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Maurizio Pellecchia

university of california riverside

61H指数
361论文数
1.4W被引数
收录论文 145
发表时间
Covalent Targeting of Histidine Residues: A Ligand-First Approach组氨酸残基的共价靶向:一种配体优先的方法
err2026-04-29
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PREAI
errGiulia Alboreggia; Emma L. Atienza; Kendall Muzzarelli; Zahra Assar; Maurizio Pellecchia
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Pre-clinical evaluation of a potent and effective Pin1-degrading agent in pancreatic cancer胰腺癌中一种强效且有效的Pin1降解剂的体外评估
err2025-11-01
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errOAAI
errAlboreggia, Giulia; Li, Tiane; Prentiss, Anne Marie; Udompholkul, Parima; Xia, Frank; Synold, Tim; Wu, Jun; Feng, Mingye; Raoof, Mustafa; Pellecchia, Maurizio
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Constrained β-Hairpins Targeting the EphA4 Ligand Binding Domain
err2024-12-10
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errOAAI
errPrentiss, Anne Marie; Baggio, Carlo; Pagett, James; Kulinich, Anna O.; Ethell, Iryna M.; Muzzarelli, Kendall; Assar, Zahra; Pellecchia, Maurizio
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Covalent Targeting of Histidine Residues with Aryl Fluorosulfates: Application to Mcl-1 BH3 Mimetics
err2024-11-12
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errOAAI
errAlboreggia, Giulia; Udompholkul, Parima; Atienza, Emma L.; Muzzarelli, Kendall; Assar, Zahra; Pellecchia, Maurizio
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Histidine-Covalent Stapled Alpha-Helical Peptides Targeting hMcl-1
err2024-05-02
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errOAAI
errAlboreggia, Giulia; Udompholkul, Parima; Baggio, Carlo; Muzzarelli, Kendall; Assar, Zahra; Pellecchia, Maurizio
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Structure Studies of Suicide Inhibitors Bound to Human Pin1
err2024-03-01
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errOAAI
errBlaha, Gregor; Alboreggia, Giulia; Rodriguez, Isaac; Pellecchia, Maurizio
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Mixture-Based Screening of Focused Combinatorial Libraries by NMR: Application to the Antiapoptotic Protein hMcl-1
err2023-07-19
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errOAAI
errAlboreggia, Giulia; Udompholkul, Parima; Baggio, Carlo; Pellecchia, Maurizio
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Characterization of a Potent and Orally Bioavailable Lys-Covalent Inhibitor of Apoptosis Protein (IAP) Antagonist
err2023-06-01
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errOAAI
errUdompholkul, Parima; Garza-Granados, Ana; Alboreggia, Giulia; Baggio, Carlo; McGuire, Jack; Pegan, Scott D. D.; Pellecchia, Maurizio
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Targefrin: A Potent Agent Targeting the Ligand Binding Domain of EphA2
err2022-11-04
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errOAAI
errBaggio, Carlo; Udompholkul, Parima; Gambini, Luca; Pellecchia, Maurizio
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Lysine Covalent Antagonists of Melanoma Inhibitors of Apoptosis Protein
err2021-10-27
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PREAI
errUdompholkul, Parima; Baggio, Carlo; Gambini, Luca; Alboreggia, Giulia; Pellecchia, Maurizio
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NMR-Guided Design of Potent and Selective EphA4 Agonistic Ligands
err2021-07-22
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errOAAI
errBaggio, Carlo; Kulinich, Anna; Dennys, Cassandra N.; Rodrigo, Rochelle; Meyer, Kathrin; Ethell, Iryna; Pellecchia, Maurizio
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Effective Tumor Targeting by EphA2-Agonist-Biotin-Streptavidin Conjugates
err2021-06-17
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errOAAI
errUdompholkul, Parima; Baggio, Carlo; Gambini, Luca; Sun, Yu; Zhao, Ming; Hoffman, Robert M.; Pellecchia, Maurizio
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Design, Synthesis, and Structural Characterization of Lysine Covalent BH3 Peptides Targeting Mcl-1
err2021-04-02
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errOAAI
errGambini, Luca; Udompholkul, Parima; Baggio, Carlo; Muralidharan, Aruljothi; Kenjic, Nikola; Assar, Zahra; Perry, J. Jefferson P.; Pellecchia, Maurizio
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Therapeutic Targeting of MMP-12 for the Treatment of Chronic Obstructive Pulmonary Disease
err2020-10-27
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errOAAI
errBaggio, Carlo; Velazquez, Jalene V.; Fragai, Marco; Nordgren, Tara M.; Pellecchia, Maurizio
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Stability and Cell Permeability of Sulfonyl Fluorides in the Design of Lys-Covalent Antagonists of Protein-Protein Interactions
err2020-10-13
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errGambini, Luca; Udompholkul, Parima; Salem, Ahmed F.; Baggio, Carlo; Pellecchia, Maurizio
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Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-7
err2020-06-28
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errGuetschow, Michael; Vanden Eynde, Jean Jacques; Jampilek, Josef; Kang, CongBao; Mangoni, Arduino A.; Fossa, Paola; Karaman, Rafik; Trabocchi, Andrea; Scott, Peter J. H.; Reynisson, Johannes; Rapposelli, Simona; Galdiero, Stefania; Winum, Jean-Yves; Brullo, Chiara; Prokai-Tatrai, Katalin; Sharma, Arun K.; Schapira, Matthieu; Azuma, Yasu-Taka; Cerchia, Laura; Spetea, Mariana; Torri, Giangiacomo; Collina, Simona; Geronikaki, Athina; Garcia-Sosa, Alfonso T.; Vasconcelos, M. Helena; Sousa, Maria Emilia; Kosalec, Ivan; Tuccinardi, Tiziano; Duarte, Iola F.; Salvador, Jorge A. R.; Bertinaria, Massimo; Pellecchia, Maurizio; Amato, Jussara; Rastelli, Giulio; Gomes, Paula A. C.; Guedes, Rita C.; Sabatier, Jean-Marc; Estevez-Braun, Ana; Pagano, Bruno; Mangani, Stefano; Ragno, Rino; Kokotos, George; Brindisi, Margherita; Gonzalez, Florenci V.; Borges, Fernanda; Miloso, Mariarosaria; Rautio, Jarkko; Munoz-Torrero, Diego
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Potential Therapeutic Targeting of Coronavirus Spike Glycoprotein Priming
err2020-05-22
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errOAAI
errBarile, Elisa; Baggio, Carlo; Gambini, Luca; Shiryaev, Sergey A.; Strongin, Alex Y.; Pellecchia, Maurizio
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