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SaveFDW028, a novel FUT8 inhibitor, impels lysosomal proteolysis of B7-H3 via chaperone-mediated autophagy pathway and exhibits potent efficacy against metastatic colorectal cancer
Wang, Mengmeng; Zhang, Zhoudong; Chen, Mengxi; Lv, Yixin; Tian, Sheng; Meng, Fanyi; Zhang, Yawen; Guo, Xuqin; Chen, Yinshuang; Yang, Man; Li, Jiawei; Qiu, Tian; Xu, Fang; Li, Zhi; Zhang, Qi; Yang, Jie; Sun, Jing; Zhang, Hongjian; Zhang, Haiyang; Li, Huanqiu; Wang, Weipeng
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SaveDiscovery of Selective P2Y6R Antagonists with High Affinity and In Vivo Efficacy for Inflammatory Disease Therapy
Zhu, Yifan; Zhou, Mengze; Cheng, Xiangyu; Wang, Hui; Li, Yehong; Guo, Yueyue; Wang, Yaxuan; Tian, Sheng; Mao, Tianqi; Zhang, Zhoudong; Li, Duxin; Hu, Qinghua; Li, Huanqiu
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