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Christian P. R. Hackenberger

Leibniz Forschungsinstitut für Molekulare Pharmakologie

44H-index
279Paper Count
7.1KCitation Count
Published Papers 96
Publication Date
A cell-permeable nanobody to restore F508del cystic fibrosis transmembrane conductance regulator activity
err2026-04-17
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errLuise Franz; Tihomir Rubil; Anita Balázs; Marie Overtus; Kristin Kemnitz-Hassanin; Cedric Govaerts; Marcus A. Mall; Christian P. R. Hackenberger
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Polyfluoroalkyl-Tagged Cell-Penetrating Peptide-Additives Enhance Intracellular Protein Delivery via Sustained Monomeric Lipid Interaction
err2026-04-14
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errSarah Hansen; Hana Zupan; Ferhat Mutlu; Jan Vincent V. Arafiles; Rubén Cruz; Palina Dubatouka; Kenichi Ataka; Martin Lehmann; Bettina G. Keller; Joachim Heberle; Christian P. R. Hackenberger
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Modular Vinyl Phosphonamidates for Cysteine-Directed Protein Targeting
err2026-02-10
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errChristian E. Stieger; Charlotte Völkel; Mathias B. Bertelsen; Michael Lisurek; Jan Vincent V. Arafiles; Jonathan Franke; Leander Crocker; Karl Schuppe; Yunjae Lim; Christiane Groneberg; Mathias Christmann; Han Sun; Christian P. R. Hackenberger
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Unsaturated Phosphorus Electrophiles to Probe Protein Tyrosine Phosphatases
err2026-02-03
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errEleftheria Poulou; Max Ruwolt; Christian E. Stieger; Kristin Kemnitz-Hassanin; Christian P. R. Hackenberger
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Targeting the Membrane-Embedded Rhomboid Protease GlpG: A Multimodal Strategy for Inhibitor Discovery and Mechanistic Insight
err2026-01-28
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errClaudia Bohg; Yurii Dubanych; Spyridon Kosteletos; Taoran Xiao; Martin Neuenschwander; Tillmann Utesch; Michael Lisurek; Carl Öster; Andreas Oder; Carola Seyffarth; Kathrin Bach; Denise-Liù Gracias Leone; František Filandr; Marc Wegert; Sascha Lange; Henry Sawczyc; Jens Peter von Kries; Christian P. R. Hackenberger; Edgar Specker; Han Sun; Kvido Stříšovský; Adam Lange
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Expanding the payload scope in antibody-drug conjugates by delivery of hydroxy-containing drugs through self-immolative phosphoramidates
err2026-01-20
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errPhilipp Ochtrop; Anil P. Jagtap; Jan G. Felber; Simon Vogt; Sarah Herterich; Isabelle Mai; Philipp Cyprys; Saskia Schmitt; Sarah Payer; Annabel Kitowski; Swetlana Wunder; Paul Machui; Julia Brandmeier; Natascia Leonardi; Elizaveta Poliak; Christian P. R. Hackenberger; Olivier Marcq; Dominik Schumacher; Jonas Helma; Annette M. Vogl; Marc-André Kasper
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Quantitative analysis of inhibitor-induced assembly disruption in human UDP-GlcNAc 2-epimerase using mass photometry
err2025-10-16
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errNico Boback; Jacob Gorenflos López; Christian P. R. Hackenberger; Santiago Di Lella; Daniel C. Lauster
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Energy-transfer photoproximity labelling in live cells using an organic cofactor
err2025-09-17
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errLeander B. Crocker; Jan Vincent V. Arafiles; Judith M. Müchler; Max Ruwolt; Kristin Kemnitz-Hassanin; Kilian Roßmann; Christian E. Stieger; Fan Liu; Nataliya Archipowa; Roger Jan Kutta; Christian P. R. Hackenberger
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Intracellular Delivery of Native Proteins by BioReversible Arginine Modification (BioRAM) on Amino Groups
