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Keiji Furuuchi

eisai co ltd

22H指数
94论文数
2.2K被引数
收录论文 31
发表时间
Farletuzumab ecteribulin and MORAb-109, folate receptor alpha and mesothelin targeting antibody-drug conjugates, show activity in poor prognosis gynaecological cancer modelsFarletuzumab ecteribulin和MORAb-109,靶向叶酸受体α和间皮素的抗体-药物偶联物,在预后不良的妇科癌症模型中显示出活性。
err2025-03-12
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errOAAI
errNesic, Ksenija; Rybinski, Katherine; Ratnayake, Gayanie; Ho, Gwo-Yaw; Lim, Ratana; Radke, Marc; Neagle, Chloe; Swisher, Elizabeth M.; Wakefield, Matthew J.; Barker, Holly E.; Furuuchi, Keiji; Scott, Clare L.; Vandenberg, Cassandra J.
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Potential Mechanisms of Interstitial Lung Disease Induced by Antibody-Drug Conjugates Based on Quantitative Analysis of Drug Distribution
err2024-10-25
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PREAI
errKoganemaru, Shigehiro; Fuchigami, Hirobumi; Morizono, Chihiro; Shinohara, Hiroko; Kuboki, Yasutoshi; Furuuchi, Keiji; Uenaka, Toshimitsu; Doi, Toshihiko; Yasunaga, Masahiro
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Intra-tissue quantitative analysis using LC/MS will determine the mechanisms of interstitial pneumonia induced by antibody-drug conjugates
err2024-03-22
err1
PREAI
errKoganemaru, Shigehiro; Fuchigami, Hirobumi; Morizono, Chihiro; Shinohara, Hiroko; Kuboki, Yasutoshi; Furuuchi, Keiji; Uenaka, Toshimitsu; Doi, Toshihiko; Yasunaga, Masahiro
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Phase I biomarker analysis of farletuzumab ecteribulin (FZEC), formerly MORAb-202, effects on cancer responses in patients with platinum resistant ovarian cance
err2023-12-01
err0
PREAI
errZhang, Yan; Zimmermann, Bob; Li, Shuyu; Uenaka, Toshimitsu; Furuuchi, Keiji; Yonemori, Kan; Shimizu, Toshio; Nishio, Shin; Yunokawa, Mayu; Matsumoto, Koji; Takehara, Kazuhiro; Hasegawa, Kosei; Hirashima, Yasuyuki; Kato, Hidenori; Otake, Yohei; Miura, Takuma; Matsui, Junji; Li, Meijuan
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Antitumor activity of farletuzumab ecteribulin in a panel of endometrial cancer patient-derived xenografts with four different molecular subtypes
err2023-10-01
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errOAAI
errHasegawa, K.; Yagishita, S.; Shintani, D.; Yoshida, H.; Suzuki, M.; Sato, S.; Ogasawara, A.; Nishikawa, T.; Yonemori, K.; Yasuda, M.; Furuuchi, K.; Uenaka, T.; Hamada, A.
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Preclinical development of BB-1701, a HER2-tageting eribulin-containing ADC with potent bystander effect and ICD activity
err2023-04-04
err1
PREAI
errWang, Yang; Xia, Bing; Cao, Lixia; Yang, Jianfeng; Feng, Cui; Jiang, Fangdun; Li, Chen; Gu, Lixia; Yang, Yifan; Tian, Jing; Cheng, Cindy; Furuuchi, Keiji; Fulmer, James; Verdi, Arielle; Rybinski, Katherine; Soto, Allis; Albone, Earl; Uenaka, Toshimitsu; Gong, Likun; Liu, Tingting; Qin, Qiuping; Wei, Ziping; Zhou, Yuhong
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MORAb-202, an antibody-drug-conjugate (ADC) targeting folate receptor alpha (FRα), exhibits durable anti-tumor efficacy in PDx models of TNBC
err2022-02-15
err1
PREAI
errFuruuchi, Keiji; Rybinski, Katherine; Fulmer, James; Moriyama, Tomoyuki; Drozdowski, Brian; Soto, Allis; Fernando, Shawn; Wilson, Kerrianne; Milinichik, Andrew; Dula, Mary Lou; Tanaka, Keigo; Cheng, Xin; Albone, Earl; Uenaka, Toshimitsu
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Folate receptor α increases chemotherapy resistance through stabilizing MDM2 in cooperation with PHB2 that is overcome by MORAb-202 in gastric cancer
err2021-06-01
err12
errOAAI
errSakai, Hitomi; Kawakami, Hisato; Teramura, Takeshi; Onodera, Yuta; Somers, Elizabeth; Furuuchi, Keiji; Uenaka, Toshimitsu; Kato, Ryoji; Nakagawa, Kazuhiko
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MORAb-109: A site-specific eribulin-conjugated ADC targeting human mesothelin
err2020-09-01
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errAlbone, E.; Cheng, X.; Verdi, A.; Jacob, S.; Fernando, S.; Furuuchi, K.; Fulmer, J.; Soto, A.; Drozdowski, B.; Mano, Y.; Nakatani, Y.; Uenaka, T.
