Design, synthesis, and biological evaluation of novel coumarine-1,2,3-triazole hybrids as dual DNA gyrase/superoxide dismutase inhibitors: molecular docking, DFT, and ADMET investigations
Patel, Gaurav B.; Bhola, Yogesh O.; Dholaria, Piyush V.; Suthar, Arvindbhai R.; Bhatt, Dhavalkumar M.
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Save Tailored pyrazolone-oxadiazole frameworks: synthetic execution, functional enzyme studies, and comprehensive docking-DFT-based antidiabetic investigation
Iqbal, Tayyiaba; Habib, Mohamed A.; Khan, Shoaib; Rehman, Wajid; Bibi, Aisha; Hussain, Rafaqat; Ibrahim, Ahmed B. M.; Kayumov, Khasan
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Save Cyclization, amino acid coupling, docking-based virtual screening and SAR: showing a strategy of the structural modification for salvianic acid A
Wu, Jianhui; Zhang, Xiaoyi; An, Wenshuo; Yang, Yifan; Zhang, Peiwen; Wang, Yaonan; Zhao, Shurui; Feng, Qiqi; Zhao, Ming; Peng, Shiqi
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Save Unveiling the potential of zingerone-1,2,3-triazole derivatives as dual anticancer and COX-2 inhibitor: design, synthesis, and biological assessments
Alam, Mohammad Mahboob; Alsenani, Nawaf I.; Elhenawy, Ahmed A.; Hussien, Rania A.; Althagafi, Saif H.; Alqurashi, Esam A.; Elbehairi, Serag Eldin I.; Shati, Ali A.; Alfaifi, Mohammad Y.; Bashir, Seham Hassan; Nazreen, Syed
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Save Design, synthesis, and antidiabetic activity of new furan-clubbed 1,2,3-triazole derivatives as α-glucosidase inhibitors
Devi, Priya; Maity, Subhadip; Singh, Aastha; Mehan, Sidharth; Singh, Gurpreet; Asati, Vivek
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