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Shao Q. Yao

National University of Singapore

70H-index
359Paper Count
1.6WCitation Count
Published Papers 195
Publication Date
Intracellular Delivery of Antibody-Based Therapeutics for Targeted Oncogenic c-Myc Degradation in Mammalian Cells and Mice
err2026-08-28
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PREAI
errLvyang Peng; Jiaoyu Chen; Xia Liu; Jiachang Yan; Yingying Gan; Chen Fang; Jingyan Ge; Shao Q. Yao; Peiyan Yuan
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Sulfonated azobenzene-derived nanogels: Hypoxia-specific degradation enables superior nucleic acid-mediated tumor therapy
err2026-04-10
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PREAI
errJia Zhou; Shubo Du; Lan Wang; Qiong Wu; Changmin Yu; Wei Du; Lin Li; Shao Q. Yao
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Large-Scale Profiling of Kinase Degradation by Using Norbornene-Based Hydrophobic Tag (HyT) Strategy
err2026-04-01
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PREAI
errGu, Mingxi; Miao, Fengfei; Peng, Lvyang; Sun, Jie; Chen, Peng; Yang, Fang; Yan, Jiachang; Gao, Liqian; Lu, Xiaoyun; Yao, Shao Q.; Yuan, Peiyan
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PROTAC-based degradation of catechol-O-methyltransferase for potential treatment of Parkinson’s disease
err2026-01-04
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PREAI
errHaixiao Fang; Panpan Li; Qi Gao; Shubo Du; Jing Gu; Xia Liu; Bo Peng; Hua Bai; Cheng-Wu Zhang; Lin Li; Shao Q. Yao
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Cell-Active, Irreversible Covalent Inhibitors Targeting a Surface-Exposed Non-Catalytic Lysine on Aurora a Kinase by Using Squarate Chemistry
err2025-08-28
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PREAI
errZuqin Wang; Xuan Wang; Yong Li; Peishan Li; Shengjie Huang; Peng Chen; Guanghui Tang; Xiaotong Ding; Prof. Dr. Zhang Zhang; Prof. Dr. Zhi-Min Zhang; Prof. Dr. Yang Zhou; Prof. Dr. Shao Q. Yao; Prof. Dr. Xiaoyun Lu
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Tumor microenvironment-responsive self-assembled nanomedicine for reversible covalent targeting of BCR-ABL kinase
err2025-06-07
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PREAI
errMenghua Xiang; Fen Yang; Peng Chen; Jiaoyu Chen; Jianzhong Zhang; Jiayi Yang; Yilin Liu; Qianqian Zhang; Jiang Pi; Peiyan Yuan; Shao Q Yao; Liqian Gao
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Chemical Probe-Enabled Lipid Droplet Proteomics
err2025-03-11
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PREAI
errXiang, Jing; Li, Tao; Zhang, Junzhe; Wu, Wenxian; Xu, Guangyu; Yan, Jiaqian; Wang, Hao; Chen, Suyuan; Yao, Shao Q.; Yi, Fan
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Rationally designed BCR-ABL kinase inhibitors for improved leukemia treatment via covalent and pro-/dual-drug targeting strategies
err2024-09-08
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errOAAI
errJie Sun; Liang Lou; Chengjun Zhu; Peng Chen; Guanghui Tang; Mingxi Gu; Shu Xia; Xiao Dong; Zhi-Min Zhang; Liqian Gao; Shao Q. Yao; Qicai Xiao
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Small Molecule-Induced Post-Translational Acetylation of Catalytic Lysine of Kinases in Mammalian Cells
err2024-08-20
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PREAI
errTang, Guanghui; Wang, Xuan; Huang, Huisi; Xu, Manyi; Ma, Xingyu; Miao, Fengfei; Lu, Xiaoyun; Zhang, Chong-Jing; Gao, Liqian; Zhang, Zhi-Min; Yao, Shao Q.