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MORAb-202, an Antibody-Drug Conjugate Utilizing Humanized Anti-human FRα Farletuzumab and the Microtubule-targeting Agent Eribulin, has Potent Antitumor Activity
err2018-12-03
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errOAAI
errCheng, Xin; Li, Jing; Tanaka, Keigo; Majumder, Utpal; Milinichik, Andrew Z.; Verdi, Arielle C.; Maddage, Christopher J.; Rybinski, Katherine A.; Fernando, Shawn; Fernando, Danielle; Kuc, Megan; Furuuchi, Keiji; Fang, Frank; Uenaka, Toshimitsu; Grasso, Luigi; Albone, Earl F.
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MORAb-202, a folate receptor-alpha (FRA)-targeting antibody-eribulin drug conjugate (ADC), exhibits durable antitumor activity and payload-mediated bystander effects on the tumor microenvironment in triple-negative breast cancer
err2018-07-01
err0
PREAI
errFuruuchi, Keiji; Cheng, Xin; Rybinski, Katherine; Moriyama, Tomoyuki; Fulmer, James; Maddage, Chris; Milinichik, Andrew; Tanaka, Keigo; Lai, George; Dula, Mary Lou; Fernando, Danielle; Grasso, Luigi; Albone, Earl; Uenaka, Toshimitsu
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Morab-202, a folate receptor alpha-targeted antibody-drug conjugate, shows a highly potent activity against a panel of FRA-expressing tumors
err2018-07-01
err1
PREAI
errMignard, Caroline; Durix, Coralie; Rybinski, Katherine; Cheng, Xin; Furuuchi, Keiji; Albone, Earl; Uenaka, Toshimitsu; de Boisferon, Marc Hillairet
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Antitumor activity of new antibody-drug conjugate with eribulin in triple-negative breast cancer PDX
err2018-01-01
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PREAI
errde Boisferon, Marc Hillairet; Mignard, Caroline; Durix, Coralie; Uenaka, Toshimitsu; Rybinski, Katherine; Cheng, Xin; Furuuchi, Keiji; Albone, Eart
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MORAb-202: a folate receptor alpha (FRA)-targeting antibody-drug conjugate, exhibiting targeted antitumor activity and bystander elimination of cancer-associated fibroblasts
err2018-01-01
err1
PREAI
errRybinski, Katherine A.; Maddage, Christopher; Cheng, Xin; Albone, Earl; Grasso, Luigi; Furuuchi, Keiji; Uenaka, Toshimitsu
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Structural basis for ligand-mediated mouse GITR activation
err2008-01-15
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errOAAI
errZhou, Zhaocai; Tone, Yukiko; Song, Xiaomin; Furuluchi, Keiji; Lear, James D.; Waldmann, Herman; Tone, Masahicle; Greene, Mark I.; Murali, Ramachandran
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Smad3 and NFAT cooperate to induce Foxp3 expression through its enhancer
err2007-12-23
err779
PREAI
errTone, Yukiko; Furuuchi, Keiji; Kojima, Yoshitsugu; Tykocinski, Mark L.; Greene, Mark I.; Tone, Masahide
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OX40 gene expression is up-regulated by chromatin remodeling in its promoter region containing Sp1/Sp3, YY1, and NF-κB binding sites
err2007-08-01
err26
errOAAI
errTone, Yukiko; Kojima, Yoshitsugu; Furuuchi, Keiji; Brady, Maya; Yashiro-Ohtani, Yumi; Tykocinski, Mark L.; Tone, Masahide
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