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William P. Tansey

vanderbilt university

45H指数
174论文数
8.6K被引数
收录论文 66
发表时间
eNRSA: a faster and more powerful approach for nascent transcriptome analysiseNRSA:一种用于新转录组分析更快且更强大的方法
err2025-01-01
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errOAAI
errWang, Jing; Chen, Hua-chang; Hiebert, Scott W.; Sheng, Quanhu; Tansey, William P.; Shyr, Yu; Liu, Qi
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Mitotic gene regulation by the N-MYC-WDR5-PDPK1 nexus
err2024-04-11
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errStreeter, Sarah A.; Williams, Alexandria G.; Evans, James R.; Wang, Jing; Guarnaccia, Alissa D.; Florian, Andrea C.; Al-Tobasei, Rafet; Liu, Qi; Tansey, William P.; Weissmiller, April M.
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WD Repeat Domain 5 Inhibitors for Cancer Therapy: Not What You Think
err2024-01-03
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errWeissmiller, April M.; Fesik, Stephen W.; Tansey, William P.
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Structure-Based Discovery of Potent, Orally Bioavailable Benzoxazepinone-Based WD Repeat Domain 5 Inhibitors
err2023-12-12
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PREAI
errTeuscher, Kevin B.; Mills, Jonathan J.; Tian, Jianhua; Han, Changho; Meyers, Kenneth M.; Sai, Jiqing; South, Taylor M.; Crow, Mackenzie M.; Van Meveren, Mayme; Sensintaffar, John L.; Zhao, Bin; Amporndanai, Kangsa; Moore, William J.; Stott, Gordon M.; Tansey, William P.; Lee, Taekyu; Fesik, Stephen W.
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WDR5 facilitates recruitment of N-MYC to conserved WDR5 gene targets in neuroblastoma cell lines
err2023-06-19
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errBumpous, Leigh A.; Moe, Kylie C.; Wang, Jing; Carver, Logan A.; Williams, Alexandria G.; Romer, Alexander S.; Scobee, Jesse D.; Maxwell, Jack N.; Jones, Cheyenne A.; Chung, Dai H.; Tansey, William P.; Liu, Qi; Weissmiller, April M.
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Targeting what is not there to treat cancer
err2023-05-13
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PREAI
errTansey, William P.
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Structure-based discovery of potent WD repeat domain 5 inhibitors that demonstrate efficacy and safety in preclinical animal models
err2022-12-27
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errOAAI
errTeuscher, Kevin B.; Chowdhury, Somenath; Meyers, Kenneth M.; Tian, Jianhua; Sai, Jiqing; Van Meveren, Mayme; South, Taylor M.; Sensintaffar, John L.; Rietz, Tyson A.; Goswami, Soumita; Wang, Jing; Grieb, Brian C.; Lorey, Shelly L.; Howard, Gregory C.; Liu, Qi; Moore, William J.; Stott, Gordon M.; Tansey, William P.; Leea, Taekyu; Fesik, Stephen W.
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Emerging Themes in Mechanisms of Tumorigenesis by SWI/SNF Subunit Mutation
err2022-07-26
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errJones, Cheyenne A.; Tansey, William P.; Weissmiller, April M.
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The SWI/SNF ATPase BRG1 facilitates multiple pro-tumorigenic gene expression programs in SMARCB1-deficient cancer cells
err2022-06-01
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errMoe, Kylie C.; Maxwell, Jack N.; Wang, Jing; Jones, Cheyenne A.; Csaki, Grace T.; Florian, Andrea C.; Romer, Alexander S.; Bryant, Daniel L.; Farone, Anthony L.; Liu, Qi; Tansey, William P.; Weissmiller, April M.
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Discovery of Potent Orally Bioavailable WD Repeat Domain 5(WDR5) Inhibitors Using a Pharmacophore-Based Optimization
err2022-04-18
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errTeuscher, Kevin B.; Meyers, Kenneth M.; Wei, Qiangqiang; Mills, Jonathan J.; Tian, Jianhua; Alvarado, Joseph; Sai, Jiqing; Van Meveren, Mayme; South, Taylor M.; Rietz, Tyson A.; Zhao, Bin; Moore, William J.; Stott, Gordon M.; Tansey, William P.; Lee, Taekyu; Fesik, Stephen W.
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Synergistic action of WDR5 and HDM2 inhibitors in SMARCB1-deficient cancer cells
err2022-03-03
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errOAAI
errFlorian, Andrea C.; Woodley, Chase M.; Wang, Jing; Grieb, Brian C.; Slota, Macey J.; Guerrazzi, Kiana; Hsu, Chih-Yuan; Matlock, Brittany K.; Flaherty, David K.; Lorey, Shelly L.; Fesik, Stephen W.; Howard, Gregory C.; Liu, Qi; Weissmiller, April M.; Tansey, William P.
