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Medicinal Chemistry Research

IF3.1
Papers260
Citations6962
Journal Papers 237
Publication Date
Indole-based derivatives as anticancer agents: recent advances in structure–activity relationships and biological mechanisms
delete2026-08-14
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PREAI
deleteAashik Malik; Mayank Yadav; Jai Parkash Kadian; Komal Mishra; Ramsha; Anurag Rathore; Manisha; Nishant Rathour
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Characterization of beddomeilactone amide as bacterial DNA gyrase inhibitor: in vitro evaluation and computational insights
delete2026-07-28
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PREAI
deleteTashi Palmo; Vishwani Jamwal; Karan Goel; Anuj Kumar; Somdutt Mujwar; Yogesh P. Bharitkar; Kuljit Singh
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Isolation, modification, structure-activity relationship (SAR) and molecular docking studies of isoflavones from Derris scandens as potent dual AChE/BuChE inhibitors
delete2026-07-17
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PREAI
deleteYuttana Siriwattanasathien; Pathumwadee Yotmanee; Kanokporn Lehboon; Ratchanaporn Chokchaisiri; Kinnicha Nunparn; Warangkana Chunglok; Apichart Suksamrarn
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Design and synthesis of pyrrolo[2,3-d]pyrimidine linked diazospiro and piperazine – piperidine libraries as anticancer agents
delete2026-07-17
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PREAI
deleteSridhar Guda; Srilakshmi V Patri; Krishna Reddy V; Vishnu Thumma; Santosh Kumar Guru
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Investigation of reported small molecule P2Y6 receptor antagonists
delete2026-07-11
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deleteChianna Dane; André D.J. McKenzie; Andrew P. Montgomery; Jonathan Du; Eryn L. Werry; Michael Kassiou
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QSAR modeling and in vitro studies of the selective action of triphenylphosphonium salts as anticancer agents against the rhabdomyosarcoma cell line
delete2026-07-11
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PREAI
deleteDiana Hodyna; Vasyl Kovalishyn; Olena Trokhimenko; Serhii Soloviov; Oksana Bahrieieva; Maryna Kachaeva; Larysa Metelytsia
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Alisols A-C and their acetate derivatives: a review of natural occurrence, pharmacology, semisynthesis, pharmacokinetics, and metabolism
delete2026-07-09
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PREAI
deleteDuong Quang Huan; Huynh Thi Ngoc Ni; Huy Dinh Vu; Tran Thi Thanh Thuy; Nguyen Hoang Ngan; Vu Kim Thoa; Nguyen Thi Hue; Ninh The Son
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Discovery of pyrrolo[2,3-d]pyrimidine derivatives with inhibitory effect on liver cancer stem cell
delete2026-06-19
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PREAI
deleteXuecong Zhang; Xuechun Chen; Liwei Wang; Yiyuan Chang; Jiaxin Li; Jijian Yang; Dongxuan Ni; Ruihan Zhang; Rong Liu; Weilie Xiao
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C(sp2)-Thio- and amino-methylated indole derivatives: one-pot synthesis, evaluation of cytotoxic and anti-inflammatory activity
delete2026-06-04
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PREAI
deleteV. R. Akhmetova; D. V. Leont’ev; N. S. Akhmadiev; V. N. Perfilova; V. S. Sirotenko; E. A. Paramonov; I. I. Prokofiev; M. A. Sagalaev; V. R. Khairullina; D. V. Ishmetova; Yu. V. Vakhitova
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