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Cerastecin Inhibition of the Lipooligosaccharide Transporter MsbA to Combat Acinetobacter baumannii: From Screening Impurity to In Vivo Efficacy Skudlarek, Jason W.; Cooke, Andrew J.; Mitchell, Helen J.; Babaoglu, Kerim; Shaw, Anthony W.; Tong, Ling; Nomland, Ashley B.; Labroli, Marc; Sha, Deyou; Mulhearn, James J.; Wu, Chengwei; Li, Sarah W.; Beshore, Douglas C.; Hughes, Jonathan M. E.; Jouffroy, Matthieu; Wang, Hao; Balibar, Carl J.; Painter, Ronald E.; Shen, Pamela; Lange, Henry S.; Ishchenko, Andrii; Chen, Yun-Ting; Klein, Daniel J.; Tracy, Rodger W.; Miller, Randy R.; Cabalu, Tamara D.; Wu, Zhe; Leithead, Andrew; Scapin, Giovanna; Hruza, Alan W.; Dzhekieva, Liudmila; Bukhtiyarova, Marina; Homsher, Michelle F.; Xu, Min; Bahnck-Teets, Carolyn; McKenney, David; Buevich, Alexei V.; Liu, Jian; Zhang, Li-Kang; Meng, Tao; Kelly, Terri; Dinunzio, Edward; Soisson, Stephen; Cheng, Robert K. Y.; Hennig, Michael; Raheem, Izzat; Walker, Scott S. 分享 收藏
Apo and ligand-bound high resolution Cryo-EM structures of the human Kv3.1 channel reveal a novel binding site for positive modulators Botte, Mathieu; Huber, Sophie; Bucher, Denis; Klint, Julie K.; Rodriguez, David; Tagmose, Lena; Chami, Mohamed; Cheng, Robert; Hennig, Michael; Rahman, Wassim Abdul 分享 收藏
Acoustic levitation and rotation of thin films and their application for room temperature protein crystallography (vol 12, 5349, 2022) Kepa, Michal. W.; Tomizaki, Takashi; Sato, Yohei; Ozerov, Dmitry; Sekiguchi, Hiroshi; Yasuda, Nobuhiro; Aoyama, Koki; Skopintsev, Petr; Standfuss, Jorg; Cheng, Robert; Hennig, Michael; Tsujino, Soichiro 分享 收藏
Cryo-EM structures of a LptDE transporter in complex with Pro-macrobodies offer insight into lipopolysaccharide translocation Botte, Mathieu; Ni, Dongchun; Schenck, Stephan; Zimmermann, Iwan; Chami, Mohamed; Bocquet, Nicolas; Egloff, Pascal; Bucher, Denis; Trabuco, Matilde; Cheng, Robert K. Y.; Brunner, Janine D.; Seeger, Markus A.; Stahlberg, Henning; Hennig, Michael 分享 收藏
Acoustic levitation and rotation of thin films and their application for room temperature protein crystallography Kepa, Michal W.; Tomizaki, Takashi; Sato, Yohei; Ozerov, Dmitry; Sekiguchi, Hiroshi; Yasuda, Nobuhiro; Aoyama, Koki; Skopintsev, Petr; Standfuss, Jorg; Cheng, Robert; Hennig, Michael; Tsujino, Soichiro 分享 收藏
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Ligand channel in pharmacologically stabilized rhodopsin Mattle, Daniel; Kuhn, Bernd; Aebi, Johannes; Bedoucha, Marc; Kekilli, Demet; Grozinger, Nathalie; Alker, Andre; Rudolph, Markus G.; Schmid, Georg; Schertler, Gebhard F. X.; Hennig, Michael; Standfuss, Jorg; Dawson, Roger J. P. 分享 收藏
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Serial millisecond crystallography for routine room-temperature structure determination at synchrotrons Weinert, Tobias; Olieric, Natacha; Cheng, Robert; Bruenle, Steffen; James, Daniel; Ozerov, Dmitry; Gashi, Dardan; Vera, Laura; Marsh, May; Jaeger, Kathrin; Dworkowski, Florian; Panepucci, Ezequiel; Basu, Shibom; Skopintsev, Petr; Dore, Andrew S.; Geng, Tian; Cooke, Robert M.; Liang, Mengning; Prota, Andrea E.; Panneels, Valerie; Nogly, Przemyslaw; Ermler, Ulrich; Schertler, Gebhard; Hennig, Michael; Steinmetz, Michel O.; Wang, Meitian; Standfuss, Jorg 分享 收藏
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Cholesteryl ester transfer between lipoproteins does not require a ternary tunnel complex with CETP Lauer, Matthias E.; Graff-Meyer, Alexandra; Rufer, Arne C.; Maugeais, Cyrille; von der Mark, Elisabeth; Matile, Hugues; D'Arcy, Brigitte; Magg, Christine; Ringler, Philippe; Mueller, Shirley A.; Scherer, Sebastian; Dernick, Gregor; Thoma, Ralf; Hennig, Michael; Niesor, Eric J.; Stahlberg, Henning 分享 收藏
Generation, characterization and structural data of chymase binding proteins based on the human Fyn kinase SH3 domain Schlatter, Daniel; Brack, Simon; Banner, David W.; Batey, Sarah; Benz, Joerg; Bertschinger, Julian; Huber, Walter; Joseph, Catherine; Rufer, Arne C.; van der Klooster, Anita; Weber, Martin; Grabulovski, Dragan; Hennig, Michael 分享 收藏
Structure of the Acid-sensing ion channel 1 in complex with the gating modifier Psalmotoxin 1 Dawson, Roger J. P.; Benz, Joerg; Stohler, Peter; Tetaz, Tim; Joseph, Catherine; Huber, Sylwia; Schmid, Georg; Huegin, Daniela; Pflimlin, Pascal; Trube, Gerd; Rudolph, Markus G.; Hennig, Michael; Ruf, Armin 分享 收藏
Unique carbohydrate-carbohydrate interactions are required for high affinity binding between FcγRIII and antibodies lacking core fucose Ferrara, Claudia; Grau, Sandra; Jaeger, Christiane; Sondermann, Peter; Bruenker, Peter; Waldhauer, Inja; Hennig, Michael; Ruf, Armin; Rufer, Arne Christian; Stihle, Martine; Umana, Pablo; Benz, Joerg 分享 收藏
A New DNA Gyrase Inhibitor Subclass of the Cyclothialidine Family Based on a Bicyclic Dilactam-Lactone Scaffold. Synthesis and Antibacterial Properties Angehrn, Peter; Goetschi, Erwin; Gmuender, Hans; Hebeisen, Paul; Hennig, Michael; Kuhn, Bernd; Luebbers, Thomas; Reindl, Peter; Ricklin, Fabienne; Schmitt-Hoffmann, Anne 分享 收藏
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Structural properties of AMP-activated protein kinase -: Dimerization, molecular shape, and changes upon ligand binding Riek, Uwe; Scholz, Roland; Konarev, Peter; Rufer, Arne; Suter, Marianne; Nazabal, Alexis; Ringler, Philippe; Chami, Mohamed; Mueller, Shirley A.; Neumann, Dietbert; Forstner, Michael; Hennig, Michael; Zenobi, Renato; Engel, Andreas; Svergun, Dmitri; Schlattner, Uwe; Wallimann, Theo 分享 收藏