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Developing novel Lin28 inhibitors by computer aided drug design Matias-Barrios, Victor M.; Radaeva, Mariia; Rosellinny, Graciella; Jia, Qiongqiong; Xie, Ning; Villanueva, Monica; Ibrahim, Hanadi; Smith, Jason; Gleave, Martin; Lallous, Nada; Straus, Suzana K.; Cherkasov, Artem; Dong, Xuesen Share Save
Characterization of novel small molecule inhibitors of estrogen receptor-activation function 2 (ER-AF2) Foo, Jane; Gentile, Francesco; Massah, Shabnam; Morin, Helene; Singh, Kriti; Lee, Joseph; Smith, Jason; Ban, Fuqiang; Leblanc, Eric; Young, Robert; Strynadka, Natalie; Lallous, Nada; Cherkasov, Artem Share Save
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Characterization of ER-AF2 inhibitors in breast cancer Foo, Jane; Gentile, Francesco; Lee, Joseph; Morin, Helene; Massah, Shabnam; Guo, Maria; Smith, Jason; Ban, Fuqiang; Cherkasov, Artem; Lallous, Nada Share Save
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Dynamic phase separation of the androgen receptor and its coactivators key to regulate gene expression Zhang, Fan; Biswas, Maitree; Massah, Shabnam; Lee, Joseph; Lingadahalli, Shreyas; Wong, Samantha; Wells, Christopher; Foo, Jane; Khan, Nabeel; Morin, Helene; Saxena, Neetu; Kung, Sonia H. Y.; Sun, Bei; Nunez, Ana Karla Parra; Sanchez, Christophe; Chan, Novia; Ung, Lauren; Altintas, Umut Berkay; Bui, Jennifer M.; Wang, Yuzhuo; Fazli, Ladan; Oo, Htoo Zarni; Rennie, Paul S.; Lack, Nathan A.; Cherkasov, Artem; Gleave, Martin E.; Gsponer, Jorg; Lallous, Nada Share Save
Structure-Based Study to Overcome Cross-Reactivity of Novel Androgen Receptor Inhibitors Radaeva, Mariia; Li, Huifang; LeBlanc, Eric; Dalal, Kush; Ban, Fuqiang; Ciesielski, Fabrice; Chow, Bonny; Morin, Helene; Awrey, Shannon; Singh, Kriti; Rennie, Paul S.; Lallous, Nada; Cherkasov, Artem Share Save
Reformation of the chondroitin sulfate glycocalyx enables progression of AR-independent prostate cancer Al-Nakouzi, Nader; Wang, Chris Kedong; Oo, Htoo Zarni; Nelepcu, Irina; Lallous, Nada; Spliid, Charlotte B.; Khazamipour, Nastaran; Lo, Joey; Truong, Sarah; Collins, Colin; Hui, Desmond; Esfandnia, Shaghayegh; Adomat, Hans; Clausen, Thomas Mandel; Gustavsson, Tobias; Choudhary, Swati; Dagil, Robert; Corey, Eva; Wang, Yuzhuo; Chauchereau, Anne; Fazli, Ladan; Esko, Jeffrey D.; Salanti, Ali; Nelson, Peter S.; Gleave, Martin E.; Daugaard, Mads Share Save
Development of 2-(5,6,7-Trifluoro-1H-Indol-3-yl)-quinoline-5-carboxamide as a Potent, Selective, and Orally Available Inhibitor of Human Androgen Receptor Targeting Its Binding Function-3 for the Treatment of Castration-Resistant Prostate Cancer Leblanc, Eric; Ban, Fuqiang; Cavga, Ayse Derya; Lawn, Sam; Huang, Chia-Chi Flora; Mohan, Sankar; Chang, Matthew E. K.; Flory, Mark R.; Ghaidi, Fariba; Lingadahalli, Shreyas; Chen, Gang; Yu, Ivan Pak Lok; Morin, Helene; Lallous, Nada; Gleave, Martin E.; Mohammed, Hisham; Young, Robert N.; Rennie, Paul S.; Lack, Nathan A.; Cherkasov, Artem Share Save
Discovery of New Catalytic Topoisomerase II Inhibitors for Anticancer Therapeutics Matias-Barrios, Victor M.; Radaeva, Mariia; Song, Yi; Alperstein, Zaccary; Lee, Ahn R.; Schmitt, Veronika; Lee, Joseph; Ban, Fuqiang; Xie, Ning; Qi, Jianfei; Lallous, Nada; Gleave, Martin E.; Cherkasov, Artem; Dong, Xuesen Share Save
Androgen receptor-binding sites are highly mutated in prostate cancer Morova, Tunc; McNeill, Daniel R.; Lallous, Nada; Gonen, Mehmet; Dalal, Kush; Wilson, David M., III; Guersoy, Attila; Keskin, Ozlem; Lack, Nathan A. Share Save
Ivermectin inhibits HSP27 and potentiates efficacy of oncogene targeting in tumor models Nappi, Lucia; Aguda, Adeleke H.; Al Nakouzi, Nader; Lelj-Garolla, Barbara; Beraldi, Eliana; Lallous, Nada; Thi, Marisa; Moore, Susan; Fazli, Ladan; Battsogt, Dulguun; Stief, Sophie; Ban, Fuqiang; Nguyen, Nham T.; Saxena, Neetu; Dueva, Evgenia; Zhang, Fan; Yamazaki, Takeshi; Zoubeidi, Amina; Cherkasov, Artem; Brayer, Gary D.; Gleave, Martin Share Save
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