, Susan; Robson, Tracy; Seifert, Roland; Stasch, Johannes-Peter; Szabo, Csaba; van der Stelt, Mario; van der Vliet, Albert; Watts, Val; Wong, Szu Shen 分享 收藏
The Concise Guide to PHARMACOLOGY 2023/24: Catalytic receptors Alexander, Stephen P. H.; Fabbro, Doriano; Kelly, Eamonn; Mathie, Alistair A.; Peters, John A.; Veale, Emma L.; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Davies, Jamie A.; Beuve, Annie; Brouckaert, Peter; Bryant, Clare; Burnett, John C.; Farndale, Richard W.; Friebe, Andreas; Garthwaite, John; Hobbs, Adrian J.; Jarvis, Gavin E.; Koesling, Doris; Kuhn, Michaela; Macewan, David; Monie, Tom P.; Potter, Lincoln R.; Russwurm, Michael; Schmidt, Harald H. H. W.; Stasch, Johannes-Peter; Waldman, Scott A. 分享 收藏
The Concise Guide to PHARMACOLOGY 2023/24: Transporters Alexander, Stephen P. H.; Fabbro, Doriano; Kelly, Eamonn; Mathie, Alistair A.; Peters, John A.; Veale, Emma L.; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Davies, Jamie A.; Amarosi, Laura; Anderson, Catriona M. H.; Beart, Philip M.; Broer, Stefan; Dawson, Paul A.; Gyimesi, Gergely; Hagenbuch, Bruno; Hammond, James R.; Hancox, Jules C.; Hershfinkel, Michal; Inui, Ken-ichi; Kanai, Yoshikatsu; Kemp, Stephan; Kunji, Edmund R. S.; Stewart, Gavin; Tavoulari, Sotiria; Thwaites, David T.; Verri, Tiziano 分享 收藏
The Concise Guide to PHARMACOLOGY 2023/24: Introduction and Other Protein Targets 药理学2023/24简明指南: 介绍和其他蛋白质靶标 Alexander, Stephen P. H.; Kelly, Eamonn; Mathie, Alistair A.; Peters, John A.; Veale, Emma L.; Armstrong, Jane F.; Buneman, O. Peter; Faccenda, Elena; Harding, Simon D.; Spedding, Michael; Cidlowski, John A.; Fabbro, Doriano; Davenport, Anthony P.; Striessnig, Joerg; Davies, Jamie A.; Ahlers-Dannen, Katelin E.; Alqinyah, Mohammed; Arumugam, Thiruma V.; Bodle, Christopher; Dagner, Josephine Buo; Chakravarti, Bandana; Choudhuri, Shreoshi P.; Druey, Kirk M.; Fisher, Rory A.; Gerber, Kyle J.; Hepler, John R.; Hooks, Shelley B.; Kantheti, Havish S.; Karaj, Behirda; Layeghi-Ghalehsoukhteh, Somayeh; Lee, Jae-Kyung; Luo, Zili; Martemyanov, Kirill; Mascarenhas, Luke D.; McNabb, Harrison; Montanez-Miranda, Carolina; Ogujiofor, Osita; Phan, Hoa; Roman, David L.; Shaw, Vincent; Sjogren, Benita; Sobey, Christopher; Spicer, Mackenzie M.; Squires, Katherine E.; Sutton, Laurie; Wendimu, Menbere; Wilkie, Thomas; Xie, Keqiang; Zhang, Qian; Zolghadri, Yalda 分享 收藏
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THE CONCISE GUIDE TO PHARMACOLOGY 2021/22: Catalytic receptors Alexander, Stephen P. H.; Fabbro, Doriano; Kelly, Eamonn; Mathie, Alistair; Peters, John A.; Veale, Emma L.; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Pawson, Adam J.; Southan, Christopher; Davies, Jamie A.; Beuve, Annie; Brouckaert, Peter; Bryant, Clare; Burnett, John C.; Farndale, Richard W.; Friebe, Andreas; Garthwaite, John; Hobbs, AdrianJ; Jarvis, Gavin E.; Kuhn, Michaela; MacEwan, David; Monie, Tom P.; Papapetropoulos, Andreas; Potter, Lincoln R.; Schmidt, Harald H. H. W.; Szabo, Csaba; Waldman, Scott A. 分享 收藏