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Reactivity-Tunable Fluorescent Platform for Selective and Biocompatible Modification of Cysteine or Lysine
err2024-06-19
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errOAAI
errRen, Xiaojie; Li, Haokun; Peng, Hui; Yang, Yang; Su, Hang; Huang, Chen; Wang, Xuan; Zhang, Jie; Liu, Zhiyang; Wei, Wenyu; Cheng, Ke; Zhu, Tianyang; Lu, Zhenpin; Li, Zhengqiu; Zhao, Qian; Tang, Ben Zhong; Yao, Shao Q.; Song, Xiangzhi; Sun, Hongyan
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Kinase Inhibition via Small Molecule-Induced Intramolecular Protein Cross-Linking
err2024-06-07
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PREAI
errWang, Xuan; Sun, Jie; Huang, Huisi; Tang, Guanghui; Chen, Peng; Xiang, Menghua; Li, Lin; Zhang, Zhi-Min; Gao, Liqian; Yao, Shao Q.
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Prodrug-conjugated tumor-seeking commensals for targeted cancer therapy
err2024-05-21
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errOAAI
errShen, Haosheng; Zhang, Changyu; Li, Shengjie; Liang, Yuanmei; Lee, Li Ting; Aggarwal, Nikhil; Wun, Kwok Soon; Liu, Jing; Nadarajan, Saravanan Prabhu; Weng, Cheng; Ling, Hua; Tay, Joshua K.; Wang, De Yun; Yao, Shao Q.; Hwang, In Young; Lee, Yung Seng; Chang, Matthew Wook
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Targeted Degradation of Cell-Surface Proteins via Chaperone-Mediated Autophagy by Using Peptide-Conjugated Antibodies
err2024-03-27
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PREAI
errShao, Jinning; Lin, Xuefen; Wang, Haoting; Zhao, Chuhan; Yao, Shao Q.; Ge, Jingyan; Zeng, Su; Qian, Linghui
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Global Reactivity Profiling of the Catalytic Lysine in Human Kinome for Covalent Inhibitor Development
err2024-02-14
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PREAI
errTang, Guanghui; Wang, Wei; Zhu, Chengjun; Huang, Huisi; Chen, Peng; Wang, Xuan; Xu, Manyi; Sun, Jie; Zhang, Chong-Jing; Xiao, Qicai; Gao, Liqian; Zhang, Zhi-Min; Yao, Shao Q.
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Cell-active, irreversible covalent inhibitors that selectively target the catalytic lysine of EGFR by using fluorosulfate-based SuFEx chemistry
err2023-11-01
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PREAI
errTang, Guanghui; Wang, Wei; Wang, Xuan; Ding, Ke; Ngan, SoFong Cam; Chen, Jiao-Yu; Sze, Siu Kwan; Gao, Liqian; Yuan, Peiyan; Lu, Xiaoyun; Yao, Shao Q.
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Insulin-like Growth Factor 2 (IGF2)-Fused Lysosomal Targeting Chimeras for Degradation of Extracellular and Membrane Proteins
err2023-10-30
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PREAI
errZhang, Bei; Brahma, Rajeev Kungur; Zhu, Liquan; Feng, Jiayi; Hu, Shiqi; Qian, Linghui; Du, Shubo; Yao, Shao Q.; Ge, Jingyan
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Tumor Metabolism-Rewriting Nanomedicines for Cancer Immunotherapy
err2023-09-22
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errOAAI
errDong, Xiao; Xia, Shu; Du, Shubo; Zhu, Mao-Hua; Lai, Xing; Yao, Shao Q.; Chen, Hong-Zhuan; Fang, Chao
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Orthogonal Strategies for Profiling Potential Cellular Targets of Anandamide and Cannabidiol
err2023-06-30
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PREAI
errTang, Guanghui; Lim, Ying-Jie; Wang, Wei; Ye, Zi; Zhang, Chong-Jing; Yao, Shao Q.
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