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ChemMedChem

IF3.4
Papers5104
Citations10115
Journal Papers 5097
Publication Date
Beyond the Active Site: First-In-Class Leishmania Infantum Trypanothione Reductase Dimerization Disruptors as Antileishmanial Leads
delete2026-09-29
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deleteMaría-José Camarasa; Miguel Maldonado; Alvaro de la Cruz-Potenciano; Sonia de Castro
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Discovery of Symmetrical o-Methylpyridine Substituted Tertiary Amines and Dy(III) Complexes as Metallo-β-Lactamase Inhibitor and Antimicrobial
delete2026-09-29
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PREAI
deleteLe Zhai; Jiazhu Chigan; Yao Zhao; Hua-Ping Xie; Yi-Qiang Wu; Sheng Zhang; Ke-Wu Yang
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Assessment of the Binding Affinity of Covalent Inhibitors of Cruzain and Cathepsin L Using Relative Binding Free Energy
delete2026-09-29
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deleteYan Carvalho Magno; Luiz Fernando Barbosa; Maycon Vinicius Damasceno de Oliveira; Jerônimo Lameira; Carlos A. Montanari
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The Sigma-1 Receptor as a Novel Target in the Neuroprotective Effects of Cannabidiol and Cannabigerol Against Mitochondrial Damage in Cultured Cerebellar Granule Neurons
delete2026-09-29
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PREAI
deleteVictoria Oviedo-Pino; Mariana Pazos; Giselle Prunell; Carlos Ferreiro-Vera; Verónica Sánchez de Medina; Miguel Reyes-Parada; David Ramírez; Cecilia Scorza; Carolina Echeverry
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Toward Combating Pseudomonas aeruginosa Infection, the Creation of Azithromycin Derivatives Based on a Trojan Horse Strategy
delete2026-09-29
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PREAI
deleteAoi Kimishima; Rina Suzuki; Taichi Kamo; Paul Wasuwanich; Hidehito Matsui; Sota Negami; Sota Honma; Yukiko Ujie; Naozumi Kondo; Hideaki Hanaki; Yukihiro Asami
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Design, Synthesis, and Biological Evaluation of Pyrazolyl Thioureas (PTUs) as SIRT1 and SIRT2 Inhibitors
delete2026-09-25
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deleteMatteo Lusardi; Cecilia Astigiano; Deianira Bellitto; Matteo Raineri; Giorgia Guccione; Annalisa Salis; Elena Cichero; Chiara Brullo; Marco Ponassi; Santina Bruzzone; Andrea Spallarossa
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Potent Caspase-1 Antagonists From Dihydropyridine Derivatives: In Vitro Fluorescence Assays and Cell Imaging
delete2026-09-21
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PREAI
deleteKittiporn Nakprasit; Thitiporn Pattarakankul; Tanapat Palaga; Thanapon Charoenwongpaiboon; Waroton Paisuwan; Kavisara Srithadindang; Rachanon Eakprachasin; Islah Muttaqin; Pattraporn Chobpradit; Sucharat Sanongkiet; Mongkol Sukwattanasinitt; Chanakan Tongsook; Anawat Ajavakom
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Synthesis, Biological Evaluation, and Molecular Modeling of Novel Pyrimidine Scaffolds as Prospective Anticancer and Antimicrobial Agents
delete2026-09-18
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PREAI
deleteVishwa Thakor; Pratik Patel; Megha Patel; Bhavin Patel; Tarun Patel; Paresh Patel
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Linker Optimization of cMYC RIBOTAC for Efficient cMYC Modulation
delete2026-09-17
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PREAI
deleteSivakumar Komachankandy; Jinseo Heo; Yerin Kim; Wonpil Im; Yeongju Lee
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Metal-Based Photosensitizers as Emerging Antibacterial Agents for Infected Wound Healing
delete2026-09-11
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PREAI
deleteArif Ali Mandal; Bhaskar Bhusan Das; Ishwar Singh; Samya Banerjee
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Phosphorylated Analogs of Paracetamol and Their Anti-Inflammatory Potential
delete2026-09-11
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PREAI
deleteOsvaldo León de la Cruz; Gabriel Alfonso Gutiérrez-Rebolledo; Carlos Zepactonal Gómez Castro; Ángel Daniel Campos Juárez; Porfirio Alonso Ruiz-Hurtado; Josué Rodríguez-Lozada; José Luis Castrejón-Flores; María Guadalupe Ramírez-Sotelo; Marco Franco-Pérez; Angel Zamudio-Medina
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Novel Steroidal (Thio)barbiturate Hybrids: From Design to Preclinical Assessment in Tumor Therapy
delete2026-09-11
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PREAI
deleteAlexandra Varges; João Serrano; Paula Arias; Pedro Soeiro; Marla Machava; Inês Figueiredo; Eurico Lima; Gilberto Alves; Adriana Oliveira Santos; Renato Boto; Paulo Almeida; Samuel Silvestre; Mariana Matias
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Synthesis and Assessment of the Enantioselectivity in Antitumor Activity of a Library of Novel Chiral Flavone Derivatives
delete2026-09-11
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PREAI
deleteCláudia Pinto; Flávia Barbosa; João Machado; Andrea Cunha; Patrícia M. A. Silva; Mariangela Agamennone; Hassan Bousbaa; Honorina Cidade; Odília Queirós; Maria Elizabeth Tiritan
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Synthesis and Evaluation of Peptoid-Based Compound Libraries as Inhibitors of Parasite Metallo-Aminopeptidases
delete2026-09-11
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deleteMirta Elisa Aguado; Gerardo M. Ojeda-Carralero; Mario Antonio Rodríguez; Isabella Rúa; Heisy Guerra; Edoardo Bailo Hernández; Guglielmo Coppola; Susana Alberti; Ariatne Rodríguez; Maikel Izquierdo; Christian Betzel; Filippo Pettazzi; Julieta Coro-Bermello; Erik V. Van der Eycken; Bernhard Westermann; Jorge González-Bacerio; Daniel G. Rivera
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Exploring the Anticancer Potential of Schiff Base Complexes: A Mini-Review
delete2026-09-10
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deleteAtif Ahmad; Anam; Marcos V. Palmeira-Mello; Sabir Khan; José Clayston Melo Pereira
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Synthesis and Biological Activity of Novel Aromatic Aminopropyl Lactams in Two Cancer Cell Models
delete2026-09-08
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PREAI
deleteM. Margarida Martins; Ruben Valente; Ruben Amaro; Maria S. Viana; Rita de Jesus; Bernardo Braga; Daniela Peixoto; Celina Schenkelberger; Matilde Simão; Pedro V. Baptista; Paula S. Branco; João Aires-de-Sousa; Alexandra R. Fernandes; Luísa M. Ferreira
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Phenols: From Replacing to Embracing
delete2026-09-08
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PREAI
deleteGilles Ouvry
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Ligand‑Based Virtual Screening Discovery of Thienopyrimidinone Derivatives as Allosteric nSMase2 Modulators and Antivirals Against West Nile Virus
delete2026-09-08
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deleteHadrián Álvarez-Fernández; Patricia Mingo-Casas; Ana-Belén Blázquez; Flavia Caridi; Miguel A. Martín-Acebes; María-Jesús Pérez-Pérez; Eva-María Priego
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