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Relating GPCR Domains with Functionality: Receptor Helix-Bundle and C-Terminus Differentially Influence GRK-Specific Functions and β-Arrestin-Mediated Regulation Matthees, Edda S. F.; Haider, Raphael S.; Klement, Laura; Reichel, Mona; Blum, Nina K.; Weitzel, Verena; Truepschuch, Thimea; Ziegler, Carla; Drube, Julia; Schulz, Stefan; Hoffmann, Carsten Share Save
Key phosphorylation sites for robust β-arrestin2 binding at the MOR revisited Underwood, Owen; Fritzwanker, Sebastian; Glenn, Jaqueline; Blum, Nina Kathleen; Batista-Gondin, Arisbel; Drube, Julia; Hoffmann, Carsten; Briddon, Stephen J.; Schulz, Stefan; Canals, Meritxell Share Save
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The Concise Guide to PHARMACOLOGY 2023/24: G protein-coupled receptors Alexander, Stephen P. H.; Christopoulos, Arthur; Davenport, Anthony P.; Kelly, Eamonn; Mathie, Alistair A.; Peters, John A.; Veale, Emma L.; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Davies, Jamie A.; Abbracchio, Maria Pia; Abraham, George; Agoulnik, Alexander; Alexander, Wayne; Al-hosaini, Khaled; Back, Magnus; Baker, Jillian G.; Barnes, Nicholas M.; Bathgate, Ross; Beaulieu, Jean-Martin; Beck-Sickinger, Annette G.; Behrens, Maik; Bernstein, Kenneth E.; Bettler, Bernhard; Birdsall, Nigel J. M.; Blaho, Victoria; Boulay, Francois; Bousquet, Corinne; Brauner-Osborne, Hans; Burnstock, Geoffrey; Calo, Girolamo; Castano, Justo P.; Catt, Kevin J.; Ceruti, Stefania; Chazot, Paul; Chiang, Nan; Chini, Bice; Chun, Jerold; Cianciulli, Antonia; Civelli, Olivier; Clapp, Lucie H.; Couture, Rejean; Cox, Helen M.; Csaba, Zsolt; Dahlgren, Claes; Dent, Gordon; Douglas, Steven D.; Dournaud, Pascal; Eguchi, Satoru; Escher, Emanuel; Filardo, Edward J.; Fong, Tung; Fumagalli, Marta; Gainetdinov, Raul R.; Garelja, Michael L.; de Gasparo, Marc; Gerard, Craig; Gershengorn, Marvin; Gobeil, Fernand; Goodfriend, Theodore L.; Goudet, Cyril; Gratz, Lukas; Gregory, Karen J.; Gundlach, Andrew L.; Hamann, Jorg; Hanson, Julien; Hauger, Richard L.; Hay, Debbie L.; Heinemann, Akos; Herr, Deron; Hollenberg, Morley D.; Holliday, Nicholas D.; Horiuchi, Mastgugu; Hoyer, Daniel; Hunyady, Laszlo; Husain, Ahsan; Ijzerman, Adriaan P.; Inagami, Tadashi; Jacobson, Kenneth A.; Jensen, Robert T.; Jockers, Ralf; Jonnalagadda, Deepa; Karnik, Sadashiva; Kaupmann, Klemens; Kemp, Jacqueline; Kennedy, Charles; Kihara, Yasuyuki; Kitazawa, Takio; Kozielewicz, Pawel; Kreienkamp, Hans-Juergen; Kukkonen, Jyrki P.; Langenhan, Tobias; Larhammar, Dan; Leach, Katie; Lecca, Davide; Lee, John D.; Leeman, Susan E.; Leprince, Jerome; Li, Xaria X.; Lolait, Stephen J.; Lupp, Amelie; Macrae, Robyn; Maguire, Janet; Malfacini, Davide; Mazella, Jean; McArdle, Craig A.; Melmed, Shlomo; Michel, Martin C.; Miller, Laurence J.; Mitolo, Vincenzo; Mouillac, Bernard; Mueller, Christa E.; Murphy, Philip M.; Nahon, Jean-Louis; Ngo, Tony; Norel, Xavier; Nyimanu, Duuamene; O'Carroll, Anne-Marie; Offermanns, Stefan; Panaro, Maria Antonietta; Parmentier, Marc; Pertwee, Roger G.; Pin, Jean-Philippe; Prossnitz, Eric R.; Quinn, Mark; Ramachandran, Rithwik; Ray, Manisha; Reinscheid, Rainer