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Structural Optimization of Cholesteryl ester transfer protein inhibitors: From Early Scaffolds to Advanced Clinical Candidates
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DOI:10.1016/j.ejmech.2026.118920.png)
Abstract
En 中文
• CETP inhibitors modulate HDL and LDL to reduce cardiovascular risk • Clinical trials reveal mixed efficacy and safety among CETP inhibitors • New-generation CETP inhibitors show improved outcomes and tolerability • Mechanistic insights explain failures of early CETP inhibitor candidates • CETP inhibition remains a promising strategy in lipid management
Keywords:
CETP inhibitors
HDL
LDL
lipid management
clinical trials
Journal
IF:
5.9
Papers:
1.7W
Citations:
6.0W
