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Artem Cherkasov

university of british columbia

56H-index
348Paper Count
1.5WCitation Count
Published Papers 137
Publication Date
The Use of DeepQSAR Models for the Discovery of Peptides With Enhanced Antimicrobial and Antibiofilm Potential
err2026-04-16
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errOAAI
errJiaying You; Hazem Mslati; Evan F. Haney; Noushin Akhoundsadegh; Robert E. W. Hancock; Artem Cherkasov
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CACHE Challenge #3: Targeting the Nsp3 Macrodomain of SARS-CoV-2
err2026-01-21
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errOAAI
errOleksandra Herasymenko; Madhushika Silva; Galen J. Correy; Abd Al-Aziz A. Abu-Saleh; Suzanne Ackloo; Cheryl Arrowsmith; Alan Ashworth; Fuqiang Ban; Hartmut Beck; Kevin P. Bishop; Hugo J. Bohórquez; Albina Bolotokova; Marko Breznik; Irene Chau; Yu Chen; Artem Cherkasov; Wim Dehaen; Dennis Della Corte; Katrin Denzinger; Niklas P. Doering; Kristina Edfeldt; Aled Edwards; Darren Fayne; Francesco Gentile; Elisa Gibson; Ozan Gokdemir; Anders Gunnarsson; Judith Günther; John J. Irwin; Jan Halborg Jensen; Rachel J. Harding; Alexander Hillisch; Laurent Hoffer; Anders Hogner; Ashley Hutchinson; Shubhangi Kandwal; Andrea Karlova; Kushal Koirala; Sergei Kotelnikov; Dima Kozakov; Juyong Lee; Soowon Lee; Uta Lessel; Sijie Liu; Xuefeng Liu; Peter Loppnau; Jens Meiler; Rocco Moretti; Yurii S. Moroz; Charuvaka Muvva; Tudor I. Oprea; Brooks Paige; Amit Pandit; Keunwan Park; Gennady Poda; Mykola V. Protopopov; Vera Pütter; Rahul Ravichandran; Didier Rognan; Edina Rosta; Yogesh Sabnis; Thomas Scott; Almagul Seitova; Purshotam Sharma; François Sindt; Minghu Song; Casper Steinmann; Rick Stevens; Valerij Talagayev; Valentyna V. Tararina; Olga Tarkhanova; Damon Tingey; John F. Trant; Dakota Treleaven; Alexander Tropsha; Patrick Walters; Jude Wells; Yvonne Westermaier; Gerhard Wolber; Lars Wortmann; Shuangjia Zheng; James S. Fraser; Matthieu Schapira
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Design of Highly Potent Antibiofilm, Antimicrobial Peptides Using Explainable Artificial Intelligence
err2025-12-01
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PREAI
errPikalyova, Karina; Akhmetshin, Tagir; Orlov, Alexey; Haney, Evan F.; Akhoundsadegh, Noushin; You, Jiaying; Hancock, Robert E. W.; Horvath, Dragos; Marcou, Gilles Gerard; Cherkasov, Artem; Varnek, Alexandre
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A scalable reinforcement learning approach for screening large peptide libraries for bioactive peptide discovery
err2025-11-27
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errOAAI
errMohit Pandey; Jane Foo; Shabnam Massah; Morgan A. Alford; Hazem Mslati; Gopeshh Subbaraj; Mira Saba; Francesco Gentile; Nada Lallous; Evan F. Haney; Robert E. W. Hancock; Martin Ester; Artem Cherkasov
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Discovery and development of novel CNS-penetrating PARP1-selective inhibitors
err2025-11-01
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errOAAI
errBacha, Jeffrey; Truong, Sarah; Ban, Fuqiang; Smith, Jason; Pandey, Mohit; Manskaia, Ekaterina; Zhai, Beibei; Ramos, Louise; Marzban, Mona; Ghaidi, Fariba; Adomat, Hans; Singh, Kally; Chen, Xiaoqi; Brown, Dennis; Langlands, John; Collins, Colin; Cherkasov, Artem; Daugaard, Mads
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The Use of DeepQSAR Models for the Discovery of Peptides with Enhanced Antimicrobial and Antibiofilm Potential
err2025-11-01
err0
PREAI
errYou, Jiaying; Mslati, Hazem; Haney, Evan F.; Akhoundsadegh, Noushin; Hancock, Robert E. W.; Cherkasov, Artem
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Functional and Structural Characterization of Treatment-Emergent Nirmatrelvir Resistance Mutations at Low Frequencies in the Main Protease (Mpro) Reveals a Unique Evolutionary Route for SARS-CoV-2 to Gain Resistance
err2025-06-01
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errOAAI
errDeschenes, Natalie M.; Perez-Vargas, Jimena; Zhong, Zoe; Thomas, Merrilee; Kenward, Calem; Mosimann, Wesley A.; Worrall, Liam J.; Waglechner, Nicholas; Li, Angel XinLiu; Maguire, Finlay; Aftanas, Patryk; Smith, Jason R.; Lim, Jared; Young, Robert N.; Cherkasov, Artem; Farooqi, Lubna; Moinuddin, Adnan; Siddiqi, Lina; Malik, Imaan; Lefebvre, Maxime; Paetzel, Mark; Strynadka, Natalie C. J.; Jean, Francois; McGeer, Allison; Kozak, Robert A.