THE CONCISE GUIDE TO PHARMACOLOGY 2021/22: Enzymes Alexander, Stephen P. H.; Fabbro, Doriano; Kelly, Eamonn; Mathie, Alistair; Peters, John A.; Veale, Emma L.; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Pawson, Adam J.; Southan, Christopher; Davies, Jamie A.; Boison, Detlev; Burns, Kathryn Elisa; Dessauer, Carmen; Gertsch, Jurg; Helsby, Nuala Ann; Izzo, Angelo A.; Koesling, Doris; Ostrom, Rennolds; Pyne, Nigel J.; Pyne, Susan; Russwurm, Michael; Seifert, Roland; Stasch, Johannes-Peter; van der Stelt, Mario; van der Vliet, Albert; Watts, Val; Wong, Szu Shen 分享 收藏
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4-(Difluoromethyl)-5-(4-((3R,5S)-3,5-dimethylmorpholino)-6-((R)-3-methylmorpholino)-1,3,5-triazin-2-yl)pyridin-2-amine (PQR626), a Potent, Orally Available, and Brain-Penetrant mTOR Inhibitor for the Treatment of Neurological Disorders Borsari, Chiara; Keles, Erhan; Rageot, Denise; Treyer, Andrea; Bohnacker, Thomas; Bissegger, Lukas; De Pascale, Martina; Melone, Anna; Sriramaratnam, Rohitha; Beaufils, Florent; Hamburger, Matthias; Hebeisen, Paul; Loscher, Wolfgang; Fabbro, Doriano; Hillmann, Petra; Wymann, Matthias P. 分享 收藏
Discovery and preclinical characterization of PQR626: A potent, orally available, and brain-penetrant mTOR inhibitor for the treatment of tuberous sclerosis complex Borsari, Chiara; Keles, Erhan; Rageot, Denise; Melone, Anna; Bohnacker, Thomas; Batchelor, Lucinda Kate; De Pascale, Martina; Hebeisen, Paul; Hillmann, Petra; Fabbro, Doriano; Wymann, Matthias 分享 收藏
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THE CONCISE GUIDE TO PHARMACOLOGY 2019/20: Catalytic receptors Alexander, Stephen P. H.; Fabbro, Doriano; Kelly, Eamonn; Mathie, Alistair; Peters, John A.; Veale, Emma L.; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Pawson, Adam J.; Sharman, Joanna L.; Southan, Christopher; Davies, Jamie A. 分享 收藏
THE CONCISE GUIDE TO PHARMACOLOGY 2019/20: Introduction and Other Protein Targets 药理学2019/20简明指南: 介绍和其他蛋白质靶标 Alexander, Stephen P. H.; Kelly, Eamonn; Mathie, Alistair; Peters, John A.; Veale, Emma L.; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Pawson, Adam J.; Sharman, Joanna L.; Southan, Christopher; Buneman, O. Peter; Cidlowski, John A.; Christopoulos, Arthur; Davenport, Anthony P.; Fabbro, Doriano; Spedding, Michael; Striessnig, Joerg; Davies, Jamie A. 分享 收藏
THE CONCISE GUIDE TO PHARMACOLOGY 2019/20: Enzymes Alexander, Stephen P. H.; Fabbro, Doriano; Kelly, Eamonn; Mathie, Alistair; Peters, John A.; Veale, Emma L.; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Pawson, Adam J.; Sharman, Joanna L.; Southan, Christopher; Davies, Jamie A. 分享 收藏
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Preclinical Development of PQR514, a Highly Potent PI3K Inhibitor Bearing a Difluoromethyl-Pyrimidine Moiety Borsari, Chiara; Rageot, Denise; Beaufils, Florent; Bohnacker, Thomas; Keles, Erhan; Buslov, Ivan; Melone, Anna; Sele, Alexander M.; Hebeisen, Paul; Fabbro, Doriano; Hillmann, Petra; Wymann, Matthias P. 分享 收藏