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rsc med. chem.

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Papers123
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Journal Papers 168
Publication Date
Exploring the Antimycobacterial Profile of N-Alkyl Imidazoles
delete2026-06-24
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PREAI
deleteAlejandro I. Recio-Balsells; Gabriel Di Gresia; Marcelo Luciano Merli; Julia Alejandra Cricco; Hector R. Morbidoni; Guillermo R Labadie
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Discovery of Novel SIRT3 Inhibitors with MLLr Leukemia Inhibitory Potency
delete2026-06-24
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PREAI
deleteShaopeng Chen; Xinyang Wei; Honggang Li; Jiangying Cao; lei zhang
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From dual norepinephrine-dopamine reuptake inhibition to selective dopamine reuptake inhibitors: a case of aromatically substituted N; 2-cyclopentylamines
delete2026-06-24
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deleteMajlen A. Dilweg; Willem Jespers; Ameya S Kasture; Rongfang Liu; Tamara A. M. Mocking; Jelle G Van Der Ploeg; M M Baselier; Gerard Van Westen; Thomas Hummel; Sonja Sucic; Adriaan P. IJzerman; Laura H. Heitman; Daan van der Es
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Combining β2-AR agonism with butyrylcholinesterase inhibition; a synergistic neuroprotective action against Alzheimer's disease
delete2026-06-24
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PREAI
deleteAlice Wang; Thomas Curel; Sylvie Claeysen; Valentin Travers-Lesage; Marie Elodie Hélène Cadot; Audrey Davis; Jana Sopkova de Oliveira Santos; Fabrice Modeste; Xavier Brazzolotto; Florian Nachon; Patrick Dallemagne; Marc Since; Christophe Rochais
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Synthesis and Bioevaluation of Substituted 2; 11-dihydroimidazo[1′; 5′:1; 2]pyrido-[3; 4-b]indoles as antiplasmodial and antiproliferative agents
delete2026-06-24
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PREAI
deleteAdilakshmi Vutla; Akash Pandey; Amanullah Sayeed; Richa Shukla; Ashan Manhas; Niti Kumar; Sanjeev Meena; Dipak Datta; Sanjay Batra
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Discovery of Novel Indazole Derivatives with Antineuroinflammatory Activity
delete2026-06-24
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PREAI
deleteQing qing Zhang; Xixi Hou; Xuanwei Zhang; Yimian Wang; Yaquan Cao; Lan Wang; Longfei Mao
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Design and synthesis of N-3-substituted quinazolinone derivatives as anticancer agents targeting EGFR
delete2026-06-23
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PREAI
deletePritam Maity; Poonam Yadav; Joydeep Chatterjee; Madhurendra Kumar Katiyar; Umashanker Navik; Raj Kumar
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The Many Facets of Sustainability in Medicinal Chemistry: Our Personal Experience
delete2026-06-23
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deleteBianca Martinengo; Eleonora Diamanti; Elisa Uliassi; Maria Laura Bolognesi
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Targeted Degradation of Pin1 by an Antagonistic Peptide Enhance Gemcitabine Therapy in Pancreatic Cancer
delete2026-06-23
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PREAI
deleteMengting Chen; Xiangyu Chu; Haipeng Zhao; Lilusi Ma; Jie Meng; Yanlian Yang; Qiaojun Fang; Xiaocui Fang; Chen Wang
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Rational design of an environment-sensitive fluorescent probe for monitoring butyrylcholinesterase activity and its application in Alzheimer's disease
delete2026-06-17
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PREAI
deleteNing Guo †; Feng Wang †; Yu Wang; Jiahao Du; Qingwen Zhang; Wenting Cao; Jiongtao Su; Fenqin Zhao; Junfeng Wang; Xiaobin Pang; Yuemin Zhou; Lin Yan
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From AlphaFold to site-selective inhibition of DNA methylation in glioblastoma multiforme
delete2026-06-11
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PREAI
deleteJean-Maxime Besson; Alain Chavanieu; Arulraj Nadaradjane; Pierre-François Cartron; Marie Lopez
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New roxadustat amino acid drug conjugation derivatives: molecular docking; molecular dynamics simulation and in vitro assay
delete2026-06-11
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PREAI
deleteMarjan Samadi; Azizollah Habibi; Leila Karami; Soroush Sardari; Ramin Ebrahimi Kiasari; Ghazaleh Ghavami; Mohammad Shahcheragh
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Discovery of a Potent Dual Target CDK8 and Cyclic C PROTAC Degrader for Treatment of Colorectal Cancer
delete2026-06-10
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PREAI
deleteXingxing Zhang; Qingsong Chen; Cencen Lei; Da Long Jin; Hao Dong Liu; Yumeng Wang; Chenyu zhao; Liping Zhi; Xinhua Liu
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Targeting DNA-PK: medicinal chemistry insights into small-molecule inhibitor discovery and optimisation
delete2026-06-09
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deleteElle Watson; Jack R. R. Hutchinson; Suzannah J. Harnor; Luke Gaughan; Celine Cano
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Synthesis; molecular modelling and evaluation of (-)-isopulegolbased 2; 4-diaminopyrimidines as promising Aurora kinase inhibitors
delete2026-06-04
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deleteTam Minh Le; Nikoletta Szemerédi; Gabriella Spengler; Minh Canh Nguyen; Huynh Nguyen Khanh Tran; Khac-Minh Thai; Zsolt Szakonyi
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Novel Hydroxytyrosol Esters as Potential Anti-Amyloid and Neuroprotective Agents for Alzheimer's Disease
delete2026-06-04
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deleteIoanna Kalpaktsi; Anthi Panara; Barbara Mavroidi; Garcia Niforos; Amalia D Kalampaliki; Ioanna C Vlachogianni; Eleftheria A Georgiou; Elizabeth Fragopoulou; Anthony Tarbopoulos; AL Skaltsounis; Maria Pelecanou; K Palikaras; Evagelos Gikas; Ioannis K. Kostakis
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Novel Urea- and Piperazine-Functionalized Alepterolic Acid Derivatives: Synthesis; Anticancer Activity; and Mechanism of Action
delete2026-06-03
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PREAI
deleteBinbin Zhang; Yating Jia; Siyu Qiu; Yanchun Sun; Lian Ma; Peixin Wang; Zixuan Tong; Fengjiao Wang; Guozheng Huang; Jianguo Cao
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A Bakuchiol-Linked Tetrazole Exhibits Narrow-spectrum Activity Against Streptococcus pneumoniae
delete2026-06-03
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PREAI
deleteNeha Sengar; Vidyadhar Pratap; Tuhin Sarkar; Vishnu Kriplani; Astha Gupta; Sanjay Mandal; Prasad V. Bharatam; Dulal Panda; Inder Pal Singh
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3-Hydroxypyrimidine-2; 4-dione derivatives as monkeypox virus resolvase (Mpr) inhibitors
delete2026-06-01
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PREAI
deleteMuhammad Syafiq Bin Shahari; Jacob P Mahoney; Ziyue Wang; Anil Pant; Ajit Jagtap; Roshan Katekar; Jiashu Xie; Zhilong Yang; Zhengqiang Wang
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