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Future Medicinal Chemistry cover

Future Medicinal Chemistry

IF3.4
Papers2925
Citations6174
Journal Papers 3338
Publication Date
PROTACs in 2025: from the laboratory concept to clinical breakthrough
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deleteXu, Yan; Li, Xin-Yu; Song, Jian; Zhang, Sai-Yang
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Discovery of novel 2,4-diarylaminopyrimidine derivatives as FAK inhibitors with potent anti-cancer potency
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deleteLv, Yu-Zheng; Song, Jian; Zhang, Sai-Yang; Xu, Yan; Xi, Shou-Min
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Mechanosynthesis and computational studies of new imidazole-based selenium adducts as potential anticancer agents against human prostate and cervical cancer
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deleteAbbas, Ghazanfar; Bokhari, Tanveer Hussain; Iqbal, Muhammad Adnan; Rehman, Saima; Ali, Akbar
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Synthesis and biological profiling of novel quinoline-thiadiazole-thiazolone scaffolds as antimicrobial agents
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deleteModi, Hetali A.; Pathak, Dushyant V.; Suradiya, Pooja D.; Chhag, Darshit B.; Mahida, Anil K.; Jadav, Ghanshyam L.
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Bioactive oxadiazolo-benzodiazepines: synthesis, α amylase inhibition, antioxidant activity, molecular docking and DFT calculation
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deleteAit Lahcen, Marouane; El Karfi, Wissal; Ait Lahcen, Nouhaila; Fadili, Driss; Hmaimou, Samir; Adardour, Mohamed; Hdoufane, Ismail; Zaballos-Garcia, Elena; Faouzi, My El Abbes; Maatallah, Mohamed; Cherqaoui, Driss; Baouid, Abdesselam
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Targets for bacterial resistance: recent advances in small-molecule FtsZ inhibitors
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deleteShao, Wu-Bin; Zhou, Xiang; Yang, Song; Zhou, Ying
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Synthesis of acyl hydrazide derivatives of α-naphthalene acetic acid as COX-2 inhibitors: in vitro evaluation, molecular docking and DFT studies
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deleteBibi, Amrina; Alam, Aftab; Fareed, Ghulam; Ayaz, Muhammad; Shah, Tanzeela Ahmad; Naz, Sumaira; Qayum, Aamir; Ali Shah, Syed Adnan; Ali, Mumtaz; Ahmad, Manzoor
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Medicinal chemistry approaches for dual inhibition of amyloid-β and tau aggregation in Alzheimer's disease
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deleteJangra, Jatin; Mahindru, Isha; Kumar, Aman; Gupta, Harikesh Kumar; Ramesh, Vishwakarma Krishna; Kumar, Rajnish
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Wogonin-derived chemotype enables discovery of novel GLS1 inhibitors with potent antitumor activity
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deleteLi, Xuhong; Liang, Yan; Zhang, Xiaoyu; Wu, Yongsheng; Wu, Tizhi; Tian, Yucheng; Tang, Cheng; Qiu, Zhixia; Wu, Hongxi; Bian, Jinlei; Li, Zhiyu; Xu, Xi; Wang, Jubo
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A comprehensive review of indole hybrids as anti-bacterial and anti-fungal agents: synthetic protocols and SAR studies
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deleteBellapukonda, Sri Mounika; Anas, K. T. Muhammed; Mishra, Shivam; Kodi, Ramakrishna; Ghosh, Subhendu; Korra, Laxma Naik; Nanduri, Srinivas; Yaddanapudi, Venkata Madhavi
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Newly synthesized 2-cyclopentylidenehydrazinylthiazoles as potential therapeutic agents against peptic ulcer
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deleteSehrish; Salar, Uzma; Naz, Farzana; Ishaq, Aqsa; Naz, Fouzia; Iqbal, Jamshed; Khan, Khalid Mohammed
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Design, synthesis, in silico, and biological evaluation of novel pyrazolopyrimidinone-based estrogen receptor inhibitors
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deleteHesham, Sara A.; Shahin, Mai I.; Ziko, Laila; Serya, Rabah A. T.; Farag, Nahla A.; Abouzid, Khaled; Mowafy, Samar
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Design, synthesis, and biological evaluation of disubstituted thiazolidinedione derivatives as pancreatic lipase inhibitors for the management of obesity
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deleteKhan, Mhd Shabbu; Khator, Rakesh; Yadav, Nisha; Jagtap, Utkarsh A.; Paul, Atish T.; Monga, Vikramdeep
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Overview of recent strategic advances in antiviral covalent inhibitors
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deleteWang, Bo; Wang, Siyuan; Zhang, Jiwei; Kim, Meehyein; Zhan, Peng
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Synthesis of anticancer agents: molecular docking and ADME studies of new hydropyrimidine linked amide-pyridine derivatives
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deleteAarthi, Rajendran; Looi, Chin-King; Mai, Chun-Wai; Ramalingan, Chennan
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