Not logged inSARS-CoV-2 3CLpro mutations T21I and E166A confer differential resistance to simnotrelvir, bofutrelvir, and ensitrelvir
Chen, Lu; Su, Haixia; Shang, Weijuan; Nie, Tianqing; Kuang, Wenhua; Wang, Chenchen; Shao, Qiang; Zhang, Leike; Liu, Wen; Xu, Yechun; Zhang, Yumin
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SaveProbing Weak Halogen Bonding in Aqueous Solution
Herbst, Manuel A.; Wu, Leyun; Woordes, Yannik T.; Peintner, Stefan; Xin, Jian; Boeckler, Frank M.; Xu, Zhijian; Zhu, Weiliang; Navarro-Vazquez, Armando; Erdelyi, Mate
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SaveDevelopment of a Fluorescence Polarization Assay for p300/CBP and Its Application Using a Direct-to-Biology Approach
Liang, Jiayin; Li, Ziyi; Jin, Lu; Wang, Yanlin; Luo, Xiaolin; Li, Xinyuan; Zhong, Hui; Du, Daohai; Luo, Cheng; Xiong, Huan
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SaveP5CS-coupled proline metabolism manipulates metabolic dysfunction-associated steatotic liver disease
Lyu, Zan; Yu, Sike; Peng, Chang; Wu, Wenbiao; Yang, Wenhua; Ma, Huan; Sun, Yan; Jing, Liya; Gu, Hongyu; Tang, Erjiang; Zhang, Xuemei; Jiang, Huihong; Jiang, Haowen; Li, Jia
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SaveDiscovery of a Potent Fluorescence Polarization Probe for Identifying USP1 Allosteric Inhibitors
Cheng, Jiawei; Wang, Peipei; Wang, Pengfei; Wang, Jiamin; Li, Baiyang; Fang, Daqing; He, Jian; Hu, Xiaobei; Kan, Weijuan; Zhou, Yubo; Li, Chunpu; Li, Jia; Liu, Hong
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SaveCovalent versus Dimeric Optimization of Nectin-4-Targeted Peptide Radiotracers: A Head-to-Head Comparison in Triple-Negative Breast Cancer Mice Models
Pei, Yang; Zhou, Xu; Gao, Fei; Sun, Mingyue; Qiu, Shanshan; Qin, Xiangyu; Qu, Chunrong; Wen, Kai; Du, Jin; Hu, Ji; Cheng, Zhen
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SaveArtemverlotolides A and B, Two Sesquiterpenes from Artemisia verlotorum Lamotte: Structural Elucidation, Bioinspired Synthesis, and Antineuroinflammatory Activity
Xu, Mingbi; Wang, Mengyu; Zhu, Chiyun; Gong, Qi; Zhang, Ruiyu; Tang, Chunping; Zhang, Haiyan; Ye, Yang; Yao, Sheng
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SaveDevelopment and Validation of a Rapid LC-MS/MS Method for the Quantification of Contezolid in Human Plasma and Liver, and Its Application to a Pharmacokinetic Study in Liver Transplant Patients
Tian, Zhuoran; Zhong, Siyi; Wei, Huimin; Pan, Anni; Zhu, Hengkai; Zhu, Dan; Lu, Jianfang; Yu, Jinghua; Diao, Xingxing; Zhuang, Li
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SaveLate-Stage Cyclization of Natural Products and Drug Molecules Enabled by C-C Bond Cleavage of Aryl Ketones
Wang, Xing; Li, Yu-Xi; Zeng, Qing-Ying; Yu, Xin-Ming; Gao, Tian-Qi; Liu, Huan; Zhang, Ling-Xia; Xu, Hui; Wang, Zhen-Yu; Lan, Lefu; Dai, Hui-Xiong
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SaveNRZ complex facilitates virus infection via enhancing ER-LD contacts
Li, Zhifang; Xing, Yifan; Huang, Xinyi; Tian, Buyun; Mei, Jie; Fu, Xinyue; Huang, Yuhan; Zhang, Qian; Ding, Binbin; Cao, Xiaobao; Xue, Yanhong; Li, Zonghong; Xu, Tao; Jiu, Yaming
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SaveIntegrated proteomic and phosphoproteomic profiling unravels an O-GlcNAc-dependent mechanism in DGAT1 inhibition-mediated protection of β-cells from lipotoxicity
Guo, Jia-Ming; Chen, Guang-Yun; Huang, Jun-Shang; Zhu, Zhen-Yun; Dong, Lin-Yue; Xie, Wen-Fan; Li, Yi-Ming; Hu, You-Hong; Wang, He-Yao; Zhou, Hu
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SaveCascade-Amplified Ratiometric Fluorescent Probe for Time-Locked Imaging Epilepsy
Wang, Xin; Li, Bohan; Li, Min; Chen, Yuncan; Tang, Yurui; Ji, Aiyan; Zhao, Jing; Sun, Chenchen; Li, Zhenrong; Ni, Dan; Cheng, Yanlong; Sun, Wanbing; Lei, Zuhai; Wang, Jing; Vezzani, Annamaria; Li, Xiaoyu; Li, Cong; Zhu, Xiao; Cheng, Zhen; Wang, Cong
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SaveNew Macrocyclolipopeptides and Steroids from Mariana Trench-Derived Fungus Cladosporium sp.
Peng, Qingyun; Lan, Shanshan; Li, Qun; Liu, Yunan; Ruan, Wu; Wu, Kun; Shen, Qianqian; Chen, Yi; Wang, Junfeng; Li, Dan; Wang, Ming-Wei
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SaveDesign, Synthesis, and Structure-Activity Relationship Studies of 7H-Pyrrolo[2,3-d]pyrimidine Derivatives as Potent Casein Kinase 1α (CK1α) Inhibitors
Liu, Meiying; Tu, Yutong; Xu, Wangyang; Gao, Lixin; Wang, Kun; Zhou, Yang; Xu, Tianfeng; Zhou, Yubo; Zhou, Chuan
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SaveBrain-Targeting Metal-Organic Framework Nanoplatform Reprogramming Ferroptosis Sensitivity of Glioblastoma
Wang, Mengzhen; Lai, Yi; Meng, Hanxue; Jin, Aojia; Zhang, Ping; Shen, Yinuo; Lin, Shutong; Yu, Haijun; Xu, Wujun; Lehto, Vesa-Pekka; Zhang, Wen; Xu, Zhiai
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