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European Journal of Medicinal Chemistry Reports cover

European Journal of Medicinal Chemistry Reports

IF4.1
Papers361
Citations626
Journal Papers 366
Publication Date
Synthesis, structure, photophysical, photochemical, and biological properties of hybrid macrocyclic structures containing two naphthalene moieties and a tri(ethylene glycol) tether
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deleteMarco Paolino; Jacopo Venditti; Gabriele Manenti; Mario Saletti; Alessandro Donati; Claudia Bonechi; Germano Giuliani; Chiara Botta; Stefania Lamponi; Valerio Ciccone; Maria Frosini; Sandra Donnini; Lucia Morbidelli; Riccardo Carletti; Filippo Sacchetta; Andrea Cappelli
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Synthesis, anti-cancer activity, Pim-3 inhibitory potency and zebrafish larvae toxicity evaluation of indolopyrazolocarbazole derivatives
delete2026-09-02
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deleteThéo Frazier; Elisabeth Pereira; Reidun Aesoy; Andrea Trentani; Francis Giraud; Lars Herfindal; Fabrice Anizon; Pascale Moreau
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Pyrazoline- and Hydrazone-Linked Thiazole-Triazole Hybrids as Potent Dual-Stage Antileishmanial Agents with Antifolate Activity
delete2026-09-01
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deleteEsraa A. Abdelsalam; Wagdy M. Eldehna; Sherif F. Hammad; Nicolas Masurier; Tamer M. Ibrahim; Kikuko Amagase; Sherry N. Nasralla; Yara E. Mansour; Hatem A. Abdel-Aziz; Adnan A. Bekhit; Radwan El-Haggar
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Small-molecule ferroptosis modulators in oncology: Design principles, evidence standards, and translational opportunities
delete2026-08-12
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deleteTania Ciaglia; Valeria Napolitano; Francesca Di Matteo; Alessia Bertamino; Isabel Maria Gomez Monterrey
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Design, synthesis and antibacterial evaluation of amphiphilic 1,2,4-oxadiazole-based pyridinium salts
delete2026-08-12
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deleteSara Amata; Virginia Talarico; Gaspare Crisà; Giuseppe Pizzolanti; Andrea Pace; Antonio Palumbo Piccionello; Cinzia Calà; Carla Rizzo
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Discovery and pharmacological evaluation of a novel series of chromenopyrazole-based GPR55 modulators in an androgen-driven model of female metabolic dysfunction
delete2026-08-06
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deleteFrancisco J. Ponce-Díaz; Francisco Ruiz-Pino; Aitor Herraiz; Beatriz Romero; Laura Cerero-Tejero; Adela García-Martín; Simon Porzio-Gonzalez; Paula Morales; Miguel A. Sánchez-Garrido; Marina Pulido; Nadine Jagerovic; Manuel Tena-Sempere; Eduardo Muñoz
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Small-molecule antibacterials and resistance-modifying agents
delete2026-08-01
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PREAI
deleteZelisko, Nataliya; Kovalenko, Iryna; Lesyk, Danylo; Vilenskyi, Andrii; Lavryk, Galyna; Rumynska, Tetyana; Zubach, Olena; Lesyk, Roman
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Integrative in silico and experimental identification of non-covalent UBE2N inhibitors enhancing PARP inhibitor sensitivity
delete2026-07-30
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deleteCôme Ghadi; Shafi Ullah Khan; Léonie Ibazizene; Florian Schwalen; Charline Kieffer; Peggy Suzanne; Julie Jaouen; Hassiba Bouafia; Xavier Thuru; Marie Cornu; Cedric Lecoutey; Matthieu Meryet-Figuiere; Anne Sophie Voisin-Chiret; Louis-Bastien Weiswald; Jana Sopkova-de Oliveira Santos
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New C-30 secondary and tertiary amines of betulin with selective antiproliferative activity toward hematological malignancies - Synthesis and biological evaluation
delete2026-07-28
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deleteJan Bachořík; Ivo Frydrych; Soňa Gurská; Štěpán Dostál; Jan Pokorný; Adam Přibylka; Martina Medvedíková; Petr Džubák; Marián Hajdúch; Milan Urban
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Marine natural products for antifungal drug discovery: An updated review (2015–2025)
delete2026-07-15
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deleteSalma A. Haggag; Ahmed K. ElHady; Nardine Adel; Mirna Y. Abouomar; Abdelrhman M. Shoman; Ebaa M. El-Hossary; Ashraf H. Abadi; Usama Ramadan Abdelmohsen; Tsong-Long Hwang; Mohammad Abdel-Halim
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A MCC950 analogue inflammasome inhibitor reduces the foreign body reaction against neural implants
delete2026-07-10
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deleteJose Crugeiras; Chiara Bisquoli; María Rodríguez-Brañas; Bruno Rodríguez-Meana; Tiziano De Ventura; Neus Hernández; Jessica Jaramillo; Alice Honovich; Ignacio Delgado-Martínez; Natalia Lago; Hanna Karlsson-Fernberg; Maria Asplund; Stefano Carli; Claudio Trapella; Giulia Turrin; Xavier Navarro
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Beyond arginine count: Rational engineering of amphipathic macrocyclic CPPs with enhanced intracellular delivery and endosomal escape
delete2026-07-04
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deleteDuc Tai Nguyen; Michael Desgagné; Ulrike Froehlich; Andréanne Laniel; Christine Lavoie; Pierre-Luc Boudreault
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Exploring sulfonamide carboxamides as promising leads for antimalarial drug development
delete2026-07-01
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deleteNyoyoko, Immaculata Fabian; Ezema, Benjamin Ebere; Onoabedje, Efeturi Abraham; Ezema, Chidinma Grace; Eze, Florence Uchenna; Conradie, Jeanet; Ugwu, David Izuchukwu
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Design, synthesis, in vitro, and in silico assays of new 4-phenylpiperazine-coumarin-triazole-acetamide hybrids as potent tyrosinase inhibitors
delete2026-06-29
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deleteMohammad Mahdi Aghanour Ashtiani; Somaye Karimian; Aida Iraji; Navid Dastyafteh; Maryam Mohammadi-Khanaposhtani; Bagher Larijani; Mohammad Mahdavi; Peyman Salehi
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Synthesis and biological evaluation of C5-(1-substituted-1,2,3-triazol-4-yl)-uridines and their phosphoramidate prodrugs
delete2026-06-10
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deleteEvan Saillard; Vincent Roy; Patrick Favetta; Dawid Warszycki; Andrzej J. Bojarski; Leentje Persoons; Dirk Daelemans; Steven De Jonghe; Luigi A. Agrofoglio
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Synthesis and first evaluation of new favipiravir analogs based on cyclic amidrazones scaffolds
delete2026-06-09
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deleteMargaux Boutin; Jacques Lebreton; Edeildo Ferreira da Silva-Júnior; Andrés Pizzorno; Aurélien Traversier; Manuel Rosa-Calatrava; Arnaud Tessier
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Small Molecule Agonists of TREM2 Reprogram Microglia and Protect Synapses in Human Alzheimer’s Models
delete2026-06-09
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deleteHossam Nada; Shaoren Yuan; Farida El Gaamouch; Sungwoo Cho; Moustafa T. Gabr
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