K.; Rondard, Philippe; Rovati, G. Enrico; Ruzza, Chiara; Sanger, Gareth J.; Schoeneberg, Torsten; Schulte, Gunnar; Schulz, Stefan; Segaloff, Deborah L.; Serhan, Charles N.; Singh, Khuraijam Dhanachandra; Smith, Craig M.; Stoddart, Leigh A.; Sugimoto, Yukihiko; Summers, Roger; Tan, Valerie P.; Thal, David; Thomas, Walter (Wally); Timmermans, Pieter B. M. W. M.; Tirupula, Kalyan; Toll, Lawrence; Tulipano, Giovanni; Unal, Hamiyet; Unger, Thomas; Valant, Celine; Vanderheyden, Patrick; Vaudry, David; Vaudry, Hubert; Vilardaga, Jean-Pierre; Walker, Christopher S.; Wang, Ji Ming; Ward, Donald T.; Wester, Hans-Juergen; Willars, Gary B.; Williams, Tom Lloyd; Woodruff, Trent M.; Yao, Chengcan; Ye, Richard D. Share Save
Phosphorylation bar-coding of free fatty acid receptor 2 is generated in a tissue-specific manner Barki, Natasja; Jenkins, Laura; Marsango, Sara; Dedeo, Domonkos; Bolognini, Daniele; Dwomoh, Louis; Abdelmalik, Aisha M.; Nilsen, Margaret; Stoffels, Manon; Nagel, Falko; Schulz, Stefan; Tobin, Andrew B.; Milligan, Graeme Share Save
Reply to: How carvedilol does not activate β2-adrenoceptors Kostenis, Evi; Gomeza, Jesus; Miess-Tanneberg, Elke; Blum, Nina Kathleen; Benkel, Tobias; Chevigne, Andy; Hoffmann, Carsten; Kolb, Peter; Nikolaev, Viacheslav; Waldhoer, Maria; Szpakowska, Martyna; Inoue, Asuka; Schulz, Stefan Share Save
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The NPXXY Motif Regulates β-Arrestin Recruitment by the CB1 Cannabinoid Receptor Leo, Luciana M.; Al-Zoubi, Rufaida; Hurst, Dow P.; Stephan, Anna P.; Zhao, Pingwei; Tilley, Douglas G.; Miess, Elke; Schulz, Stefan; Abood, Mary E.; Reggio, Patricia H. Share Save
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A Switch of G Protein-Coupled Receptor Binding Preference from Phosphoinositide 3-Kinase (PI3K)-p85 to Filamin A Negatively Controls the PI3K Pathway Najib, Souad; Saint-Laurent, Nathalie; Esteve, Jean-Pierre; Schulz, Stefan; Boutet-Robinet, Elisa; Fourmy, Daniel; Laettig, Jens; Mollereau, Catherine; Pyronnet, Stephane; Susini, Christiane; Bousquet, Corinne Share Save
How Carvedilol activates β2-adrenoceptors Benkel, Tobias; Zimmermann, Mirjam; Zeiner, Julian; Bravo, Sergi; Merten, Nicole; Lim, Victor Jun Yu; Matthees, Edda Sofie Fabienne; Drube, Julia; Miess-Tanneberg, Elke; Malan, Daniela; Szpakowska, Martyna; Monteleone, Stefania; Grimes, Jak; Koszegi, Zsombor; Lanoiselee, Yann; O'Brien, Shannon; Pavlaki, Nikoleta; Dobberstein, Nadine; Inoue, Asuka; Nikolaev, Viacheslav; Calebiro, Davide; Chevigne, Andy; Sasse, Philipp; Schulz, Stefan; Hoffmann, Carsten; Kolb, Peter; Waldhoer, Maria; Simon, Katharina; Gomeza, Jesus; Kostenis, Evi Share Save
A bead-based GPCR phosphorylation immunoassay for high-throughput ligand profiling and GRK inhibitor screening Kaufmann, Johanna; Blum, Nina Kathleen; Nagel, Falko; Schuler, Anna; Drube, Julia; Degenhart, Carsten; Engel, Julian; Eickhoff, Jan Eicke; Dasgupta, Pooja; Fritzwanker, Sebastian; Guastadisegni, Maria; Schulte, Clemens; Miess-Tanneberg, Elke; Maric, Hans Michael; Spetea, Mariana; Kliewer, Andrea; Baumann, Matthias; Klebl, Bert; Reinscheid, Rainer K.; Hoffmann, Carsten; Schulz, Stefan Share Save
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