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ACS Medicinal Chemistry Letters

IF4
Papers4422
Citations9951
Journal Papers 4447
Publication Date
Uncompetitive Allosteric Inhibition of PTP1B by BP-1-102 Reveals a Potential Dual-Target Strategy toward the PTP1B–STAT3 Oncogenic Axis: Biochemical and Computational Evidence
delete2026-06-12
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deleteMartín González-Andrade; Rodolfo A. Lizárraga-Valadez; Alejandro Sosa-Peinado; Francisco Cortés-Benítez; Nathaly Vasquez-Martínez
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Novel Substituted Carboxamides as SSTR4 Agonists
delete2026-06-11
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deleteJian Rong; Steven H. Liang
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Design and Optimization of Benzoic Acid Inhibitors Targeting the EBNA1 DNA-Binding Interface
delete2026-06-11
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deleteGarry R. Smith; Mark E. McDonnell; Yan Zhang; Venkata Velvadapu; Shuai Chen; Lois Tolvinski; Julianna Deakyne; Samantha S. Soldan; Paul M. Lieberman; Allen B. Reitz; Troy E. Messick
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Discovery of MK-2118; a Small-Molecule Agonist of STING
delete2026-06-11
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deleteTimothy Henderson; Michael D. Altman; Alexei V. Buevich; Brandon Cash; Saso Cemerski; Wonsuk Chang; Yiping Chen; Matthew Childers; Jared Cumming; Peter J. Dandliker; Guo Feng; Andrew Haidle; Robert P. Hayes; Thu Ho; James P. Jewell; Ilona Kariv; Ian Knemeyer; Johnny Kopinja; Brian M. Lacey; Jason Laskey; Charles A. Lesburg; Rui Liang; Jongwon Lim; Brian J. Long; Min Lu; Yanhong Ma; Ellen C. Minnihan; Ryan D. Otte; Gregory O’Donnell; Bo-Sheng Pan; Samanthi A. Perera; Jennifer A. Piesvaux; Jeremy P. Presland; Laura Price; Larissa Rakhilina; Berengere Sauvagnat; Gottfried K. Schroeder; Sharad Sharma; B. Wesley Trotter; Sriram Tyagarajan; Hyun Woo; Daniel F. Wyss; Serena Xu; George H. Addona; David Jonathan Bennett
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Vasicine-Based Synergistic Antifungal Agents against FLC-Resistant Candida albicans Targeting Ras/cAMP/PKA Pathway
delete2026-06-10
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deleteDi Zhao; Wengang Wang; Zhichang Xu; Zewei Mao; Ruirui Wang; Huan Chen; Chunyan Hu
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Eco-Friendly Access to Indenodiazepinones from o-Formylynones and o-Phenylenediamines and Their Preliminary Antibacterial Activity
delete2026-06-07
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PREAI
deleteBilal Ahmad Ganaie; Debapriya Mukherjee; Alagesan Balasubramani; Pallab Ghosh; Raju S. Rajmani; Dipshikha Chakravortty; Goverdhan Mehta
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Design of PKC-Targeting Benzolactams as Gli Inhibitors
delete2026-06-04
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PREAI
deleteMarianna Haddad; Jo Chvatal; Alexandria Kifer; Jayannah Herdrich; McCarthy Poljak; Kelvin L. Billingsley
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Discovery of NKT2152; a Potent and Selective HIF-2α Inhibitor with Favorable Pharmacokinetic Properties
delete2026-06-04
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PREAI
deleteJiping Fu; Yigang He; Jing Lu; Hairong Wei; Wenfeng Sun; Jianlin Geng; Ke Liu; Jessica Jingchun Liu; Zhihong Liu; Keshi Wang; Jim Xiao; Zhenhai Gao; Yan Lou
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Synthesis of Nitazoxanide Derivatives as Potent and Orally Available HBx-DDB1 Inhibitors against Hepatitis B Virus
delete2026-06-04
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deleteSeong Gon Kim; Hyeon-Min Cha; Minwoo Kim; Inseong Jo; Soo Bong Han; Meehyein Kim; Wonseo Park; Youyoung Kim; Chunkyu Ko; Dong-Su Kim
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Structure-Guided Discovery of Novel Highly Potent and Selective MTA-Cooperative PRMT5 Inhibitors
delete2026-06-03
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PREAI
deleteChuping Huang; Min Liang; Ping Zhang; Gang Liu; Chenzhong Liao
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Call for Papers: Allosteric Modulators in Drug Discovery
delete2026-06-01
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deleteMaria-Jesus Blanco; Zoe Cournia; Rong Huang; Choong Yee Siew
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