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SaveStructure and mechanism of a phage-encoded SAM lyase revises catalytic function of enzyme family
Guo, Xiaohu; Soderholm, Annika; Kanchugal, Sandesh P.; Isaksen, Geir, V; Warsi, Omar; Eckhard, Ulrich; Triguis, Silvia; Gogoll, Adolf; Jerlstrom-Hultqvist, Jon; Aqvist, Johan; Andersson, Dan, I; Selmer, Maria
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Save3,4-Dihydropyrimidin-2(1H)-ones as Antagonists of the Human A2B Adenosine Receptor: Optimization, Structure-Activity Relationship Studies, and Enantiospecific Recognition
Majellaro, Maria; Jespers, Willem; Crespo, Abel; Nunez, Maria J.; Novio, Silvia; Azuaje, Jhonny; Prieto-Diaz, Ruben; Gioe, Claudia; Alispahic, Belma; Brea, Jose; Loza, Maria, I; Freire-Garabal, Manuel; Garcia-Santiago, Carlota; Rodriguez-Garcia, Carlos; Garcia-Mera, Xerardo; Caamano, Olga; Fernandez-Masaguer, Christian; Sardina, Javier F.; Stefanachi, Angela; El Maatougui, Abdelaziz; Mallo-Abreu, Ana; Aqvist, Johan; Gutierrez-de-Teran, Hugo; Sotelo, Eddy
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SaveDissecting the Mechanism of (R)-3-Hydroxybutyrate Dehydrogenase by Kinetic Isotope Effects, Protein Crystallography, and Computational Chemistry
Machado, Teresa F. G.; Purg, Miha; McMahon, Stephen A.; Read, Benjamin J.; Oehler, Verena; Aqvist, Johan; Gloster, Tracey M.; da Silva, Rafael G.
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SaveX-Ray Crystallography and Free Energy Calculations Reveal the Binding Mechanism of A2A Adenosine Receptor Antagonists
Jespers, Willem; Verdon, Gregory; Azuaje, Jhonny; Majellaro, Maria; Keranen, Henrik; Garcia-Mera, Xerardo; Congreve, Miles; Deflorian, Francesca; de Graaf, Chris; Zhukov, Andrei; Dore, Andrew S.; Mason, Jonathan S.; Aqvist, Johan; Cooke, Robert M.; Sotelo, Eddy; Gutierrez-de-Teran, Hugo
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