Markus A. Queisser - Publications, H-index & Citations

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Markus A. Queisser

GSK

15H-index

37Paper Count

2.7KCitation Count

Published Papers 17

Publication Date

A Systematic Direct-to-Biology Approach Identified Potent Cereblon HaloPROTACs

ACS Chemical Biology

IF3.8

2026-06-29

PREAI

Rebecca Stevens; Kwok-Ho Chan; Alice Moore; Sam Hardie; Glenn A. Burley; Jennifer J. Knickelbine; Kristin M. Riching; Agnieszka Konopacka; Markus A. Queisser; Afjal H. Miah

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Identification of an allosteric site on the E3 ligase adapter cereblon

Nature

IF48.5

2026-01-21

PREAI

Vanessa N. Dippon; Zeba Rizvi; Anthony E. Choudhry; Chun-wa Chung; Ibrahim F. Alkuraya; Wenqing Xu; Xavier B. Tao; Anthony J. Jurewicz; Jessica L. Schneck; Wenqian Chen; Nicole M. Curnutt; Farah Kabir; Kwok-Ho Chan; Markus A. Queisser; Caterina Musetti; Han Dai; Gabriel C. Lander; Andrew B. Benowitz; Christina M. Woo

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Orthogonal IMiD-Degron Pairs Induce Selective Protein Degradation in Cells

ACS Chemical Biology

IF3.8

2025-11-02

OAAI

Patrick J. Brennan; Rebecca E. Saunders; Mary Spanou; Sarah E. Singleton; Marta Serafini; Liang Sun; Guillaume P. Heger; Agnieszka Konopacka; Ryan D. Beveridge; C. Cameron Taylor; Peter DePaola IV; Laurie Gordon; Shenaz B. Bunally; Aurore Saudemont; Andrew B. Benowitz; Carlos Martinez-Fleites; Danielle L. Schmitt; Robert Damoiseaux; Markus A. Queisser; Heeseon An; Charlotte M. Deane; Michael M. Hann; Lewis L. Brayshaw; Stuart J. Conway

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Optimization and Evaluation of Complementary Degrader Discovery Assays for Application in Screening

ACS Pharmacology & Translational Science

IF3.7

2025-07-20

OAAI

Johanna Huchting; Arjen Weller; Moyra Schweizer; Mona Brandt; Jan Heering; Maria Kuzikov; Markus Wolf; Jeanette Reinshagen; Markus A. Queisser; Philip Gribbon; Andrea Zaliani; Ole Pless; Aimo Kannt

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Structure-Guided Design and Optimization of Covalent VHL-Targeted Sulfonyl Fluoride PROTACs

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2024-03-13

OAAI

Shah, Rishi R.; De Vita, Elena; Sathyamurthi, Preethi S.; Conole, Daniel; Zhang, Xinyue; Fellows, Elliot; Dickinson, Eleanor R.; Fleites, Carlos M.; Queisser, Markus A.; Harling, John D.; Tate, Edward W.

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Antibody-Proteolysis Targeting Chimera Conjugate Enables Selective Degradation of Receptor-Interacting Serine/Threonine-Protein Kinase 2 in HER2+Cell Lines

BIOCONJUGATE CHEMISTRY

IF3.9

2023-11-02

OAAI

Chan, Karina; Sathyamurthi, Preethi Soundarya; Queisser, Markus A.; Mullin, Michael; Shrives, Harry; Coe, Diane M.; Burley, Glenn A.

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Identification of KLHDC2 as an efficient proximity-induced degrader of K-RAS, STK33,β-catenin, and FoxP3

CELL CHEMICAL BIOLOGY

IF7.2

2023-10-01

OAAI

Roth, Sascha; Kocaturk, Nur Mehpare; Sathyamurthi, Preethi S.; Carton, Bill; Watt, Matthew; Macartney, Thomas J.; Chan, Kwok-Ho; Isidro-Llobet, Albert; Konopacka, Agnieszka; Queisser, Markus A.; Sapkota, Gopal P.

