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BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

IF2.2
Papers144
Citations
Journal Papers 142
Publication Date
Identification of TYK2 activators. Part 2: Optimization of terminal alkyne substituents to enhance activation potency
delete2026-07-07
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PREAI
deleteHirokazu Matsumoto; Tien-Cheng Wang; Fumio Nakajima; Haruka Taniguchi; Takayoshi Kinoshita; Masaaki Sawa
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Novel 1H-pyrrole-2,5-dione derivatives as potential anti-diabetic agents: design, synthesis, in vitro, in ovo, and molecular docking studies
delete2026-06-13
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PREAI
deleteDilan Gezer; Zeynep Ozyıldız; Zeliha Gokmen; Eda Dagsuyu; Ozlem Sacan; Remzi Okan Akar; Elifnur Gizem Yıldırım; Engin Ulukaya; Kaan Adacan; Aslı Kutlu
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A rapid and scalable microwave-assisted strategy for the synthesis of neocryptolepine and its analogues: Comprehensive bioactivity profiling
delete2026-06-02
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PREAI
deleteSiddhi Salgaonkar; Melita Rebello; Delicia Avilla Barretto; Supriya Tilvi; Vinod Mandrekar
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Cannabidiol-thiosemicarbazone exhibits dual tyrosinase inhibition and antioxidant activity in human skin-derived cells
delete2026-06-02
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PREAI
deleteMaytal Shabat-Simon; Oriyan Cohen; Larisa Yaval; Salam Hujerat; Paula Adriana Pitashny; Karen Jackson; Sanaa Musa
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Small molecule inhibition of CPSF3 may impact R-loop distribution and abundance
delete2026-05-28
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deleteCristina R. Hofman; Victor Tse; Jiaxin Hu; David R. Corey
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Disulfide bond formation between Cys22 and Cys44 in SARS-CoV-2 main protease
delete2026-05-25
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PREAI
deleteLauren R. Blankenship; Kai Yang; Chia-Chuan Dean Cho; Yi-Ju Penny Chen; Banumathi Sankaran; Wenshe Ray Liu
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Chlorophenylpyrazolone derivatives as novel PD-L1-targeted inhibitors of the PD-1/PD-L1 immune checkpoint
delete2026-05-25
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PREAI
deleteFrédérique Klupsch; Raphaël Le Biannic; Hassiba El Bouazzati; Romain Magnez; Morgane Rivoal; Bryan Thiroux; Morgane Tardy; Gérard Vergoten; Christian Bailly; Bruno Quesnel; Xavier Thuru; Natascha Leleu-Chavain; Régis Millet
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