err2025-07-09
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errJonathan Franke; Jan Vincent V. Arafiles; Christian Leis; Christian P. R. Hackenberger
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Unsaturated Phosphine Oxides for Modular Antibody Rebridging and Single Reagent Peptide-Cyclisation-Bioconjugation
err2025-06-30
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PREAI
errDr. Christian E. Stieger; Dr. Alastair J. McMillan; Dr. Mark A. R. de Geus; Dr. Jan Vincent V. Arafiles; Dr. Luise Franz; Prof. Dr. Christian P. R. Hackenberger
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Fluorogenic cell surface glycan labelling with fluorescence molecular rotor dyes and nucleic acid stains
err2024-01-01
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errKocak, Alen; Homer, Amal K.; Feida, Antonia; Telschow, Florian; Gorenflos Lopez, Jacob L.; Baydaroglu, Cihan; Gradzielski, Michael; Hackenberger, Christian P. R.; Alexiev, Ulrike; Seitz, Oliver
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Rapid building block-economic synthesis of long, multi-O-GalNAcylated MUC5AC tandem repeat peptides
err2024-01-01
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errGalashov, Arseniy; Kazakova, Ekaterina; Stieger, Christian E.; Hackenberger, Christian P. R.; Seitz, Oliver
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Cell-Surface-Retained Peptide Additives for the Cytosolic Delivery of Functional Proteins
err2023-10-31
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errArafiles, Jan Vincent V.; Franke, Jonathan; Franz, Luise; Gomez-Gonzalez, Jacobo; Kemnitz-Hassanin, Kristin; Hackenberger, Christian P. R.
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Design and Evaluation of Phosphonamidate-Linked Exatecan Constructs for Highly Loaded, Stable, and Efficacious Antibody-Drug Conjugates
err2023-10-12
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errSchmitt, Saskia; Machui, Paul; Mai, Isabelle; Herterich, Sarah; Wunder, Swetlana; Cyprys, Philipp; Gerlach, Marcus; Ochtrop, Philipp; Hackenberger, Christian P. R.; Schumacher, Dominik; Helma, Jonas; Vogl, Annette M.; Kasper, Marc-Andre
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(3+2)-Cyclization Reactions of Unsaturated Phosphonites with Aldehydes and Thioketones
err2023-04-27
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errMunasinghe, Don S.; Kasper, Marc-Andre; Jasinski, Radomir; Kula, Karolina; Palusiak, Marcin; Celeda, Malgorzata; Mloston, Grzegorz; Hackenberger, Christian P. R.
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Real-time monitoring of the sialic acid biosynthesis pathway by NMR
err2023-01-01
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errLopez, Jacob Gorenflos L.; Schmieder, Peter; Kemnitz-Hassanin, Kristin; Asikoglu, Hatice Ceyda; Celik, Arif; Stieger, Christian E.; Fiedler, Dorothea; Hinderlich, Stephan; Hackenberger, Christian P. R.
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Compact hydrophilic electrophiles enable highly efficacious high DAR ADCs with excellent in vivo PK profile
err2023-01-01
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errOchtrop, Philipp; Jahzerah, Jahaziel; Machui, Paul; Mai, Isabelle; Schumacher, Dominik; Helma, Jonas; Kasper, Marc-Andre; Hackenberger, Christian P. R.
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DFT-Guided Discovery of Ethynyl-Triazolyl-Phosphinates as Modular Electrophiles for Chemoselective Cysteine Bioconjugation and Profiling
err2022-08-22
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errStieger, Christian E.; Park, Yerin; de Geus, Mark A. R.; Kim, Dongju; Huhn, Christiane; Slenczka, J. Sophia; Ochtrop, Philipp; Muechler, Judith M.; Suessmuth, Roderich D.; Broichhagen, Johannes; Baik, Mu-Hyun; Hackenberger, Christian P. R.
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