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Discovery and Characterisation of Highly Cooperative FAK-Degrading PROTACs

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

IF16.9

2021-09-17

PREAI

Law, Robert P.; Nunes, Joao; Chung, Chun-wa; Bantscheff, Marcus; Buda, Karol; Dai, Han; Evans, John P.; Flinders, Adam; Klimaszewska, Diana; Lewis, Antonia J.; Muelbaier, Marcel; Scott-Stevens, Paul; Stacey, Peter; Tame, Christopher J.; Watt, Gillian F.; Zinn, Nico; Queisser, Markus A.; Harling, John D.; Benowitz, Andrew B.

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The PROTACtable genome

NATURE REVIEWS DRUG DISCOVERY

IF101.8

2021-07-20

143

PREAI

Schneider, Melanie; Radoux, Chris J.; Hercules, Andrew; Ochoa, David; Dunham, Ian; Zalmas, Lykourgos-Panagiotis; Hessler, Gerhard; Ruf, Sven; Shanmugasundaram, Veerabahu; Hann, Michael M.; Thomas, Pam J.; Queisser, Markus A.; Benowitz, Andrew B.; Brown, Kris; Leach, Andrew R.

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Targeting Endogenous K-RAS for Degradation through the Affinity-Directed Protein Missile System

CELL CHEMICAL BIOLOGY

IF7.2

2020-09-01

OAAI

Roth, Sascha; Macartney, Thomas J.; Konopacka, Agnieszka; Chan, Kwok-Ho; Zhou, Houjiang; Queisser, Markus A.; Sapkota, Gopal P.

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Structural Insights into PROTAC-Mediated Degradation of BcI-xL

ACS CHEMICAL BIOLOGY

IF3.8

2020-07-22

PREAI

Chung, Chun-wa; Dai, Han; Fernandez, Esther; Tinworth, Christopher P.; Churcher, Ian; Cryan, Jenni; Denyer, Jane; Harling, John D.; Konopacka, Agnieszka; Queisser, Markus A.; Tame, Christopher J.; Watt, Gillian; Jiang, Fan; Qian, Dongming; Benowitz, Andrew B.

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HIF and HOIL-1L-mediated PKCζ degradation stabilizes plasma membrane Na,K-ATPase to protect against hypoxia-induced lung injury

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

IF9.1

2017-11-06

OAAI

Magnani, Natalia D.; Dada, Laura A.; Queisser, Markus A.; Brazee, Patricia L.; Welch, Lynn C.; Anekalla, Kishore R.; Zhou, Guofei; Vagin, Olga; Misharin, Alexander V.; Budinger, G. R. Scott; Iwai, Kazuhiro; Ciechanover, Aaron J.; Sznajder, Jacob I.

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Conserved cytoplasmic domains promote Hrd1 ubiquitin ligase complex formation for ER-associated degradation (ERAD)

JOURNAL OF CELL SCIENCE

IF3.6

2017-10-01

OAAI

Schulz, Jasmin; Avci, Donem; Queisser, Markus A.; Gutschmidt, Aljona; Dreher, Lena-Sophie; Fenech, Emma J.; Volkmar, Norbert; Hayashi, Yuki; Hoppe, Thorsten; Christianson, John C.

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HOIL-1L Functions as the PKCζ Ubiquitin Ligase to Promote Lung Tumor Growth

AMERICAN JOURNAL OF RESPIRATORY AND CRITICAL CARE MEDICINE

IF19.4

2014-09-15

OAAI

Queisser, Markus A.; Dada, Laura A.; Deiss-Yehiely, Nimrod; Angulo, Martin; Zhou, Guofei; Kouri, Fotini M.; Knab, Lawrence M.; Liu, Jing; Stegh, Alexander H.; DeCamp, Malcolm M.; Budinger, G. R. Scott; Chandel, Navdeep S.; Ciechanover, Aaron; Lwai, Kazuhiro; Sznajder, Jacob I.

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Hyperglycemia Impairs Proteasome Function by Methylglyoxal

DIABETES

IF7.5

2009-12-15

171

OAAI

Queisser, Markus A.; Yao, Dachun; Geisler, Sven; Hammes, Hans-Peter; Lochnit, Guenter; Schleicher, Erwin D.; Brownlee, Michael; Preissner, Klaus T.

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Loss of RAGE in pulmonary fibrosis -: Molecular relations to functional changes in pulmonary cell types

AMERICAN JOURNAL OF RESPIRATORY CELL AND MOLECULAR BIOLOGY

IF5.3