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Structural Optimization of Cholesteryl ester transfer protein inhibitors: From Early Scaffolds to Advanced Clinical Candidates

delete2026-05-08
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PRE
AI
M
Mahla Abdollahzadeh
M
Mahin Ramezani
M
Mahdi Hatamipour *
DOI:10.1016/j.ejmech.2026.118920delete
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Abstract

Abstract

En 中文
• CETP inhibitors modulate HDL and LDL to reduce cardiovascular risk • Clinical trials reveal mixed efficacy and safety among CETP inhibitors • New-generation CETP inhibitors show improved outcomes and tolerability • Mechanistic insights explain failures of early CETP inhibitor candidates • CETP inhibition remains a promising strategy in lipid management
Keywords:
CETP inhibitors
HDL
LDL
lipid management
clinical trials

Journal

European Journal of Medicinal Chemistry cover
European Journal of Medicinal Chemistry
IF:
5.9
Papers:
1.7W
Citations:
6.0W

Organization

M
Mashhad University of Medical Sciences
Scholars:
1.1W
Papers: 6.5K
Citations: 7.6K
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