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The Six Ds of Exponentials and drug discovery: A path toward reversing Eroom's law
err2025-04-01
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PREAI
errTropsha, Alexander; Martin, Holli-Joi; Cherkasov, Artem
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Developing novel Lin28 inhibitors by computer aided drug design
err2025-01-12
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errOAAI
errMatias-Barrios, Victor M.; Radaeva, Mariia; Rosellinny, Graciella; Jia, Qiongqiong; Xie, Ning; Villanueva, Monica; Ibrahim, Hanadi; Smith, Jason; Gleave, Martin; Lallous, Nada; Straus, Suzana K.; Cherkasov, Artem; Dong, Xuesen
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Blood matters: the hematological signatures of Coronavirus infection
err2024-11-28
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errOAAI
errToro, Ayelen; Arevalo, Ana P.; Pereira-Gomez, Marianoel; Sabater, Agustina; Zizzi, Eric A.; Perbolianachis, Paula; Pascual, Gaston; Lage-Vickers, Sofia; Porfido, Jorge L.; Achinelli, Ines; Seniuk, Rocio; Bizzotto, Juan; Sanchis, Pablo; Olivera, Alvaro; Leyva, Alejandro; Moreno, Pilar; Costabile, Alicia; Fajardo, Alvaro; Carrion, Federico; Flo, Martin; Olivero-Deibe, Natalia; Rodriguez, Fernando; Nin, Nicolas; Anselmino, Nicolas; Labanca, Estefania; Vazquez, Elba; Cotignola, Javier; Alonso, Daniel F.; Valacco, Maria P.; Marti, Marcelo; Gentile, Francesco; Cherkasov, Artem; Crispo, Martina; Moratorio, Gonzalo; Gueron, Geraldine
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Characterization of novel small molecule inhibitors of estrogen receptor-activation function 2 (ER-AF2)
err2024-11-26
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errOAAI
errFoo, Jane; Gentile, Francesco; Massah, Shabnam; Morin, Helene; Singh, Kriti; Lee, Joseph; Smith, Jason; Ban, Fuqiang; Leblanc, Eric; Young, Robert; Strynadka, Natalie; Lallous, Nada; Cherkasov, Artem
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UTILIZING DEEP DOCKING AND ARTIFICIAL INTELLIGENCE FOR THE DISCOVERY OF NOVEL PARP1-SELECTIVE INHIBITORS FOR USE AGAINST BRAIN TUMORS
err2024-11-11
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PREAI
errTruong, Sarah; Ban, Fuqiang; Smith, Jason; Zhai, Beibei; Ramos, Louise; Marzban, Mona; Ghaidi, Fariba; Adomat, Hans; Chen, Xiaoqi; Langlands, John; Brown, Dennis; Bacha, Jeffrey; Collins, Colin; Cherkasov, Artem; Daugaard, Mads
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CACHE Challenge #1: Targeting the WDR Domain of LRRK2, A Parkinson's Disease Associated Protein
err2024-11-05
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errOAAI
errLi, Fengling; Ackloo, Suzanne; Arrowsmith, Cheryl H.; Ban, Fuqiang; Barden, Christopher J.; Beck, Hartmut; Beranek, Jan; Berenger, Francois; Bolotokova, Albina; Bret, Guillaume; Breznik, Marko; Carosati, Emanuele; Chau, Irene; Chen, Yu; Cherkasov, Artem; Della Corte, Dennis; Denzinger, Katrin; Dong, Aiping; Draga, Sorin; Dunn, Ian; Edfeldt, Kristina; Edwards, Aled; Eguida, Merveille; Eisenhuth, Paul; Friedrich, Lukas; Fuerll, Alexander; Gardiner, Spencer S.; Gentile, Francesco; Ghiabi, Pegah; Gibson, Elisa; Glavatskikh, Marta; Gorgulla, Christoph; Guenther, Judith; Gunnarsson, Anders; Gusev, Filipp; Gutkin, Evgeny; Halabelian, Levon; Harding, Rachel J.; Hillisch, Alexander; Hoffer, Laurent; Hogner, Anders; Houliston, Scott; Irwin, John