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WIN site inhibition disrupts a subset of WDR5 function
err2022-02-03
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errSiladi, Andrew J.; Wang, Jing; Florian, Andrea C.; Thomas, Lance R.; Creighton, Joy H.; Matlock, Brittany K.; Flaherty, David K.; Lorey, Shelly L.; Howard, Gregory C.; Fesik, Stephen W.; Weissmiller, April M.; Liu, Qi; Tansey, William P.
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Multiple interactions of the oncoprotein transcription factor MYC with the SWI/SNF chromatin remodeler
err2021-04-30
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errWoodley, Chase M.; Romer, Alexander S.; Wang, Jing; Guarnaccia, Alissa D.; Elion, David L.; Maxwell, Jack N.; Guerrazzi, Kiana; McCann, Tyler S.; Popay, Tessa M.; Matlock, Brittany K.; Flaherty, David K.; Lorey, Shelly L.; Liu, Qi; Tansey, William P.; Weissmiller, April M.
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MYC regulates ribosome biogenesis and mitochondrial gene expression programs through its interaction with host cell factor-1MYC通过与宿主细胞因子-1的相互作用调节核糖体生物合成和线粒体基因表达程序
err2021-01-08
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errPopay, Tessa M.; Wang, Jing; Adams, Clare M.; Howard, Gregory Caleb; Codreanu, Simona G.; Sherrod, Stacy D.; McLean, John A.; Thomas, Lance R.; Lorey, Shelly L.; Machida, Yuichi J.; Weissmiller, April M.; Eischen, Christine M.; Liu, Qi; Tansey, William P.
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Impact of WIN site inhibitor on the WDR5 interactome
err2021-01-01
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errGuarnaccia, Alissa D.; Rose, Kristie L.; Wang, Jing; Zhao, Bin; Popay, Tessa M.; Wang, Christina E.; Guerrazzi, Kiana; Hill, Salisha; Woodley, Chase M.; Hansen, Tyler J.; Lorey, Shelly L.; Shaw, J. Grace; Payne, William G.; Weissmiller, April M.; Olejniczak, Edward T.; Fesik, Stephen W.; Liu, Qi; Tansey, William P.
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Discovery of WD Repeat-Containing Protein 5 (WDR5)-MYC Inhibitors Using Fragment-Based Methods and Structure-Based Design
err2020-03-30
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errSimon, Selena Chacon; Wang, Feng; Thomas, Lance R.; Phan, Jason; Zhao, Bin; Olejniczak, Edward T.; Macdonald, Jonathan D.; Shaw, J. Grace; Schlund, Caden; Payne, William; Creighton, Joy; Stauffer, Shaun R.; Waterson, Alex G.; Tansey, William P.; Fesik, Stephen W.
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WDR5 is a conserved regulator of protein synthesis gene expression
err2020-01-30
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errBryan, Audra F.; Wang, Jing; Howard, Gregory C.; Guarnaccia, Alissa D.; Woodley, Chase M.; Aho, Erin R.; Rellinger, Eric J.; Matlock, Brittany K.; Flaherty, David K.; Lorey, Shelly L.; Chung, Dai H.; Fesik, Stephen W.; Liu, Qi; Weissmiller, April M.; Tansey, William P.
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Discovery and Structure-Based Optimization of Potent and Selective WD Repeat Domain 5 (WDR5) Inhibitors Containing a Dihydroisoquinolinone Bicyclic Core
err2019-12-20
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errTian, Jianhua; Teuscher, Kevin B.; Aho, Erin R.; Alvarado, Joseph R.; Mills, Jonathan J.; Meyers, Kenneth M.; Gogliotti, Rocco D.; Han, Changho; Macdonald, Jonathan D.; Sai, Jiqing; Shaw, J. Grace; Sensintaffar, John L.; Zhao, Bin; Rietz, Tyson A.; Thomas, Lance R.; Payne, William G.; Moore, William J.; Stott, Gordon M.; Kondo, Jumpei; Inoue, Masahiro; Coffey, Robert J.; Tansey, William P.; Stauffer, Shaun R.; Lee, Taekyu; Fesik, Stephen W.
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Interaction of the oncoprotein transcription factor MYC with its chromatin cofactor WDR5 is essential for tumor maintenance
err2019-11-25
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errThomas, Lance R.; Adams, Clare M.; Wang, Jing; Weissmiller, April M.; Creighton, Joy; Lorey, Shelly L.; Liu, Qi; Fesik, Stephen W.; Eischen, Christine M.; Tansey, William P.
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