J.; Isayev, Olexandr; Ivanova, Aleksandra; Jacquemard, Celien; Jarrett, Austin J.; Jensen, Jan H.; Kireev, Dmitri; Kleber, Julian; Koby, S. Benjamin; Koes, David; Kumar, Ashutosh; Kurnikova, Maria G.; Kutlushina, Alina; Lessel, Uta; Liessmann, Fabian; Liu, Sijie; Lu, Wei; Meiler, Jens; Mettu, Akhila; Minibaeva, Guzel; Moretti, Rocco; Morris, Connor J.; Narangoda, Chamali; Noonan, Theresa; Obendorf, Leon; Pach, Szymon; Pandit, Amit; Perveen, Sumera; Poda, Gennady; Polishchuk, Pavel; Puls, Kristina; Puetter, Vera; Rognan, Didier; Roskams-Edris, Dylan; Schindler, Christina; Sindt, Francois; Spiwok, Vojtech; Steinmann, Casper; Stevens, Rick L.; Talagayev, Valerij; Tingey, Damon; Vu, Oanh; Walters, W. Patrick; Wang, Xiaowen; Wang, Zhenyu; Wolber, Gerhard; Wolf, Clemens Alexander; Wortmann, Lars; Zeng, Hong; Zepeda, Carlos A.; Zhang, Kam Y. J.; Zhang, Jixian; Zheng, Shuangjia; Schapira, Matthieu
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Pharmacokinetics Profiler (PhaKinPro): Model Development, Validation, and Implementation as a Web Tool for Triaging Compounds with Undesired Pharmacokinetics Profiles
err2024-04-03
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PREAI
errRath, Marielle; Wellnitz, James; Martin, Holli-Joi; Melo-Filho, Cleber; Hochuli, Joshua E.; Silva, Guilherme Martins; Beasley, Jon-Michael; Travis, Maxfield; Sessions, Zoe L.; Popov, Konstantin I.; Zakharov, Alexey V.; Cherkasov, Artem; Alves, Vinicius; Muratov, Eugene N.; Tropsha, Alexander
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Clinically-observed FOXA1 mutations upregulate SEMA3C through transcriptional derepression in prostate cancer
err2024-03-25
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errOAAI
errTam, Kevin J.; Liu, Liangliang; Hsing, Michael; Dalal, Kush; Thaper, Daksh; McConeghy, Brian; Yenki, Parvin; Bhasin, Satyam; Peacock, James W.; Wang, Yuzhuo; Cherkasov, Artem; Rennie, Paul S.; Gleave, Martin E.; Ong, Christopher J.
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Targeting the translation initiation complex component eIF4G1 in melanoma
err2024-03-22
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PREAI
errFeng, Yongmei; Radaeva, Mariia; Kim, Hyungsoo; Deshpande, Anagha; Deshpande, Ani; Jovanovic, Predrag; Murad, Rabi; Topisirovic, Ivan; Olson, Steven; Cherkasov, Artem; Ronai, Ze'ev
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Anti-tumor immune function of NR2F6, an orphan nuclear receptor, in stromal cells
err2024-03-22
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PREAI
errKim, Hyungsoo; Feng, Yongmei; Radaeva, Marria; Sergienko, Eduard; Cherkasov, Artem; Ronai, Ze'ev A.
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Optimization of Lin28 inhibitors: A promising therapeutic approach for the suppression of cancer cell proliferation, stemness properties, and spheroid growth
err2024-03-22
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PREAI
errMatias-Barrios, Victor M.; Radaeva, Mariia; Rosellinny, Graciella; Cherkasov, Artem; Dong, Xuesen
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In silico screening of LRRK2 WDR domain inhibitors using deep docking and free energy simulations
err2024-01-01
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errOAAI
errGutkin, Evgeny; Gusev, Filipp; Gentile, Francesco; Ban, Fuqiang; Koby, S. Benjamin; Narangoda, Chamali; Isayev, Olexandr; Cherkasov, Artem; Kurnikova, Maria G.
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